ZA200410102B - Use of nefopam for the treatment of nausea or emesis - Google Patents
Use of nefopam for the treatment of nausea or emesis Download PDFInfo
- Publication number
- ZA200410102B ZA200410102B ZA200410102A ZA200410102A ZA200410102B ZA 200410102 B ZA200410102 B ZA 200410102B ZA 200410102 A ZA200410102 A ZA 200410102A ZA 200410102 A ZA200410102 A ZA 200410102A ZA 200410102 B ZA200410102 B ZA 200410102B
- Authority
- ZA
- South Africa
- Prior art keywords
- use according
- condition
- nefopam
- induced
- emesis
- Prior art date
Links
- RGPDEAGGEXEMMM-UHFFFAOYSA-N Nefopam Chemical compound C12=CC=CC=C2CN(C)CCOC1C1=CC=CC=C1 RGPDEAGGEXEMMM-UHFFFAOYSA-N 0.000 title claims description 24
- 229960000751 nefopam Drugs 0.000 title claims description 23
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- 206010028813 Nausea Diseases 0.000 title claims description 4
- 230000008693 nausea Effects 0.000 title claims description 4
- LNEPOXFFQSENCJ-UHFFFAOYSA-N haloperidol Chemical compound C1CC(O)(C=2C=CC(Cl)=CC=2)CCN1CCCC(=O)C1=CC=C(F)C=C1 LNEPOXFFQSENCJ-UHFFFAOYSA-N 0.000 claims description 6
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- YEHCICAEULNIGD-MZMPZRCHSA-N pergolide Chemical compound C1=CC([C@H]2C[C@@H](CSC)CN([C@@H]2C2)CCC)=C3C2=CNC3=C1 YEHCICAEULNIGD-MZMPZRCHSA-N 0.000 description 1
- 230000003389 potentiating effect Effects 0.000 description 1
- 238000002360 preparation method Methods 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/5545—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having eight-membered rings not containing additional condensed or non-condensed nitrogen-containing 3-7 membered rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0213869.1A GB0213869D0 (en) | 2002-06-17 | 2002-06-17 | The treatment of pain |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200410102B true ZA200410102B (en) | 2006-07-26 |
Family
ID=9938718
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200410102A ZA200410102B (en) | 2002-06-17 | 2004-12-14 | Use of nefopam for the treatment of nausea or emesis |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US20060063753A1 (es) |
| EP (2) | EP1513518A1 (es) |
| JP (2) | JP2005533784A (es) |
| CN (1) | CN100482221C (es) |
| AU (2) | AU2003240113B2 (es) |
| BR (1) | BR0311874A (es) |
| CA (2) | CA2489306A1 (es) |
| GB (1) | GB0213869D0 (es) |
| IL (1) | IL165773A0 (es) |
| MX (1) | MXPA04012826A (es) |
| NO (1) | NO20045496L (es) |
| NZ (1) | NZ537197A (es) |
| PL (1) | PL374418A1 (es) |
| WO (2) | WO2003105833A1 (es) |
| ZA (1) | ZA200410102B (es) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0330049D0 (en) * | 2003-12-24 | 2004-02-04 | Arakis Ltd | The treatment of neuropathic pain conditions |
| GB0408864D0 (en) * | 2004-04-21 | 2004-05-26 | Arakis Ltd | Novel benzoxazocines |
| GB0515703D0 (en) * | 2005-07-29 | 2005-09-07 | Arakis Ltd | Therapeutic use of nefopam |
| CA2962043A1 (en) * | 2007-06-22 | 2008-12-31 | Hydra Biosciences, Inc. | Xanthine derivatives for the treatment of diseases mediated by trpa1 |
| GB0721013D0 (en) | 2007-10-25 | 2007-12-05 | Sosei R & D Ltd | New Salts |
| CN102046170B (zh) | 2008-05-27 | 2012-11-28 | 墨尔本大学 | 治疗患有咽鼓管功能障碍的哺乳动物的方法 |
| US20110092493A1 (en) * | 2008-09-24 | 2011-04-21 | Clark Levi | Dose-controlled transdermal promethazine compositions and methods of use |
| RU2608458C2 (ru) * | 2009-05-20 | 2017-01-18 | Инсерм (Энститю Насьональ Де Ля Сантэ Э Де Ля Решерш Медикаль) | Антагонисты серотониновых 5-нт3-рецепторов для применения при лечении вестибулярных нарушений с повреждениями |
| EP2512468B1 (en) * | 2009-12-15 | 2016-08-24 | The Hospital for Sick Children | METHOD OF TREATING SCARS AND ß-CATENIN-MEDIATED DISORDERS USING NEFOPAM COMPOUNDS |
| EP4335508A3 (en) | 2016-04-14 | 2024-07-10 | Sensorion | (+)-azasetron for use in the treatment of ear disorders |
| US10736905B1 (en) | 2016-09-09 | 2020-08-11 | Shahin Fatholahi | Nefopam dosage forms and methods of treatment |
| US10736874B1 (en) | 2017-09-08 | 2020-08-11 | Shahin Fatholahi | Methods for treating pain associated with sickle cell disease |
| US11446311B2 (en) | 2017-09-08 | 2022-09-20 | Shahin Fatholahi | Methods for treating pain associated with sickle cell disease |
| RS65140B1 (sr) * | 2019-05-06 | 2024-02-29 | Chemcom Sa | Upotreba kompozicije protiv neprijatnih mirisa i povezani postupak |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2338753C (en) * | 1998-07-24 | 2006-11-21 | Jago Research Ag | Medicinal aerosol formulations |
| US20020013331A1 (en) * | 2000-06-26 | 2002-01-31 | Williams Robert O. | Methods and compositions for treating pain of the mucous membrane |
-
2002
- 2002-06-17 GB GBGB0213869.1A patent/GB0213869D0/en not_active Ceased
-
2003
- 2003-06-17 BR BR0311874-6A patent/BR0311874A/pt not_active IP Right Cessation
- 2003-06-17 JP JP2004512736A patent/JP2005533784A/ja active Pending
- 2003-06-17 EP EP03740737A patent/EP1513518A1/en not_active Withdrawn
- 2003-06-17 US US10/517,881 patent/US20060063753A1/en not_active Abandoned
- 2003-06-17 JP JP2004512737A patent/JP2005531612A/ja active Pending
- 2003-06-17 PL PL03374418A patent/PL374418A1/xx not_active Application Discontinuation
- 2003-06-17 CA CA002489306A patent/CA2489306A1/en not_active Abandoned
- 2003-06-17 US US10/517,882 patent/US20060040905A1/en not_active Abandoned
- 2003-06-17 WO PCT/GB2003/002618 patent/WO2003105833A1/en active Application Filing
- 2003-06-17 MX MXPA04012826A patent/MXPA04012826A/es unknown
- 2003-06-17 CA CA002489315A patent/CA2489315A1/en not_active Abandoned
- 2003-06-17 NZ NZ537197A patent/NZ537197A/en unknown
- 2003-06-17 AU AU2003240113A patent/AU2003240113B2/en not_active Ceased
- 2003-06-17 AU AU2003277077A patent/AU2003277077B2/en not_active Ceased
- 2003-06-17 EP EP03732727A patent/EP1513517A1/en not_active Withdrawn
- 2003-06-17 CN CNB038167050A patent/CN100482221C/zh not_active Expired - Fee Related
- 2003-06-17 WO PCT/GB2003/002586 patent/WO2003105832A1/en active Application Filing
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2004
- 2004-12-14 IL IL16577304A patent/IL165773A0/xx unknown
- 2004-12-14 ZA ZA200410102A patent/ZA200410102B/en unknown
- 2004-12-16 NO NO20045496A patent/NO20045496L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| BR0311874A (pt) | 2005-05-10 |
| AU2003277077B2 (en) | 2006-11-02 |
| GB0213869D0 (en) | 2002-07-31 |
| CN100482221C (zh) | 2009-04-29 |
| CA2489315A1 (en) | 2003-12-24 |
| WO2003105833A1 (en) | 2003-12-24 |
| PL374418A1 (en) | 2005-10-17 |
| EP1513518A1 (en) | 2005-03-16 |
| AU2003240113B2 (en) | 2006-11-16 |
| CN1668294A (zh) | 2005-09-14 |
| IL165773A0 (en) | 2006-01-15 |
| AU2003277077A1 (en) | 2003-12-31 |
| CA2489306A1 (en) | 2003-12-24 |
| US20060040905A1 (en) | 2006-02-23 |
| US20060063753A1 (en) | 2006-03-23 |
| MXPA04012826A (es) | 2005-03-31 |
| AU2003240113A1 (en) | 2003-12-31 |
| NO20045496L (no) | 2005-01-12 |
| WO2003105832A1 (en) | 2003-12-24 |
| EP1513517A1 (en) | 2005-03-16 |
| NZ537197A (en) | 2007-10-26 |
| JP2005531612A (ja) | 2005-10-20 |
| JP2005533784A (ja) | 2005-11-10 |
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