YU87101A - Derivati benzena, postupak za njihovo dobijanje i farmaceutski preparati koji ih sadrže - Google Patents

Derivati benzena, postupak za njihovo dobijanje i farmaceutski preparati koji ih sadrže

Info

Publication number
YU87101A
YU87101A YU87101A YUP87101A YU87101A YU 87101 A YU87101 A YU 87101A YU 87101 A YU87101 A YU 87101A YU P87101 A YUP87101 A YU P87101A YU 87101 A YU87101 A YU 87101A
Authority
YU
Yugoslavia
Prior art keywords
preparation
pharmaceutical compositions
benzene derivatives
same
compositions containg
Prior art date
Application number
YU87101A
Other languages
English (en)
Inventor
Robert Boigegrain
Bernard Bourrie
Martine Bourrie
Pierre Casellas
Jean Marc Herbert
Pierre Lair
Dino Nisato
Raymond Paul
Jean Claude Vernieres
Original Assignee
Sanofi-Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi-Synthelabo filed Critical Sanofi-Synthelabo
Publication of YU87101A publication Critical patent/YU87101A/sh
Publication of RS49998B publication Critical patent/RS49998B/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/33—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C07C211/34—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton
    • C07C211/35—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton containing only non-condensed rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/33—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C07C211/39—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton
    • C07C211/40—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton containing only non-condensed rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/56—Ring systems containing bridged rings
    • C07C2603/58—Ring systems containing bridged rings containing three rings
    • C07C2603/70—Ring systems containing bridged rings containing three rings containing only six-membered rings
    • C07C2603/74—Adamantanes

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Transplantation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrane Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Pronalazak se odnosi na jedinjenja formule (I), gde A, X, Y, n, R1, R2 i R3 su kao što je definisano u zathevu 1. Pomenuta jedinjenja se specifično vezuju na sigma receptore naročito one perifernog nervnog sistema.
YUP-871/01A 1999-06-11 2000-06-08 Derivati benzena, postupak za njihovo dobijanje i farmaceutski preparati koji ih sadrže RS49998B (sr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9907396A FR2794742B1 (fr) 1999-06-11 1999-06-11 Nouveaux derives du benzene, un procede pour leur preparation et les compositions pharmaceutiques les contenant

Publications (2)

Publication Number Publication Date
YU87101A true YU87101A (sh) 2004-07-15
RS49998B RS49998B (sr) 2008-09-29

Family

ID=9546664

Country Status (33)

Country Link
US (1) US6482986B1 (sh)
EP (1) EP1192122B1 (sh)
JP (1) JP4711579B2 (sh)
KR (1) KR100668581B1 (sh)
CN (1) CN1210250C (sh)
AR (1) AR033793A1 (sh)
AT (1) ATE252542T1 (sh)
AU (1) AU768420B2 (sh)
BR (1) BR0011738A (sh)
CA (1) CA2374631C (sh)
CO (1) CO5180554A1 (sh)
CZ (1) CZ299659B6 (sh)
DE (1) DE60006113T2 (sh)
DK (1) DK1192122T3 (sh)
ES (1) ES2208345T3 (sh)
FR (1) FR2794742B1 (sh)
HK (1) HK1042891B (sh)
HU (1) HU228683B1 (sh)
IL (1) IL146545A0 (sh)
MX (1) MXPA01012783A (sh)
NO (1) NO327778B1 (sh)
NZ (1) NZ515529A (sh)
PL (1) PL196491B1 (sh)
PT (1) PT1192122E (sh)
RS (1) RS49998B (sh)
RU (1) RU2248964C2 (sh)
SI (1) SI1192122T1 (sh)
SK (1) SK286390B6 (sh)
TW (1) TWI279398B (sh)
UA (1) UA71959C2 (sh)
UY (1) UY26199A1 (sh)
WO (1) WO2000076953A1 (sh)
ZA (1) ZA200109486B (sh)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10110750A1 (de) * 2001-03-07 2002-09-12 Bayer Ag Neuartige Aminodicarbonsäurederivate mit pharmazeutischen Eigenschaften
GB2410947B (en) * 2004-02-11 2008-09-17 Cambridge Lab Ltd Pharmaceutical compounds
CA2571710A1 (en) 2004-06-24 2006-11-02 Nicholas Valiante Small molecule immunopotentiators and assays for their detection
EP1634598A1 (en) * 2004-09-07 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Use of piperazine derivatives and analogues for the manufacture of a medicament for the prophylaxis and/or treatment of disorders of food ingestion
EP2479814B1 (en) 2005-03-28 2015-07-22 Semiconductor Energy Laboratory Co, Ltd. Light emitting device comprising a carbazole-anthracene derivative
FR2887454B1 (fr) * 2005-06-28 2009-06-05 Sanofi Aventis Sa Combinaisons antitumorales contenant des derives du taxane et des sigma ligands
GB0514501D0 (en) * 2005-07-14 2005-08-24 Cambridge Lab Ireland Ltd Pharmaceutical compounds
GB0516168D0 (en) * 2005-08-05 2005-09-14 Cambridge Lab Ireland Ltd Pharmaceutical compounds
US7731377B2 (en) * 2006-03-21 2010-06-08 Semiconductor Energy Laboratory Co., Ltd. Backlight device and display device
WO2008026614A1 (en) * 2006-08-30 2008-03-06 Semiconductor Energy Laboratory Co., Ltd. Method for synthesizing anthracene derivative and anthracene derivative, light emitting element, light emitting device, electronic device
GR1005865B (el) * 2007-01-17 2008-04-07 Anavex Life Sciences Corp. Νεοι συνδετες των σιγμα υποδοχεων με αντι-αποπτωτικες και/η προ-αποπτωτικες ιδιοτητες επι των κυτταρικων βιοχημικων μηχανισμων, με νευρο-προστατευτικη, αντικαρκινικη, αντι-μεταστατικη και αντι- αντι-(χρονιο)φλεγμονικη δραση.
US7723722B2 (en) * 2007-03-23 2010-05-25 Semiconductor Energy Laboratory Co., Ltd. Organic compound, anthracene derivative, and light-emitting element, light-emitting device, and electronic device using anthracene derivative
FR2915994B1 (fr) * 2007-05-11 2009-07-03 Galderma Res & Dev Procede de synthese de l'acide (z)-3-[2-butoxy-3'-(3-heptyl-1-methyl-ureido)-biphenyl-4-yl] -2-methoxy-acrylique.
US20080286445A1 (en) * 2007-05-17 2008-11-20 Semiconductor Energy Laboratory Co., Ltd. Composition, and method of fabricating light-emitting element
GB0810857D0 (en) * 2008-06-13 2008-07-23 Cambridge Lab Ireland Ltd Pharmaceutical compounds
CN102089282A (zh) * 2008-07-08 2011-06-08 株式会社半导体能源研究所 咔唑衍生物、发光元件用材料、发光元件以及发光装置
US20110053866A1 (en) * 2008-08-12 2011-03-03 Biovail Laboratories International (Barbados) S.R.L. Pharmaceutical compositions
GB2462611A (en) * 2008-08-12 2010-02-17 Cambridge Lab Pharmaceutical composition comprising tetrabenazine
GB2463451A (en) * 2008-09-08 2010-03-17 Cambridge Lab 3, 11b cis-dihydrotetrabenazine compounds for use in the treatment of dementia
GB2463452A (en) * 2008-09-08 2010-03-17 Cambridge Lab Desmethyl derivatives of tetrabenazine and pharmaceutical compositions thereof
GB2463283A (en) * 2008-09-08 2010-03-10 Cambridge Lab 3,11b-cis-dihydrotetrabenazine for use in treating asthma
KR101661328B1 (ko) * 2008-09-19 2016-09-29 가부시키가이샤 한도오따이 에네루기 켄큐쇼 카르바졸 유도체 및 그 제조 방법
US8349898B2 (en) * 2008-11-18 2013-01-08 Wisconsin Alumni Research Foundation Sigma-1 receptor ligands and methods of use
GR1006794B (el) * 2009-02-26 2010-06-04 Αλεξανδρος Βαμβακιδης Προσδετες των σιγμα υποδοχεων, αντι-αποπτωτικες και προ-αποπτωτικες ιδιοτητες επι των κυτταρικων μηχανισμων, και με πρωτοτυπη κυτταρο-προστατευτικη αλλα και αντικαρκινικη δραση
JP6492432B2 (ja) * 2013-07-09 2019-04-03 東ソー株式会社 アダマンチル基を有する環状アジン化合物、その製造方法、及びそれを構成成分とする有機電界発光素子
KR20170101128A (ko) 2016-02-26 2017-09-05 가부시키가이샤 한도오따이 에네루기 켄큐쇼 유기 화합물, 발광 소자, 발광 장치, 전자 기기, 및 조명 장치
CA3031818A1 (en) 2016-07-27 2018-02-01 Case Western Reserve University Compounds and methods of promoting myelination
WO2019126702A1 (en) 2017-12-22 2019-06-27 Case Western Reserve University Compounds for promoting myelination
WO2019126759A1 (en) * 2017-12-22 2019-06-27 Convelo Therapeutics, Inc. Compounds and methods of promoting myelination
CA3229664A1 (en) * 2021-08-23 2023-03-02 William A. DONALDSON Synthesis and evaluation of novel (4-hydroxyphenyl) substituted carbocycles as potent and selective estrogen receptor beta agonists

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4104383A (en) * 1973-11-02 1978-08-01 C M Industries Derivatives of phenylpropenylamine
FR2641276B1 (fr) 1988-12-30 1991-07-12 Sanofi Sa Derives du benzene, leur preparation et les compositions pharmaceutiques en contenant
WO1991009594A1 (en) * 1989-12-28 1991-07-11 Virginia Commonwealth University Sigma receptor ligands and the use thereof
ZA909902B (en) * 1989-12-21 1991-10-30 Himont Inc Graft copolymers of polyolefins and a method of producing same
FR2663328B1 (fr) 1990-06-14 1994-08-05 Sanofi Sa Derives d'hexahydroazepines, un procede pour leur preparation et compositions pharmaceutiques les contenant.
CA2111957A1 (en) * 1991-06-27 1993-01-07 Richard A. Glennon Sigma receptor ligands and the use thereof
US5449639A (en) 1994-10-24 1995-09-12 Taiwan Semiconductor Manufacturing Company Ltd. Disposable metal anti-reflection coating process used together with metal dry/wet etch
FR2751645B1 (fr) * 1996-07-29 1998-12-24 Sanofi Sa Amines pour la fabrication de medicaments destines a empecher la proliferation de cellules tumorales

Also Published As

Publication number Publication date
TWI279398B (en) 2007-04-21
NZ515529A (en) 2004-01-30
DE60006113T2 (de) 2004-07-15
CA2374631C (en) 2010-10-19
WO2000076953A1 (fr) 2000-12-21
KR20020009632A (ko) 2002-02-01
RU2248964C2 (ru) 2005-03-27
PL196491B1 (pl) 2008-01-31
PL352742A1 (en) 2003-09-08
AU768420B2 (en) 2003-12-11
CO5180554A1 (es) 2002-07-30
ES2208345T3 (es) 2004-06-16
ATE252542T1 (de) 2003-11-15
MXPA01012783A (es) 2002-09-18
SK286390B6 (sk) 2008-09-05
HUP0201953A3 (en) 2006-03-28
HUP0201953A2 (hu) 2002-12-28
AR033793A1 (es) 2004-01-07
IL146545A0 (en) 2002-07-25
DK1192122T3 (da) 2004-03-01
AU5539600A (en) 2001-01-02
HK1042891A1 (en) 2002-08-30
HK1042891B (zh) 2004-04-08
BR0011738A (pt) 2002-03-05
CN1210250C (zh) 2005-07-13
PT1192122E (pt) 2004-03-31
HU228683B1 (en) 2013-05-28
CN1355782A (zh) 2002-06-26
FR2794742A1 (fr) 2000-12-15
SI1192122T1 (en) 2004-04-30
CZ20014443A3 (cs) 2002-05-15
EP1192122B1 (fr) 2003-10-22
CA2374631A1 (en) 2000-12-21
EP1192122A1 (fr) 2002-04-03
CZ299659B6 (cs) 2008-10-08
UA71959C2 (en) 2005-01-17
RS49998B (sr) 2008-09-29
UY26199A1 (es) 2001-01-31
DE60006113D1 (de) 2003-11-27
JP2003502306A (ja) 2003-01-21
JP4711579B2 (ja) 2011-06-29
NO20016038L (no) 2002-02-11
NO327778B1 (no) 2009-09-21
FR2794742B1 (fr) 2005-06-03
US6482986B1 (en) 2002-11-19
NO20016038D0 (no) 2001-12-10
SK18062001A3 (sk) 2002-05-09
KR100668581B1 (ko) 2007-01-17
ZA200109486B (en) 2002-11-18

Similar Documents

Publication Publication Date Title
YU87101A (sh) Derivati benzena, postupak za njihovo dobijanje i farmaceutski preparati koji ih sadrže
YU11997A (sh) Laktamski derivati i njihove farmaceutske kompozicije
MEP45308A (en) [1,8]naphthyridin-2-ones and related compounds for the treatment of schizophrenia
ATE339408T1 (de) Terphenylderivate, deren herstellung und zusammensetzungen, die diese enthalten
RS50035B (sr) Farmaceutska kompozicija koja sadrži fenofibrat i postupak za njeno dobijanje
BRPI0108395B8 (pt) derivados de pirrolopirimidinona, processos de preparação e uso
AP9801169A0 (en) N-hydroxy-B-sulfonyl propionamide derivatives.
DE60204452D1 (de) Pyrazolo[1,5]pyridinderivate
DE60129697D1 (de) Kondensierte azepinderivate und ihre verwendung als als antidiuretisches mittel
IL151172A0 (en) Amine derivatives, their preparation and use as bax modulators
ES2140961T3 (es) Nuevos derivados de 19-nor-pregneno.
RU94038064A (ru) Производные пиперазина и пиперидина, их применение в качестве противопсихотических средств, способ их получения фармацевтическая композиция
ATE300541T1 (de) Pyrazolopyridinderivate
ES2174298T3 (es) Derivados de aminotiazol, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.
ES2107284T3 (es) Nuevas n-piridil-carboxamidas, su procedimiento de preparacion y composiciones farmaceuticas que las contienen.
NO20020282L (no) Nytt difenyl-piperidinderivat
RS50046B (sr) Farmaceutske kompozicije tizoksanida i nitazoksanida
MA28286A1 (fr) Dérivés de 1-N-phenyl-amino-1H-imidazole et compositions pharmaceutiques les contenant
YU44301A (sh) 5ht1 antagonisti za antidepresantnu terapiju
TR200200125T2 (tr) Yeni aminotiyazol türevleri, bunların hazırlanması ve bunları içeren farmasötik kompozisyonlar.
TR200000153T2 (tr) İl-5 inhibite eden 6-azaurasil türevleri.
RU94038042A (ru) Производные гексагидроазепинов, фармацевтическая композиция на их основе и антипсихотропный агент
DE69624308D1 (de) Bernsteinsäurederivate als abbaubare Chelatbildner, ihre Verwendungen und Zusammensetzungen
BR0009470A (pt) Tablete detergente perfumado
BRPI0415034A (pt) derivados de aminopiridina como inibidores de não-sintase induzìveis