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Application filed by Pfizer Inc.filedCriticalPfizer Inc.
Priority to YU19691ApriorityCriticalpatent/YU48204B/en
Publication of YU19691ApublicationCriticalpatent/YU19691A/en
Publication of YU48204BpublicationCriticalpatent/YU48204B/en
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Abstract
NEURO-ZAŠTITNI DERIVATI 3-PIPERIDINO-4-HIDROK-SIHROMANA, u ovoj prijavi se opisuju 3-piperidino-1-hromanol derivati i analozi sledeće formule: gde su A i B uzeti zajedno i predstavljaju -CH2CH2-ili A i B su uzeti odvojeno i predstavljaju H; X je CH2 ili O; X1 je H ili OH; Z je H, F, Cl, Br, ili OH; Zl je H, F, Cl, Br ili (C1-C3) alkil; n je 0 ili 1; a m je m je 0 ili ceo broj od 1 do 6; njihove farmaceutske kompozicije; postupke za tretiranje CNS oštećenja i intermedijere korisne za dobijanje navedenih jedinjenja.NEURO-PROTECTIVE DERIVATIVES OF 3-PIPERIDINO-4-HYDROCH-SICHROMANES, this application describes 3-piperidino-1-chromanol derivatives and analogs of the following formula: wherein A and B are taken together and represent -CH2CH2- or A and B are taken separately and represent H; X is CH2 or O; X1 is H or OH; Z is H, F, Cl, Br, or OH; Z1 is H, F, Cl, Br or (C1-C3) alkyl; n is 0 or 1; and m is m is 0 or an integer from 1 to 6; pharmaceutical compositions thereof; methods for treating CNS damage and intermediates useful for preparing said compounds.
YU19691A1991-02-051991-02-05
NEURO-PROTECTIVE DERIVATIVES OF 3-PIPERIDINO-4-HYDROXYCHROMANES AND THE PROCEDURE FOR THEIR PREPARATION
YU48204B
(en)
Benzimidazolyl-, benzoxazolyl- and benzothiazolyloxazolidinone benzocyclopentan-oxazolidinone containing hetero atoms derivatives, process for the preparation thereof and pharmaceutical compositons containing them
PROCESS FOR MANUFACTURING A PHARMACEUTICAL PREPARATION WITH ANTIMICROBIC ACTION BASED ON A 14-DESOXY-14-ACETOXYMUTILINE DERIVATIVE AND METHOD FOR PREPARING A COMPOUND SUITABLE FOR THE SAID PROCESS.
4-OH-quinoline-carboxylic-acid derivatives substituted in position 2 by a dihydroxy-substituted group, possibly etherified or esterified, process and intermediates for their preparation, their use as medicaments and compositions containing them.
Novel 1(2h) quinoline carboxylic acid derivatives, process of preparation thereof and their application in the synthesis of products having antibiotic effects