WO2013127764A1 - Process for the preparation of phenyl substituted 3 - difluoromethyl - 1 -methyl - 1h - pyrazole - 4 - carboxylic n-methoxy- [1 -methyl- 2 - phenylethyl] amides - Google Patents
Process for the preparation of phenyl substituted 3 - difluoromethyl - 1 -methyl - 1h - pyrazole - 4 - carboxylic n-methoxy- [1 -methyl- 2 - phenylethyl] amides Download PDFInfo
- Publication number
- WO2013127764A1 WO2013127764A1 PCT/EP2013/053773 EP2013053773W WO2013127764A1 WO 2013127764 A1 WO2013127764 A1 WO 2013127764A1 EP 2013053773 W EP2013053773 W EP 2013053773W WO 2013127764 A1 WO2013127764 A1 WO 2013127764A1
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- formula
- compound
- methyl
- preparation
- phenyl
- Prior art date
Links
- 0 Cc1cc(*)cc(*)c1N Chemical compound Cc1cc(*)cc(*)c1N 0.000 description 3
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Description
Claims
Priority Applications (15)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PL13705816T PL2819997T3 (en) | 2012-02-28 | 2013-02-26 | Process for the preparation of phenyl substituted 3 - difluoromethyl - 1 -methyl - 1h - pyrazole - 4 - carboxylic acid n-methoxy- [1 -methyl- 2 - phenylethyl]amides |
CA2863467A CA2863467C (en) | 2012-02-28 | 2013-02-26 | Process for the preparation of phenyl substituted 3-difluoromethyl-1-methyl-1h-pyrazole-4-carboxylic acid n-methoxy- [1-methyl-2-phenylethyl] amides |
JP2014559177A JP6078563B2 (en) | 2012-02-28 | 2013-02-26 | Process for preparing phenyl substituted 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylic acid N-methoxy- [1-methyl-2-phenylethyl] amide |
CN201380011368.1A CN104144914B (en) | 2012-02-28 | 2013-02-26 | For the preparation of the method for 3-difluoromethyl-1-methyl isophthalic acid H-pyrazoles-4-carboxylic acid methoxy-[1-methyl-2-phenyl-ethyl group]-acid amides of phenyl-replacement |
DK13705816.0T DK2819997T3 (en) | 2012-02-28 | 2013-02-26 | Process for the preparation of phenyl-substituted 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylic acid N-methoxy- [1-methyl-2-phenylethyl] amides |
KR1020147024947A KR102031809B1 (en) | 2012-02-28 | 2013-02-26 | Process for the preparation of phenyl substituted 3-difluoromethyl-1-methyl-1h-pyrazole-4-carboxylic acid n-methoxy-[1-methyl-2-phenylethyl] amides |
ES13705816.0T ES2558586T3 (en) | 2012-02-28 | 2013-02-26 | Process for the preparation of phenyl-substituted 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylic acid N-methoxy- [1-methyl-2-phenylethyl] amides |
AU2013225123A AU2013225123B2 (en) | 2012-02-28 | 2013-02-26 | Process for the preparation of phenyl substituted 3 - difluoromethyl - 1 -methyl - 1H - pyrazole - 4 - carboxylic n-methoxy- [1 -methyl- 2 - phenylethyl] amides |
MX2014009948A MX347564B (en) | 2012-02-28 | 2013-02-26 | Process for the preparation of phenyl substituted 3 - difluoromethyl - 1 -methyl - 1h - pyrazole - 4 - carboxylic n-methoxy- [1 -methyl- 2 - phenylethyl] amides. |
BR112014020556A BR112014020556B1 (en) | 2012-02-28 | 2013-02-26 | process for the preparation of phenyl-substituted 3-difluoromethyl-1-methyl-1h-pyrazol-4-carboxylic acid n-methoxy [1-methyl-2-phenylethyl] amides |
EP13705816.0A EP2819997B1 (en) | 2012-02-28 | 2013-02-26 | Process for the preparation of phenyl substituted 3 - difluoromethyl - 1 -methyl - 1h - pyrazole - 4 - carboxylic acid n-methoxy- [1 -methyl- 2 - phenylethyl]amides |
US14/374,547 US9051272B2 (en) | 2012-02-28 | 2013-02-26 | Process for the preparation of phenyl substituted 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylic acid N-methoxy-[1-methyl-2 phenylethyl] amides |
IL233937A IL233937A (en) | 2012-02-28 | 2014-08-04 | Process for the preparation of phenyl substituted 3-difluoromethyl-1-methyl-1h-pyrazole-4-carboxylic n-methoxy-[1-methyl-2-phenylethyl]amides |
ZA2014/05823A ZA201405823B (en) | 2012-02-28 | 2014-08-07 | Process for the preparation of phenyl substituted 3-diflouromethyl -1-methyl-1h-pyrazole-4-carboxylic acid n-methoxy-[1-methyl-2-phenylethyl]amides |
HRP20160001TT HRP20160001T1 (en) | 2012-02-28 | 2015-12-31 | Process for the preparation of phenyl substituted 3 - difluoromethyl - 1 -methyl - 1h - pyrazole - 4 - carboxylic n-methoxy- [1 -methyl- 2 - phenylethyl]amides |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP12157354 | 2012-02-28 | ||
EP12157354.7 | 2012-02-28 |
Publications (1)
Publication Number | Publication Date |
---|---|
WO2013127764A1 true WO2013127764A1 (en) | 2013-09-06 |
Family
ID=47748653
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/EP2013/053773 WO2013127764A1 (en) | 2012-02-28 | 2013-02-26 | Process for the preparation of phenyl substituted 3 - difluoromethyl - 1 -methyl - 1h - pyrazole - 4 - carboxylic n-methoxy- [1 -methyl- 2 - phenylethyl] amides |
Country Status (20)
Country | Link |
---|---|
US (1) | US9051272B2 (en) |
EP (1) | EP2819997B1 (en) |
JP (1) | JP6078563B2 (en) |
KR (1) | KR102031809B1 (en) |
CN (1) | CN104144914B (en) |
AR (1) | AR090172A1 (en) |
AU (1) | AU2013225123B2 (en) |
BR (1) | BR112014020556B1 (en) |
CA (1) | CA2863467C (en) |
CO (1) | CO7051031A2 (en) |
DK (1) | DK2819997T3 (en) |
ES (1) | ES2558586T3 (en) |
HR (1) | HRP20160001T1 (en) |
HU (1) | HUE026564T2 (en) |
IL (1) | IL233937A (en) |
MX (1) | MX347564B (en) |
PL (1) | PL2819997T3 (en) |
TW (1) | TWI491594B (en) |
WO (1) | WO2013127764A1 (en) |
ZA (1) | ZA201405823B (en) |
Cited By (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2016174042A1 (en) | 2015-04-27 | 2016-11-03 | BASF Agro B.V. | Pesticidal compositions |
WO2017207368A1 (en) | 2016-06-02 | 2017-12-07 | BASF Agro B.V. | Fungicidal compositions |
US10130095B2 (en) | 2014-02-19 | 2018-11-20 | BASF Agro B.V. | Fungicidal compositions of pyrazolecarboxylic acid alkoxyamides |
WO2020094527A1 (en) | 2018-11-06 | 2020-05-14 | Syngenta Crop Protection Ag | Hydrogenation process of oxime derivatives |
WO2020128091A1 (en) | 2018-12-21 | 2020-06-25 | Syngenta Participations Ag | Nematicidal compositions |
WO2022157122A1 (en) | 2021-01-22 | 2022-07-28 | Syngenta Crop Protection Ag | Method for the control or suppression of phytopathogenic bacteria |
WO2024038053A1 (en) | 2022-08-16 | 2024-02-22 | Syngenta Crop Protection Ag | New use of pydiflumetofen |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN108610290B (en) * | 2018-06-11 | 2020-04-24 | 武汉工程大学 | Preparation method of fluxapyroxad |
GB201818117D0 (en) * | 2018-11-06 | 2018-12-19 | Syngenta Participations Ag | Enantioselective process |
CN115703701A (en) * | 2021-08-16 | 2023-02-17 | 上海晓明检测技术服务有限公司 | Method for continuously synthesizing 1- (2,4,6-trichloro-phenyl) -propan-2-one by micro-channel |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0810195A1 (en) * | 1996-05-29 | 1997-12-03 | ALFA CHEMICALS ITALIANA S.p.A. | Process for manufacturing 1-(3-trifluoromethyl)phenyl-propan-2-one intermediate in the synthesis of the fenfluramine |
WO2000034229A1 (en) | 1998-12-10 | 2000-06-15 | Bayer Aktiengesellschaft | Process for the preparation of strobilurin intermediates |
WO2010063700A2 (en) | 2008-12-05 | 2010-06-10 | Syngenta Participations Ag | Novel microbiocides |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2006099077A1 (en) * | 2005-03-10 | 2006-09-21 | Merck & Co., Inc. | Novel crystalline forms of antidiabetic compounds |
EP2592931A4 (en) * | 2010-07-13 | 2013-12-11 | Syngenta Participations Ag | Safener compositions and methods for reducing mycotoxins |
-
2013
- 2013-02-26 DK DK13705816.0T patent/DK2819997T3/en active
- 2013-02-26 CA CA2863467A patent/CA2863467C/en active Active
- 2013-02-26 JP JP2014559177A patent/JP6078563B2/en active Active
- 2013-02-26 BR BR112014020556A patent/BR112014020556B1/en active IP Right Grant
- 2013-02-26 KR KR1020147024947A patent/KR102031809B1/en active IP Right Grant
- 2013-02-26 ES ES13705816.0T patent/ES2558586T3/en active Active
- 2013-02-26 MX MX2014009948A patent/MX347564B/en active IP Right Grant
- 2013-02-26 TW TW102106650A patent/TWI491594B/en active
- 2013-02-26 US US14/374,547 patent/US9051272B2/en active Active
- 2013-02-26 CN CN201380011368.1A patent/CN104144914B/en active Active
- 2013-02-26 WO PCT/EP2013/053773 patent/WO2013127764A1/en active Application Filing
- 2013-02-26 EP EP13705816.0A patent/EP2819997B1/en active Active
- 2013-02-26 PL PL13705816T patent/PL2819997T3/en unknown
- 2013-02-26 HU HUE13705816A patent/HUE026564T2/en unknown
- 2013-02-26 AU AU2013225123A patent/AU2013225123B2/en active Active
- 2013-02-27 AR ARP130100601A patent/AR090172A1/en active IP Right Grant
-
2014
- 2014-08-04 IL IL233937A patent/IL233937A/en active IP Right Grant
- 2014-08-07 ZA ZA2014/05823A patent/ZA201405823B/en unknown
- 2014-08-26 CO CO14187079A patent/CO7051031A2/en unknown
-
2015
- 2015-12-31 HR HRP20160001TT patent/HRP20160001T1/en unknown
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0810195A1 (en) * | 1996-05-29 | 1997-12-03 | ALFA CHEMICALS ITALIANA S.p.A. | Process for manufacturing 1-(3-trifluoromethyl)phenyl-propan-2-one intermediate in the synthesis of the fenfluramine |
WO2000034229A1 (en) | 1998-12-10 | 2000-06-15 | Bayer Aktiengesellschaft | Process for the preparation of strobilurin intermediates |
WO2010063700A2 (en) | 2008-12-05 | 2010-06-10 | Syngenta Participations Ag | Novel microbiocides |
Non-Patent Citations (1)
Title |
---|
LI LIA ET AL: "Facile Synthesis of 1-Aryl-2-propanones from Aromatic Amine", SYNTHETIC COMMUNICATIONS: AN INTERNATIONAL JOURNAL FOR RAPID COMMUNICATION OF SYNTHETIC ORGANIC CHEMISTRY, TAYLOR & FRANCIS INC, PHILADELPHIA, PA; US, vol. 37, no. 6, 31 December 2007 (2007-12-31), pages 985 - 991, XP002666726, ISSN: 0039-7911, [retrieved on 20070224], DOI: 10.1080/00397910601163950 * |
Cited By (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US10130095B2 (en) | 2014-02-19 | 2018-11-20 | BASF Agro B.V. | Fungicidal compositions of pyrazolecarboxylic acid alkoxyamides |
WO2016174042A1 (en) | 2015-04-27 | 2016-11-03 | BASF Agro B.V. | Pesticidal compositions |
WO2017207368A1 (en) | 2016-06-02 | 2017-12-07 | BASF Agro B.V. | Fungicidal compositions |
WO2020094527A1 (en) | 2018-11-06 | 2020-05-14 | Syngenta Crop Protection Ag | Hydrogenation process of oxime derivatives |
WO2020128091A1 (en) | 2018-12-21 | 2020-06-25 | Syngenta Participations Ag | Nematicidal compositions |
WO2022157122A1 (en) | 2021-01-22 | 2022-07-28 | Syngenta Crop Protection Ag | Method for the control or suppression of phytopathogenic bacteria |
WO2024038053A1 (en) | 2022-08-16 | 2024-02-22 | Syngenta Crop Protection Ag | New use of pydiflumetofen |
Also Published As
Publication number | Publication date |
---|---|
HRP20160001T1 (en) | 2016-02-12 |
JP2015508794A (en) | 2015-03-23 |
PL2819997T3 (en) | 2016-03-31 |
AU2013225123B2 (en) | 2016-10-20 |
EP2819997A1 (en) | 2015-01-07 |
MX347564B (en) | 2017-05-03 |
IL233937A (en) | 2016-04-21 |
HUE026564T2 (en) | 2016-06-28 |
KR20140138154A (en) | 2014-12-03 |
CN104144914A (en) | 2014-11-12 |
ES2558586T3 (en) | 2016-02-05 |
TW201348209A (en) | 2013-12-01 |
CA2863467C (en) | 2020-03-10 |
BR112014020556B1 (en) | 2019-11-26 |
CO7051031A2 (en) | 2014-09-10 |
AU2013225123A1 (en) | 2014-09-18 |
US9051272B2 (en) | 2015-06-09 |
ZA201405823B (en) | 2015-11-25 |
DK2819997T3 (en) | 2016-01-18 |
TWI491594B (en) | 2015-07-11 |
EP2819997B1 (en) | 2015-10-28 |
IL233937A0 (en) | 2014-09-30 |
US20150018562A1 (en) | 2015-01-15 |
CN104144914B (en) | 2016-03-02 |
CA2863467A1 (en) | 2013-09-06 |
AR090172A1 (en) | 2014-10-22 |
MX2014009948A (en) | 2014-11-12 |
JP6078563B2 (en) | 2017-02-08 |
KR102031809B1 (en) | 2019-10-14 |
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