WO2010149794A3 - Novel pharmaceutical composition comprising poly (allylamin-co-n,n'-diallyl- 1,3-diamino-2-hydroxypropane) - Google Patents

Novel pharmaceutical composition comprising poly (allylamin-co-n,n'-diallyl- 1,3-diamino-2-hydroxypropane) Download PDF

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Publication number
WO2010149794A3
WO2010149794A3 PCT/EP2010/059149 EP2010059149W WO2010149794A3 WO 2010149794 A3 WO2010149794 A3 WO 2010149794A3 EP 2010059149 W EP2010059149 W EP 2010059149W WO 2010149794 A3 WO2010149794 A3 WO 2010149794A3
Authority
WO
WIPO (PCT)
Prior art keywords
pharmaceutical composition
allylamin
hydroxypropane
diallyl
diamino
Prior art date
Application number
PCT/EP2010/059149
Other languages
French (fr)
Other versions
WO2010149794A2 (en
Inventor
Sergio Lloret Pérez
Laura Díaz Guasch
Original Assignee
Combino Pharm, S.L.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from ES200930368A external-priority patent/ES2350999B1/en
Application filed by Combino Pharm, S.L. filed Critical Combino Pharm, S.L.
Publication of WO2010149794A2 publication Critical patent/WO2010149794A2/en
Publication of WO2010149794A3 publication Critical patent/WO2010149794A3/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/74Synthetic polymeric materials
    • A61K31/785Polymers containing nitrogen

Abstract

A solid, pharmaceutical composition for oral administration comprising from about 80% to about 94% by weight of sevelamer including the water of hydration and at least one pharmaceutically acceptable excipient.
PCT/EP2010/059149 2009-06-26 2010-06-28 Novel pharmaceutical composition comprising poly (allylamin-co-n,n'-diallyl- 1,3-diamino-2-hydroxypropane) WO2010149794A2 (en)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
ES200930368 2009-06-26
ES200930368A ES2350999B1 (en) 2009-06-26 2009-06-26 NEW PHARMACEUTICAL COMPOSITION UNDERSTANDING POLY HYDROCHLORIDE (ALILAMIN-CO-N, N'-DIALIL-1,3-DIAMINO-2-PROPANE HYDROXY).
EPPCT/EP2009/058122 2009-06-29
PCT/EP2009/058122 WO2010149230A1 (en) 2009-06-26 2009-06-29 Novel pharmaceutical composition comprising poly (allylamin-co-n,n'-diallyl- 1,3-diamino-2-hydroxypropane) hydrochloride
ARP20100102272 2010-06-25
ARP100102272A AR077244A1 (en) 2009-06-26 2010-06-25 PHARMACEUTICAL COMPOSITION THAT INCLUDES POLI (ALILAMIN-CO-N, N'-DIALIL-1,3-DIAMINO-2-HYDROXIPROPANE)

Publications (2)

Publication Number Publication Date
WO2010149794A2 WO2010149794A2 (en) 2010-12-29
WO2010149794A3 true WO2010149794A3 (en) 2011-06-16

Family

ID=43386953

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2010/059149 WO2010149794A2 (en) 2009-06-26 2010-06-28 Novel pharmaceutical composition comprising poly (allylamin-co-n,n'-diallyl- 1,3-diamino-2-hydroxypropane)

Country Status (1)

Country Link
WO (1) WO2010149794A2 (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103159881A (en) * 2011-12-14 2013-06-19 上海亿法医药科技有限公司 Preparation method for sevelamer hydrochloride
CN103159880B (en) * 2011-12-14 2016-06-22 上海亿法医药科技有限公司 The preparation method of 2-Propen-1-amine polymer with(chloromethyl)oxirane carbonate

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2545907A1 (en) * 2011-07-15 2013-01-16 Combino Pharm, S.L. Aqueous wet granulation process for cross-linked polyallylamine polymers
CN111773190A (en) * 2020-06-24 2020-10-16 北京瑞迪道森医药科技有限公司 Sevelamer carbonate tablet for improving safety of preparation and preparation method thereof

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001028527A2 (en) * 1999-10-19 2001-04-26 Geltex Pharmaceuticals, Inc. Direct compression polymer tablet core
WO2007094779A1 (en) * 2006-02-14 2007-08-23 Teva Pharmaceutical Industries Ltd. Pharmaceutical formulations of aliphatic amine polymers and methods for their manufacture
WO2008062437A2 (en) * 2006-09-01 2008-05-29 Usv Limited Process for the preparation of sevelamer hydrochloride and formulation thereof
WO2009034540A1 (en) * 2007-09-11 2009-03-19 Ranbaxy Laboratories Limited Pharmaceutical composition of sevelamer

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW592727B (en) 1997-04-04 2004-06-21 Chugai Pharmaceutical Co Ltd Phosphate-binding polymer preparations

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001028527A2 (en) * 1999-10-19 2001-04-26 Geltex Pharmaceuticals, Inc. Direct compression polymer tablet core
WO2007094779A1 (en) * 2006-02-14 2007-08-23 Teva Pharmaceutical Industries Ltd. Pharmaceutical formulations of aliphatic amine polymers and methods for their manufacture
WO2008062437A2 (en) * 2006-09-01 2008-05-29 Usv Limited Process for the preparation of sevelamer hydrochloride and formulation thereof
WO2009034540A1 (en) * 2007-09-11 2009-03-19 Ranbaxy Laboratories Limited Pharmaceutical composition of sevelamer

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103159881A (en) * 2011-12-14 2013-06-19 上海亿法医药科技有限公司 Preparation method for sevelamer hydrochloride
CN103159881B (en) * 2011-12-14 2016-04-27 上海亿法医药科技有限公司 The preparation method of sevelamer hydrochloride
CN103159880B (en) * 2011-12-14 2016-06-22 上海亿法医药科技有限公司 The preparation method of 2-Propen-1-amine polymer with(chloromethyl)oxirane carbonate

Also Published As

Publication number Publication date
WO2010149794A2 (en) 2010-12-29

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