UY33393A - Una composición farmacéutica de liberación controlada de losartan - Google Patents
Una composición farmacéutica de liberación controlada de losartanInfo
- Publication number
- UY33393A UY33393A UY0001033393A UY33393A UY33393A UY 33393 A UY33393 A UY 33393A UY 0001033393 A UY0001033393 A UY 0001033393A UY 33393 A UY33393 A UY 33393A UY 33393 A UY33393 A UY 33393A
- Authority
- UY
- Uruguay
- Prior art keywords
- losartan
- pharmaceutical composition
- controlled liberation
- controlled release
- controlled
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
- A61P5/40—Mineralocorticosteroids, e.g. aldosterone; Drugs increasing or potentiating the activity of mineralocorticosteroids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
La presente invención se refiere a una composición farmacéutica de liberación controlada de losartan que comprende un núcleo de retención gástrica con losartan y una cantidad comprendida entre 5 y 25% en peso de hidroxipropilmetilcelulosa como único polímero de liberación controlada, y una capa activa de liberación inmediata que contiene losartan, a su procedimiento de preparación y a su uso para la profilaxis y el tratamiento de la hipertensión
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10382135A EP2392318A1 (en) | 2010-05-21 | 2010-05-21 | A pharmaceutical controlled release composition of losartan |
Publications (1)
Publication Number | Publication Date |
---|---|
UY33393A true UY33393A (es) | 2011-12-30 |
Family
ID=42635468
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY0001033393A UY33393A (es) | 2010-05-21 | 2011-05-17 | Una composición farmacéutica de liberación controlada de losartan |
Country Status (7)
Country | Link |
---|---|
EP (2) | EP2392318A1 (es) |
AR (1) | AR081400A1 (es) |
BR (1) | BR112012029565A2 (es) |
MX (1) | MX2012013362A (es) |
TW (1) | TW201201800A (es) |
UY (1) | UY33393A (es) |
WO (1) | WO2011144724A1 (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2018002673A1 (en) * | 2016-07-01 | 2018-01-04 | N4 Pharma Uk Limited | Novel formulations of angiotensin ii receptor antagonists |
CN107789326A (zh) * | 2016-08-29 | 2018-03-13 | 北京科信必成医药科技发展有限公司 | 一种氢氯噻嗪微片及其制备方法 |
IT201800011123A1 (it) | 2018-12-14 | 2020-06-14 | Dpl Pharma S P A | Composizioni farmaceutiche orali solide per la somministrazione cronotropica di sartani |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2005508358A (ja) | 2001-10-25 | 2005-03-31 | デポメド・インコーポレイテッド | 胃滞留型ロサルタン投与量を用いる治療方法 |
KR100888131B1 (ko) * | 2006-10-10 | 2009-03-11 | 한올제약주식회사 | 시간차 투약 원리를 이용한 심혈관계 질환 치료용 복합제제 |
WO2008054123A1 (en) * | 2006-10-30 | 2008-05-08 | Hanall Pharmaceutical Company, Ltd. | Controlled release complex composition comprising angiotensin-ii-receptor blockers and hmg-coa reductase inhibitors |
-
2010
- 2010-05-21 EP EP10382135A patent/EP2392318A1/en not_active Withdrawn
-
2011
- 2011-05-16 TW TW100117019A patent/TW201201800A/zh unknown
- 2011-05-17 AR ARP110101685A patent/AR081400A1/es not_active Application Discontinuation
- 2011-05-17 UY UY0001033393A patent/UY33393A/es not_active Application Discontinuation
- 2011-05-20 WO PCT/EP2011/058229 patent/WO2011144724A1/en active Application Filing
- 2011-05-20 EP EP11720522A patent/EP2571495A1/en not_active Withdrawn
- 2011-05-20 MX MX2012013362A patent/MX2012013362A/es active IP Right Grant
- 2011-05-20 BR BR112012029565A patent/BR112012029565A2/pt not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AR081400A1 (es) | 2012-08-29 |
EP2571495A1 (en) | 2013-03-27 |
WO2011144724A1 (en) | 2011-11-24 |
EP2392318A1 (en) | 2011-12-07 |
MX2012013362A (es) | 2013-05-01 |
TW201201800A (en) | 2012-01-16 |
BR112012029565A2 (pt) | 2016-12-13 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20210602 |