US20180305315A1 - Pd-1/pd-l1 inhibitors - Google Patents

Pd-1/pd-l1 inhibitors Download PDF

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Publication number
US20180305315A1
US20180305315A1 US15/957,739 US201815957739A US2018305315A1 US 20180305315 A1 US20180305315 A1 US 20180305315A1 US 201815957739 A US201815957739 A US 201815957739A US 2018305315 A1 US2018305315 A1 US 2018305315A1
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United States
Prior art keywords
nr
cycloalkyl
bis
hz
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Abandoned
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US15/957,739
Inventor
Evangelos Aktoudianakis
Todd Appleby
Aesop Cho
Zhimin Du
Michael Graupe
Juan A. Guerrero
Salman Y. Jabri
Lateshkumar Thakorlal Lad
Paulo A. Machicao Tello
Jonathan William Medley
Samuel E. Metobo
Prasenjit Kumar Mukherjee
Devan Naduthambi
Gregory Notte
Eric Q. Parkhill
Barton W. Phillips
Scott Preston Simonovich
Neil H. Squires
Chandrasekar Venkataramani
Peiyuan Wang
William J. Watkins
Jie Xu
Kin Shing Yang
Christopher Allen Ziebenhaus
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Gilead Sciences Inc
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Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Priority to US201762488017P priority Critical
Priority to US201762507678P priority
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Priority to US15/957,739 priority patent/US20180305315A1/en
Assigned to GILEAD SCIENCES, INC. reassignment GILEAD SCIENCES, INC. ASSIGNMENT OF ASSIGNORS INTEREST (SEE DOCUMENT FOR DETAILS). Assignors: MACHICAO TELLO, PAULO A, WANG, PEIYUAN
Assigned to GILEAD SCIENCES, INC. reassignment GILEAD SCIENCES, INC. ASSIGNMENT OF ASSIGNORS INTEREST (SEE DOCUMENT FOR DETAILS). Assignors: VENKATARAMANI, CHANDRASEKAR, GRAUPE, MICHAEL, SIMONOVICH, SCOTT PRESTON, WATKINS, WILLIAM J
Assigned to GILEAD SCIENCES, INC. reassignment GILEAD SCIENCES, INC. ASSIGNMENT OF ASSIGNORS INTEREST (SEE DOCUMENT FOR DETAILS). Assignors: JABRI, SALMAN Y, METOBO, SAMUEL E, AKTOUDIANAKIS, EVANGELOS, APPLEBY, TODD, CHO, AESOP, DU, ZHIMIN, GUERRERO, JUAN A, LAD, Lateshkumar Thakorlal, MEDLEY, Jonathan William, MUKHERJEE, Prasenjit Kumar, NADUTHAMBI, DEVAN, NOTTE, GREGORY, PARKHILL, ERIC Q, PHILLIPS, BARTON W, SQUIRES, NEIL H, XU, JIE, YANG, Kin Shing, ZIEBENHAUS, CHRISTOPHER ALLEN
Publication of US20180305315A1 publication Critical patent/US20180305315A1/en
Application status is Abandoned legal-status Critical

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