UA114106C2 - Спосіб лікування прогестерон-залежного стану антипрогестином - Google Patents

Спосіб лікування прогестерон-залежного стану антипрогестином Download PDF

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Publication number
UA114106C2
UA114106C2 UAA201414106A UAA201414106A UA114106C2 UA 114106 C2 UA114106 C2 UA 114106C2 UA A201414106 A UAA201414106 A UA A201414106A UA A201414106 A UAA201414106 A UA A201414106A UA 114106 C2 UA114106 C2 UA 114106C2
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UA
Ukraine
Prior art keywords
capsule
progesterone
amount
filling
oral
Prior art date
Application number
UAA201414106A
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English (en)
Ukrainian (uk)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48614182&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA114106(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of UA114106C2 publication Critical patent/UA114106C2/uk

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0034Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4816Wall or shell material
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/02Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30Oestrogens

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Reproductive Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
UAA201414106A 2012-05-31 2013-05-30 Спосіб лікування прогестерон-залежного стану антипрогестином UA114106C2 (xx)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261653674P 2012-05-31 2012-05-31
PCT/US2013/043447 WO2013181449A1 (en) 2012-05-31 2013-05-30 Formulations and methods for vaginal delivery of antiprogestins

Publications (1)

Publication Number Publication Date
UA114106C2 true UA114106C2 (xx) 2017-04-25

Family

ID=48614182

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201414106A UA114106C2 (xx) 2012-05-31 2013-05-30 Спосіб лікування прогестерон-залежного стану антипрогестином

Country Status (22)

Country Link
US (1) US10328022B2 (en:Method)
EP (1) EP2854763B1 (en:Method)
JP (1) JP6341910B2 (en:Method)
KR (1) KR102127348B1 (en:Method)
CN (1) CN104334158B (en:Method)
AU (1) AU2013267359C1 (en:Method)
BR (1) BR112014029131B1 (en:Method)
CA (1) CA2872644A1 (en:Method)
CL (1) CL2014003232A1 (en:Method)
CO (1) CO7141411A2 (en:Method)
CR (1) CR20140567A (en:Method)
EA (1) EA030444B1 (en:Method)
ES (1) ES2701400T3 (en:Method)
IL (1) IL235450B (en:Method)
IN (1) IN2014DN10548A (en:Method)
MX (2) MX363640B (en:Method)
NZ (1) NZ702467A (en:Method)
PH (1) PH12014502516A1 (en:Method)
SG (2) SG11201407397WA (en:Method)
UA (1) UA114106C2 (en:Method)
WO (1) WO2013181449A1 (en:Method)
ZA (1) ZA201408262B (en:Method)

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RS62297B1 (sr) 2011-11-23 2021-09-30 Therapeuticsmd Inc Prirodne kombinovane hormonske supstitucione formulacije i terapije
US9301920B2 (en) 2012-06-18 2016-04-05 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US20130338122A1 (en) 2012-06-18 2013-12-19 Therapeuticsmd, Inc. Transdermal hormone replacement therapies
US20150196640A1 (en) 2012-06-18 2015-07-16 Therapeuticsmd, Inc. Progesterone formulations having a desirable pk profile
US10806697B2 (en) 2012-12-21 2020-10-20 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10806740B2 (en) 2012-06-18 2020-10-20 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US10471072B2 (en) 2012-12-21 2019-11-12 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10537581B2 (en) 2012-12-21 2020-01-21 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US9180091B2 (en) 2012-12-21 2015-11-10 Therapeuticsmd, Inc. Soluble estradiol capsule for vaginal insertion
US10568891B2 (en) 2012-12-21 2020-02-25 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US11246875B2 (en) 2012-12-21 2022-02-15 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US11266661B2 (en) 2012-12-21 2022-03-08 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
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KR20180126582A (ko) 2016-04-01 2018-11-27 쎄러퓨틱스엠디, 인코퍼레이티드 스테로이드 호르몬 약제학적 조성물
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CN110678555B (zh) 2017-04-14 2023-10-13 比利时胶囊公司 制作普鲁兰的方法

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Also Published As

Publication number Publication date
CN104334158B (zh) 2018-08-10
AU2013267359B2 (en) 2016-05-26
CO7141411A2 (es) 2014-12-12
BR112014029131B1 (pt) 2021-03-09
CL2014003232A1 (es) 2015-03-13
MX2014014054A (es) 2015-02-12
KR20150014928A (ko) 2015-02-09
EP2854763B1 (en) 2018-09-26
KR102127348B1 (ko) 2020-06-29
NZ702467A (en) 2016-07-29
PH12014502516B1 (en) 2015-01-12
US10328022B2 (en) 2019-06-25
CA2872644A1 (en) 2013-12-05
IL235450A0 (en) 2014-12-31
EA201492290A1 (ru) 2015-03-31
IN2014DN10548A (en:Method) 2015-08-21
MX363640B (es) 2019-03-28
AU2013267359C1 (en) 2016-09-29
CN104334158A (zh) 2015-02-04
US20150111862A1 (en) 2015-04-23
SG11201407397WA (en) 2014-12-30
ES2701400T3 (es) 2019-02-22
MX382986B (es) 2025-03-13
SG10201704858PA (en) 2017-07-28
AU2013267359A1 (en) 2014-11-20
EP2854763A1 (en) 2015-04-08
PH12014502516A1 (en) 2015-01-12
JP2015518052A (ja) 2015-06-25
CR20140567A (es) 2015-03-09
WO2013181449A1 (en) 2013-12-05
BR112014029131A2 (pt) 2018-05-29
ZA201408262B (en) 2015-12-23
IL235450B (en) 2020-02-27
EA030444B1 (ru) 2018-08-31
JP6341910B2 (ja) 2018-06-13
HK1206622A1 (en) 2016-01-15
MX2019003467A (es) 2019-06-06

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