TW200524602A - Nitrogen-containing heterocycles affecting glutamatergic synaptic transmission - Google Patents
Nitrogen-containing heterocycles affecting glutamatergic synaptic transmission Download PDFInfo
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- TW200524602A TW200524602A TW093139143A TW93139143A TW200524602A TW 200524602 A TW200524602 A TW 200524602A TW 093139143 A TW093139143 A TW 093139143A TW 93139143 A TW93139143 A TW 93139143A TW 200524602 A TW200524602 A TW 200524602A
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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| AR058807A1 (es) | 2005-09-29 | 2008-02-27 | Astrazeneca Ab | 5-(fenilisoxazoletoxi)-triazol-3-il piridinas sustituidas, para el tratamiento de trastornos mediados por el receptor mglur5 |
| US8349852B2 (en) | 2009-01-13 | 2013-01-08 | Novartis Ag | Quinazolinone derivatives useful as vanilloid antagonists |
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| WO2011073298A1 (en) * | 2009-12-18 | 2011-06-23 | Neurosearch A/S | Tetrazole derivatives as nicotinic acetylcholine receptor modulators |
| US20120309792A1 (en) * | 2009-12-18 | 2012-12-06 | Neurosearch A/S | Tetrazole derivatives as nicotinic acetylcholine receptor modulators |
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| EP2531490B1 (en) | 2010-02-02 | 2014-10-15 | Novartis AG | Cyclohexyl amide derivatives as crf receptor antagonists |
| GB201312800D0 (en) | 2013-07-17 | 2013-08-28 | Heptares Therapeutics Ltd | mGlu5 modulators |
| WO2016001452A1 (en) | 2014-07-04 | 2016-01-07 | Universität Zürich | Compounds, in particular for use in the treatment of a disease or condition for which a bromodomain inhibitor is indicated |
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| US6660753B2 (en) * | 1999-08-19 | 2003-12-09 | Nps Pharmaceuticals, Inc. | Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
| CN1853630A (zh) * | 2001-02-21 | 2006-11-01 | Nps制药公司 | 杂多环化合物及其在亲代谢的谷氨酸受体拮抗剂中的应用 |
| DE60226756D1 (de) * | 2001-10-04 | 2008-07-03 | Merck & Co Inc | Heteroarylsubstituierte tetrazolmodulatoren des metabotropischen glutamatrezeptors-5 |
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| NO20062533L (no) | 2006-09-19 |
| AU2004312342A1 (en) | 2005-07-21 |
| AR046768A1 (es) | 2005-12-21 |
| CA2548039A1 (en) | 2005-07-21 |
| IL175909A0 (en) | 2008-02-09 |
| CN1906187A (zh) | 2007-01-31 |
| UY28685A1 (es) | 2005-06-30 |
| EP1713791A1 (en) | 2006-10-25 |
| DE602004013469T9 (de) | 2009-09-24 |
| KR20060126993A (ko) | 2006-12-11 |
| BRPI0417308A (pt) | 2007-09-11 |
| HK1095598A1 (en) | 2007-05-11 |
| MXPA06006674A (es) | 2007-04-16 |
| ES2303969T3 (es) | 2008-09-01 |
| ATE393767T1 (de) | 2008-05-15 |
| DE602004013469T2 (de) | 2009-06-18 |
| EP1713791B1 (en) | 2008-04-30 |
| ZA200604681B (en) | 2007-04-25 |
| US20070255061A1 (en) | 2007-11-01 |
| WO2005066155A1 (en) | 2005-07-21 |
| DE602004013469D1 (de) | 2008-06-12 |
| JP2007514790A (ja) | 2007-06-07 |
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