SK283394B6 - Zlúčeniny 4-fenylpiperidínu a jej farmaceuticky prijateľné soli, spôsob ich prípravy, liečivo s ich obsahom a ich použitie - Google Patents

Zlúčeniny 4-fenylpiperidínu a jej farmaceuticky prijateľné soli, spôsob ich prípravy, liečivo s ich obsahom a ich použitie Download PDF

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Publication number
SK283394B6
SK283394B6 SK1619-99A SK161999A SK283394B6 SK 283394 B6 SK283394 B6 SK 283394B6 SK 161999 A SK161999 A SK 161999A SK 283394 B6 SK283394 B6 SK 283394B6
Authority
SK
Slovakia
Prior art keywords
alkyl
compound according
paroxetine
group
compound
Prior art date
Application number
SK1619-99A
Other languages
English (en)
Slovak (sk)
Other versions
SK161999A3 (en
Inventor
Franciscus Bernardus Gemma Benneker
Dalen Frans Van
Jacobus Maria Lemmens
Theodorus Hendricus Antonium Peters
Franti�Ek P�Cha
Original Assignee
Synthon B. V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26647319&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK283394(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Synthon B. V. filed Critical Synthon B. V.
Publication of SK161999A3 publication Critical patent/SK161999A3/sk
Publication of SK283394B6 publication Critical patent/SK283394B6/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
SK1619-99A 1997-06-10 1997-06-10 Zlúčeniny 4-fenylpiperidínu a jej farmaceuticky prijateľné soli, spôsob ich prípravy, liečivo s ich obsahom a ich použitie SK283394B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/NL1997/000328 WO1998056787A1 (de) 1997-06-10 1997-06-10 4-Phenylpiperidin-Derivate
US08/872,023 US5874447A (en) 1997-06-10 1997-06-10 4-Phenylpiperidine compounds for treating depression

Publications (2)

Publication Number Publication Date
SK161999A3 SK161999A3 (en) 2000-08-14
SK283394B6 true SK283394B6 (sk) 2003-07-01

Family

ID=26647319

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1619-99A SK283394B6 (sk) 1997-06-10 1997-06-10 Zlúčeniny 4-fenylpiperidínu a jej farmaceuticky prijateľné soli, spôsob ich prípravy, liečivo s ich obsahom a ich použitie

Country Status (26)

Country Link
US (4) US5874447A (de)
EP (2) EP1078925A1 (de)
JP (1) JP2002503248A (de)
KR (1) KR100543614B1 (de)
AT (1) ATE200781T1 (de)
AU (1) AU3108097A (de)
BG (1) BG64315B1 (de)
BR (1) BR9714787A (de)
CA (1) CA2293247C (de)
CZ (1) CZ295301B6 (de)
DE (2) DE69704679T2 (de)
DK (1) DK0994872T3 (de)
EE (2) EE03970B1 (de)
ES (1) ES2155995T3 (de)
GR (1) GR3035784T3 (de)
HK (1) HK1027352A1 (de)
HU (1) HUP0003141A3 (de)
IL (1) IL133366A (de)
IS (2) IS1927B (de)
NO (3) NO317371B1 (de)
PL (1) PL188450B1 (de)
PT (1) PT994872E (de)
SI (1) SI0994872T1 (de)
SK (1) SK283394B6 (de)
TR (2) TR200201156T2 (de)
WO (1) WO1998056787A1 (de)

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Also Published As

Publication number Publication date
US20010031767A1 (en) 2001-10-18
EE9900570A (et) 2000-08-15
NO20033766D0 (no) 2003-08-25
CZ295301B6 (cs) 2005-07-13
HK1027352A1 (en) 2001-01-12
NO20033765D0 (no) 2003-08-25
JP2002503248A (ja) 2002-01-29
PL188450B1 (pl) 2005-02-28
NO317371B1 (no) 2004-10-18
GR3035784T3 (en) 2001-07-31
IS7098A (is) 2004-01-08
CZ429599A3 (cs) 2000-04-12
CA2293247C (en) 2005-04-12
DK0994872T3 (da) 2001-05-28
NO20033766L (no) 2000-02-09
CA2293247A1 (en) 1998-12-17
ATE200781T1 (de) 2001-05-15
BG64315B1 (bg) 2004-09-30
DE29724281U1 (de) 2000-08-10
US20090326233A1 (en) 2009-12-31
US7598271B1 (en) 2009-10-06
SK161999A3 (en) 2000-08-14
EE200200633A (et) 2003-02-17
BR9714787A (pt) 2000-07-18
EE03970B1 (et) 2003-02-17
TR199903025T2 (xx) 2000-07-21
WO1998056787A1 (de) 1998-12-17
BG103980A (en) 2000-07-31
KR20010013615A (de) 2001-02-26
HUP0003141A2 (en) 2001-03-28
EP0994872B9 (de) 2001-12-05
ES2155995T3 (es) 2001-06-01
IS1927B (is) 2004-04-15
NO995455D0 (no) 1999-11-08
US6900327B2 (en) 2005-05-31
IL133366A (en) 2005-11-20
SI0994872T1 (de) 2001-08-31
IL133366A0 (en) 2001-04-30
EP1078925A1 (de) 2001-02-28
EP0994872B1 (de) 2001-04-25
PT994872E (pt) 2001-09-28
NO20033765L (no) 2000-02-09
PL336895A1 (en) 2000-07-17
KR100543614B1 (ko) 2006-01-20
AU3108097A (en) 1998-12-30
TR200201156T2 (tr) 2002-07-22
NO995455L (no) 2000-02-09
DE69704679T2 (de) 2001-09-13
EP0994872A1 (de) 2000-04-26
US5874447A (en) 1999-02-23
IS5249A (is) 1999-11-16
DE69704679D1 (de) 2001-05-31
HUP0003141A3 (en) 2001-04-28

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