SK1822002A3 - Heterocyclic compounds inhibiting angiogenesis - Google Patents
Heterocyclic compounds inhibiting angiogenesis Download PDFInfo
- Publication number
- SK1822002A3 SK1822002A3 SK182-2002A SK1822002A SK1822002A3 SK 1822002 A3 SK1822002 A3 SK 1822002A3 SK 1822002 A SK1822002 A SK 1822002A SK 1822002 A3 SK1822002 A3 SK 1822002A3
- Authority
- SK
- Slovakia
- Prior art keywords
- borelidine
- compound
- group
- alkyl
- nitrogen
- Prior art date
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- 230000033115 angiogenesis Effects 0.000 title claims abstract description 21
- 230000002401 inhibitory effect Effects 0.000 title abstract description 16
- 150000002391 heterocyclic compounds Chemical class 0.000 title 1
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- 125000001072 heteroaryl group Chemical group 0.000 claims abstract description 4
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- 238000002360 preparation method Methods 0.000 claims description 15
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- 238000011282 treatment Methods 0.000 claims description 10
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- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims description 9
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D313/00—Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Ophthalmology & Optometry (AREA)
- Dermatology (AREA)
- Oncology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrane Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU9902628A HUP9902628A3 (en) | 1999-08-02 | 1999-08-02 | Angiogenesis inhibiting borrelidin derivatives, their use and pharmaceutical compositions containing them |
| PCT/HU2000/000088 WO2001009113A2 (en) | 1999-08-02 | 2000-08-02 | Heterocyclic compounds inhibiting angiogenesis |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SK1822002A3 true SK1822002A3 (en) | 2002-08-06 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK182-2002A SK1822002A3 (en) | 1999-08-02 | 2000-08-02 | Heterocyclic compounds inhibiting angiogenesis |
Country Status (32)
| Country | Link |
|---|---|
| US (1) | US6815465B1 (ja) |
| EP (1) | EP1206462B1 (ja) |
| JP (1) | JP2003506366A (ja) |
| KR (1) | KR20020068495A (ja) |
| CN (1) | CN1243746C (ja) |
| AP (1) | AP1383A (ja) |
| AT (1) | ATE241611T1 (ja) |
| AU (1) | AU772206B2 (ja) |
| BG (1) | BG106373A (ja) |
| BR (1) | BR0012968A (ja) |
| CA (1) | CA2378176A1 (ja) |
| CZ (1) | CZ2002405A3 (ja) |
| DE (1) | DE60003045T2 (ja) |
| DK (1) | DK1206462T3 (ja) |
| ES (1) | ES2200900T3 (ja) |
| HK (1) | HK1048995B (ja) |
| HR (1) | HRP20020103B1 (ja) |
| HU (1) | HUP9902628A3 (ja) |
| IL (1) | IL147904A (ja) |
| IS (1) | IS2137B (ja) |
| MX (1) | MXPA02001117A (ja) |
| NO (1) | NO20020485L (ja) |
| NZ (1) | NZ517422A (ja) |
| OA (1) | OA12004A (ja) |
| PL (1) | PL354281A1 (ja) |
| PT (1) | PT1206462E (ja) |
| RU (1) | RU2247723C2 (ja) |
| SK (1) | SK1822002A3 (ja) |
| UA (1) | UA74341C2 (ja) |
| WO (1) | WO2001009113A2 (ja) |
| YU (1) | YU7302A (ja) |
| ZA (1) | ZA200200838B (ja) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6693099B2 (en) * | 2000-10-17 | 2004-02-17 | The Procter & Gamble Company | Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance |
| ES2337134T3 (es) | 2002-03-12 | 2010-04-21 | Bristol-Myers Squibb Company | Derivados de c3-ciano-epotilona. |
| GB0230217D0 (en) | 2002-12-27 | 2003-02-05 | Biotica Tech Ltd | Borrelidin-producing polyketide synthase and its uses |
| US8440217B1 (en) | 2005-06-15 | 2013-05-14 | Mawaheb M. EL-Naggar | Method and system with contact lens product for treating and preventing adverse eye conditions |
| GB0609981D0 (en) * | 2006-05-19 | 2006-06-28 | Biotica Tech Ltd | Novel compounds |
| GB0713563D0 (en) * | 2007-07-13 | 2007-08-22 | Biotica Tech Ltd | Methods of screening for anti-angiogenic compounds |
| ES2423932T3 (es) * | 2007-08-27 | 2013-09-25 | Basf Se | Compuestos de pirazol para controlar plagas de invertebrados |
| DE102008014077A1 (de) | 2008-03-13 | 2009-09-17 | Discovery Partner International Gmbh | Borrelidin-Derivate |
| WO2009141786A2 (en) * | 2008-05-21 | 2009-11-26 | Piramal Life Sciences Limited | Anti-inflammatory compounds |
| EP3034522B1 (en) | 2014-12-15 | 2019-02-06 | Borealis AG | Use of a polypropylene composition |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH08173176A (ja) * | 1994-12-22 | 1996-07-09 | Mercian Corp | 血管新生阻害剤 |
| JP3786461B2 (ja) * | 1996-02-22 | 2006-06-14 | メルシャン株式会社 | 新生理活性物質 |
-
1999
- 1999-08-02 HU HU9902628A patent/HUP9902628A3/hu unknown
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2000
- 2000-08-02 EP EP00949831A patent/EP1206462B1/en not_active Expired - Lifetime
- 2000-08-02 PL PL00354281A patent/PL354281A1/xx not_active Application Discontinuation
- 2000-08-02 CZ CZ2002405A patent/CZ2002405A3/cs unknown
- 2000-08-02 RU RU2002105518/04A patent/RU2247723C2/ru not_active IP Right Cessation
- 2000-08-02 NZ NZ517422A patent/NZ517422A/en unknown
- 2000-08-02 JP JP2001514316A patent/JP2003506366A/ja not_active Withdrawn
- 2000-08-02 CA CA002378176A patent/CA2378176A1/en not_active Abandoned
- 2000-08-02 US US10/048,659 patent/US6815465B1/en not_active Expired - Fee Related
- 2000-08-02 YU YU7302A patent/YU7302A/sh unknown
- 2000-08-02 WO PCT/HU2000/000088 patent/WO2001009113A2/en not_active Application Discontinuation
- 2000-08-02 AT AT00949831T patent/ATE241611T1/de not_active IP Right Cessation
- 2000-08-02 UA UA2002010814A patent/UA74341C2/uk unknown
- 2000-08-02 ES ES00949831T patent/ES2200900T3/es not_active Expired - Lifetime
- 2000-08-02 AP APAP/P/2002/002413A patent/AP1383A/en active
- 2000-08-02 BR BR0012968-2A patent/BR0012968A/pt not_active IP Right Cessation
- 2000-08-02 PT PT00949831T patent/PT1206462E/pt unknown
- 2000-08-02 CN CNB008123578A patent/CN1243746C/zh not_active Expired - Fee Related
- 2000-08-02 KR KR1020027001484A patent/KR20020068495A/ko not_active Application Discontinuation
- 2000-08-02 DK DK00949831T patent/DK1206462T3/da active
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- 2000-08-02 MX MXPA02001117A patent/MXPA02001117A/es active IP Right Grant
- 2000-08-02 AU AU63090/00A patent/AU772206B2/en not_active Ceased
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2002
- 2002-01-30 NO NO20020485A patent/NO20020485L/no not_active Application Discontinuation
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- 2002-02-01 HR HR20020103A patent/HRP20020103B1/xx not_active IP Right Cessation
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2003
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