SK15162001A3 - Deriváty 13-metylerytromycínu - Google Patents

Deriváty 13-metylerytromycínu Download PDF

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Publication number
SK15162001A3
SK15162001A3 SK1516-2001A SK15162001A SK15162001A3 SK 15162001 A3 SK15162001 A3 SK 15162001A3 SK 15162001 A SK15162001 A SK 15162001A SK 15162001 A3 SK15162001 A3 SK 15162001A3
Authority
SK
Slovakia
Prior art keywords
group
alkyl
compounds
formula
compound
Prior art date
Application number
SK1516-2001A
Other languages
English (en)
Slovak (sk)
Inventor
John Philip Dirlam
Takushi Kaneko
Hamish Alastair Irvine Mcarthur
Wei-Guo Su
Yong-Jin Wu
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of SK15162001A3 publication Critical patent/SK15162001A3/sk

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
SK1516-2001A 1999-05-24 2000-04-25 Deriváty 13-metylerytromycínu SK15162001A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13546899P 1999-05-24 1999-05-24
PCT/IB2000/000502 WO2000071557A1 (en) 1999-05-24 2000-04-25 13-methyl-erythromycin derivatives

Publications (1)

Publication Number Publication Date
SK15162001A3 true SK15162001A3 (sk) 2003-02-04

Family

ID=22468240

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1516-2001A SK15162001A3 (sk) 1999-05-24 2000-04-25 Deriváty 13-metylerytromycínu

Country Status (32)

Country Link
US (2) US20030100518A1 (hr)
EP (1) EP1180110A1 (hr)
JP (1) JP2003500414A (hr)
KR (1) KR20020016799A (hr)
CN (1) CN1351608A (hr)
AP (1) AP2001002302A0 (hr)
AR (1) AR020032A1 (hr)
AU (1) AU3832100A (hr)
BG (1) BG106127A (hr)
BR (1) BR0010938A (hr)
CA (1) CA2373117C (hr)
CZ (1) CZ20013733A3 (hr)
DZ (1) DZ3045A1 (hr)
EA (1) EA200100983A1 (hr)
EE (1) EE200100613A (hr)
HK (1) HK1045523A1 (hr)
HR (1) HRP20010866A2 (hr)
HU (1) HUP0201516A3 (hr)
IL (1) IL145739A0 (hr)
IS (1) IS6128A (hr)
MA (1) MA26740A1 (hr)
NO (1) NO20015172L (hr)
OA (1) OA11945A (hr)
PA (1) PA8495101A1 (hr)
PE (1) PE20010171A1 (hr)
PL (1) PL352720A1 (hr)
SK (1) SK15162001A3 (hr)
TN (1) TNSN00108A1 (hr)
TR (1) TR200103395T2 (hr)
UY (1) UY26161A1 (hr)
WO (1) WO2000071557A1 (hr)
ZA (1) ZA200109595B (hr)

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AR085286A1 (es) 2011-02-21 2013-09-18 Taisho Pharmaceutical Co Ltd Derivado de macrolido sustituido en la posicion c-4
KR20150098675A (ko) 2012-12-24 2015-08-28 라모트 앳 텔-아비브 유니버시티 리미티드 넌센스 돌연변이로부터 생긴 유전적 질환을 치료하기 위한 물질 및 이를 확인하는 방법
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EP3211997A4 (en) 2014-10-08 2018-10-24 President and Fellows of Harvard College 14-membered ketolides and methods of their preparation and use
WO2016154591A1 (en) 2015-03-25 2016-09-29 President And Fellows Of Harvard College Macrolides with modified desosamine sugars and uses thereof

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Also Published As

Publication number Publication date
DZ3045A1 (fr) 2004-03-27
CN1351608A (zh) 2002-05-29
NO20015172L (no) 2002-01-23
AU3832100A (en) 2000-12-12
TNSN00108A1 (fr) 2002-05-30
OA11945A (en) 2006-04-13
PL352720A1 (en) 2003-09-08
CZ20013733A3 (cs) 2002-11-13
HK1045523A1 (zh) 2002-11-29
US20030229031A1 (en) 2003-12-11
CA2373117C (en) 2006-02-28
JP2003500414A (ja) 2003-01-07
HRP20010866A2 (en) 2003-06-30
IS6128A (is) 2001-10-26
EP1180110A1 (en) 2002-02-20
ZA200109595B (en) 2003-05-28
HUP0201516A2 (en) 2002-08-28
AR020032A1 (es) 2002-03-27
CA2373117A1 (en) 2000-11-30
UY26161A1 (es) 2000-12-29
MA26740A1 (fr) 2004-12-20
WO2000071557A1 (en) 2000-11-30
PE20010171A1 (es) 2001-02-10
BG106127A (bg) 2002-05-31
AP2001002302A0 (en) 2001-10-25
IL145739A0 (en) 2002-07-25
EA200100983A1 (ru) 2002-10-31
KR20020016799A (ko) 2002-03-06
BR0010938A (pt) 2002-03-19
PA8495101A1 (es) 2002-08-26
TR200103395T2 (tr) 2002-04-22
US6777543B2 (en) 2004-08-17
US20030100518A1 (en) 2003-05-29
NO20015172D0 (no) 2001-10-23
HUP0201516A3 (en) 2003-03-28
EE200100613A (et) 2003-02-17

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