SI9600050B - Substituted benzenesulphonyl ureas and thioureas, processes for the preparation thereof and use of pharmaceutical preparations on the basis of these compounds as well as medicines containing them - Google Patents

Substituted benzenesulphonyl ureas and thioureas, processes for the preparation thereof and use of pharmaceutical preparations on the basis of these compounds as well as medicines containing them Download PDF

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Publication number
SI9600050B
SI9600050B SI9600050A SI9600050A SI9600050B SI 9600050 B SI9600050 B SI 9600050B SI 9600050 A SI9600050 A SI 9600050A SI 9600050 A SI9600050 A SI 9600050A SI 9600050 B SI9600050 B SI 9600050B
Authority
SI
Slovenia
Prior art keywords
carbon atoms
alkyl
hydrogen
formula
cycloalkyl
Prior art date
Application number
SI9600050A
Other languages
English (en)
Slovenian (sl)
Other versions
SI9600050A (en
Inventor
Heinrich Englert
Uwe Gerlach
Dieter Mania
Heinz Goegelein
Joachim Kaiser
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19505398A external-priority patent/DE19505398A1/de
Priority claimed from DE19522920A external-priority patent/DE19522920A1/de
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of SI9600050A publication Critical patent/SI9600050A/sl
Publication of SI9600050B publication Critical patent/SI9600050B/sl

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C335/00Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C335/40Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of thiourea or isothiourea groups further bound to other hetero atoms
    • C07C335/42Sulfonylthioureas; Sulfonylisothioureas
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/50Compounds containing any of the groups, X being a hetero atom, Y being any atom
    • C07C311/52Y being a hetero atom
    • C07C311/54Y being a hetero atom either X or Y, but not both, being nitrogen atoms, e.g. N-sulfonylurea
    • C07C311/57Y being a hetero atom either X or Y, but not both, being nitrogen atoms, e.g. N-sulfonylurea having sulfur atoms of the sulfonylurea groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/58Y being a hetero atom either X or Y, but not both, being nitrogen atoms, e.g. N-sulfonylurea having sulfur atoms of the sulfonylurea groups bound to carbon atoms of six-membered aromatic rings having nitrogen atoms of the sulfonylurea groups bound to hydrogen atoms or to acyclic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/02Systems containing only non-condensed rings with a three-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/12Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14The ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SI9600050A 1995-02-17 1996-02-16 Substituted benzenesulphonyl ureas and thioureas, processes for the preparation thereof and use of pharmaceutical preparations on the basis of these compounds as well as medicines containing them SI9600050B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19505398A DE19505398A1 (de) 1995-02-17 1995-02-17 Substituierte Benzolsulfonylharnstoffe und -thioharnstoffe, Verfahren zu ihrer Herstellung und Verwendung pharmazeutischer Präparate auf Basis dieser Verbindungen sowie sie enthaltende Heilmittel
DE19522920A DE19522920A1 (de) 1995-06-23 1995-06-23 Substituierte Benzolsulfonylharnstoffe und -thioharnstoffe, Verfahren zu ihrer Herstellung und Verwendung pharmazeutischer Präparate auf Basis dieser Verbindungen sowie sie enthaltende Heilmittel

Publications (2)

Publication Number Publication Date
SI9600050A SI9600050A (en) 1996-10-31
SI9600050B true SI9600050B (en) 2001-12-31

Family

ID=26012537

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9600050A SI9600050B (en) 1995-02-17 1996-02-16 Substituted benzenesulphonyl ureas and thioureas, processes for the preparation thereof and use of pharmaceutical preparations on the basis of these compounds as well as medicines containing them

Country Status (29)

Country Link
US (2) US5880155A (cs)
EP (1) EP0727417B1 (cs)
JP (1) JP3905573B2 (cs)
KR (1) KR100432259B1 (cs)
CN (1) CN1060162C (cs)
AR (1) AR002708A1 (cs)
AT (1) ATE199541T1 (cs)
AU (1) AU700254B2 (cs)
BR (1) BR9600779A (cs)
CA (1) CA2169696C (cs)
CZ (1) CZ291793B6 (cs)
DE (1) DE59606531D1 (cs)
DK (1) DK0727417T3 (cs)
ES (1) ES2155546T3 (cs)
FI (1) FI120391B (cs)
GR (1) GR3035710T3 (cs)
HR (1) HRP960076B1 (cs)
HU (1) HU226462B1 (cs)
IL (1) IL117152A (cs)
MY (1) MY115795A (cs)
NO (1) NO305795B1 (cs)
NZ (1) NZ280992A (cs)
PL (1) PL181792B1 (cs)
PT (1) PT727417E (cs)
RU (1) RU2198872C2 (cs)
SI (1) SI9600050B (cs)
SK (1) SK282131B6 (cs)
TR (1) TR199600117A2 (cs)
TW (1) TW357141B (cs)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19546736A1 (de) * 1995-12-14 1997-06-19 Hoechst Ag Substituierte Chromanylsulfonyl(thio)harnstoffe, Verfahren zu ihrer Herstellung und ihre Verwendung zur Herstellung pharmazeutischer Präparate
BR9714328A (pt) * 1997-01-29 2000-03-21 Pfizer da atividade de interleucina-1
DE19832009A1 (de) 1998-07-16 2000-01-20 Hoechst Marion Roussel De Gmbh 2,5-Substituierte Benzolsulfonylharnstoffe und -thioharnstoffe, Verfahren zu ihrer Herstellung, ihre Verwendung und sie enthaltende pharamazeutische Präparate
DE10129704A1 (de) * 2001-06-22 2003-01-02 Aventis Pharma Gmbh Verwendung von Benzolsulfonyl(thio)harnstoffen in der Behandlung des septischen Schocks
EA011867B1 (ru) 2004-11-22 2009-06-30 Эли Лилли Энд Компани Потенциаторы рецепторов глутамата
CN104649945B (zh) * 2015-02-05 2017-02-22 中国农业大学 一种磺酰脲类、磺酰胺基甲酸酯类化合物的制备方法
US20250145564A1 (en) * 2021-08-16 2025-05-08 Shanghai Institute Of Materia Medica, Chinese Academy Of Sciences Sulfonylurea compound, preparation method therefor, and application thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1198354B (de) * 1963-09-25 1965-08-12 Hoechst Ag Verfahren zur Herstellung von Benzol-sulfonylharnstoffen
DE1185180B (de) * 1963-10-19 1965-01-14 Hoechst Ag Verfahren zur Herstellung von Benzolsulfonylharnstoffen
BE754454A (fr) * 1969-08-06 1971-02-05 Bayer Ag Nouveaux composes hypoglycemiques du type d'arylsulfonylurees et d'arylsulfonylsemicarbazides contenant des groupes carbonamide
DE2413514C3 (de) * 1974-03-21 1982-03-04 Hoechst Ag, 6000 Frankfurt N-Acylaminoathylbenzolsulfonyl-N'-methylharnstoffe, Verfahren zu ihrer Herstellung und deren Verwendung
US4927453A (en) * 1986-10-17 1990-05-22 E. I. Du Pont De Nemours And Company Herbicidal sulfonamides
EP0612724B1 (de) * 1993-02-23 1996-12-27 Hoechst Aktiengesellschaft Substituierte Benzolsulfonylharnstoffe und -thioharnstoffe- Verfahren zu ihrer Herstellung und ihre Verwendung als Pharmazeutika

Also Published As

Publication number Publication date
PL312530A1 (en) 1996-08-19
HUT73982A (en) 1996-10-28
ATE199541T1 (de) 2001-03-15
KR960031432A (ko) 1996-09-17
GR3035710T3 (en) 2001-07-31
BR9600779A (pt) 1997-12-23
EP0727417B1 (de) 2001-03-07
CZ43596A3 (en) 1996-09-11
AU700254B2 (en) 1998-12-24
FI120391B (fi) 2009-10-15
PT727417E (pt) 2001-08-30
TR199600117A2 (tr) 1996-10-21
SK282131B6 (sk) 2001-11-06
IL117152A (en) 2002-07-25
NO305795B1 (no) 1999-07-26
SK21296A3 (en) 1996-10-02
JPH08245556A (ja) 1996-09-24
IL117152A0 (en) 1996-06-18
KR100432259B1 (ko) 2004-09-18
TW357141B (en) 1999-05-01
MY115795A (en) 2003-09-30
AU4555996A (en) 1996-08-29
DK0727417T3 (da) 2001-07-09
US5880155A (en) 1999-03-09
FI960688L (fi) 1996-08-18
CN1134415A (zh) 1996-10-30
SI9600050A (en) 1996-10-31
HU9503877D0 (en) 1996-02-28
RU2198872C2 (ru) 2003-02-20
FI960688A0 (fi) 1996-02-15
NO960628L (no) 1996-08-19
DE59606531D1 (de) 2001-04-12
PL181792B1 (pl) 2001-09-28
CA2169696A1 (en) 1996-08-18
ES2155546T3 (es) 2001-05-16
HU226462B1 (en) 2008-12-29
CN1060162C (zh) 2001-01-03
CZ291793B6 (cs) 2003-05-14
JP3905573B2 (ja) 2007-04-18
AR002708A1 (es) 1998-04-29
EP0727417A1 (de) 1996-08-21
CA2169696C (en) 2008-09-02
HRP960076A2 (en) 1997-12-31
NZ280992A (en) 1996-10-28
US5977177A (en) 1999-11-02
HRP960076B1 (en) 2001-12-31
NO960628D0 (no) 1996-02-16

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Effective date: 20121017