SI9200332A - Method for making of prolinboronate ester - Google Patents

Method for making of prolinboronate ester Download PDF

Info

Publication number
SI9200332A
SI9200332A SI19929200332A SI9200332A SI9200332A SI 9200332 A SI9200332 A SI 9200332A SI 19929200332 A SI19929200332 A SI 19929200332A SI 9200332 A SI9200332 A SI 9200332A SI 9200332 A SI9200332 A SI 9200332A
Authority
SI
Slovenia
Prior art keywords
formula
group
ester
pinandiol
compound
Prior art date
Application number
SI19929200332A
Other languages
English (en)
Slovenian (sl)
Inventor
Roger Snow
Terence A. Kelly
Julian Adams
Simon Coutts
Clark Perry
Original Assignee
Boehringer Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim filed Critical Boehringer Ingelheim
Publication of SI9200332A publication Critical patent/SI9200332A/sl

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyrrole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
SI19929200332A 1991-11-22 1992-11-19 Method for making of prolinboronate ester SI9200332A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79614891A 1991-11-22 1991-11-22
US93619892A 1992-08-26 1992-08-26

Publications (1)

Publication Number Publication Date
SI9200332A true SI9200332A (en) 1993-06-30

Family

ID=27121696

Family Applications (1)

Application Number Title Priority Date Filing Date
SI19929200332A SI9200332A (en) 1991-11-22 1992-11-19 Method for making of prolinboronate ester

Country Status (17)

Country Link
EP (1) EP0641347A1 (enrdf_load_stackoverflow)
JP (1) JPH07501078A (enrdf_load_stackoverflow)
CN (1) CN1073946A (enrdf_load_stackoverflow)
AU (1) AU661362B2 (enrdf_load_stackoverflow)
CA (1) CA2123128A1 (enrdf_load_stackoverflow)
CZ (1) CZ124494A3 (enrdf_load_stackoverflow)
FI (1) FI942345A7 (enrdf_load_stackoverflow)
HU (1) HUT67937A (enrdf_load_stackoverflow)
IL (1) IL103817A0 (enrdf_load_stackoverflow)
MX (1) MX9206628A (enrdf_load_stackoverflow)
NO (1) NO941905L (enrdf_load_stackoverflow)
NZ (1) NZ245207A (enrdf_load_stackoverflow)
PT (1) PT101079A (enrdf_load_stackoverflow)
SI (1) SI9200332A (enrdf_load_stackoverflow)
SK (1) SK59294A3 (enrdf_load_stackoverflow)
TW (1) TW232697B (enrdf_load_stackoverflow)
WO (1) WO1993010127A1 (enrdf_load_stackoverflow)

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JP2002513762A (ja) 1998-05-04 2002-05-14 ポイント セラピューティクス， インコーポレイテッド 造血刺激
BR9910907A (pt) * 1998-06-05 2002-02-13 Point Therapeutics Inc Compostos cìclicos de boroprolina
US6979697B1 (en) 1998-08-21 2005-12-27 Point Therapeutics, Inc. Regulation of substrate activity
US6890904B1 (en) 1999-05-25 2005-05-10 Point Therapeutics, Inc. Anti-tumor agents
JP2003523396A (ja) * 2000-02-25 2003-08-05 ノボ ノルディスク アクティーゼルスカブ ベータ細胞変性の抑制
AU2003218969A1 (en) * 2002-02-01 2003-09-02 Probiodrug Ag Modulation of t lymphocytes using dp iv inhibitors
US7576121B2 (en) 2003-11-12 2009-08-18 Phenomix Corporation Pyrrolidine compounds and methods for selective inhibition of dipeptidyl peptidase-IV
US7317109B2 (en) 2003-11-12 2008-01-08 Phenomix Corporation Pyrrolidine compounds and methods for selective inhibition of dipeptidyl peptidase-IV
US7767828B2 (en) 2003-11-12 2010-08-03 Phenomix Corporation Methyl and ethyl substituted pyrrolidine compounds and methods for selective inhibition of dipeptidyl peptidase-IV
WO2005047297A1 (en) * 2003-11-12 2005-05-26 Phenomix Corporation Heterocyclic boronic acid compounds
CA2545641A1 (en) 2003-11-17 2005-06-02 Novartis Ag Use of organic compounds
SI3366283T1 (sl) 2004-01-20 2021-12-31 Novartis Ag Formulacija za neposredno stiskanje in postopek
AR049631A1 (es) * 2004-04-27 2006-08-23 Wyeth Corp Proceso de acoplamiento para la generacion de derivados reactivos de pirrol -2- carbonitrilo n- sustituidos con contenido de boro para producir biarilos
DOP2006000008A (es) 2005-01-10 2006-08-31 Arena Pharm Inc Terapia combinada para el tratamiento de la diabetes y afecciones relacionadas y para el tratamiento de afecciones que mejoran mediante un incremento de la concentración sanguínea de glp-1
CA2606785A1 (en) 2005-05-19 2006-11-23 Genentech, Inc. Fibroblast activation protein inhibitor compounds and methods
US7825139B2 (en) 2005-05-25 2010-11-02 Forest Laboratories Holdings Limited (BM) Compounds and methods for selective inhibition of dipeptidyl peptidase-IV
CN1331835C (zh) * 2005-10-18 2007-08-15 武汉大学 光活性β－羟基酮的制备方法
BRPI0620027A2 (pt) 2005-12-19 2011-10-25 Tufts College inibidores da protease soft e formas pró-soft
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UA97479C2 (ru) 2006-04-11 2012-02-27 Арена Фармасьютикалз, Инк. Применение g-белок-связанного рецептора (gpcr) для идентификации средств, которые усиливают секрецию глюкозозависимого инсулинотропного пептида (gi)
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SI2318419T1 (sl) * 2008-06-17 2015-07-31 Millennium Pharmaceuticals, Inc. Spojine boronat estra in njihovi farmacevtski sestavki
AR077642A1 (es) 2009-07-09 2011-09-14 Arena Pharm Inc Moduladores del metabolismo y el tratamiento de trastornos relacionados con el mismo
AU2011237775A1 (en) 2010-04-06 2012-11-22 Arena Pharmaceuticals, Inc. Modulators of the GPR119 receptor and the treatment of disorders related thereto
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SG10202003693RA (en) 2014-05-20 2020-05-28 Millennium Pharm Inc Boron-containing proteasome inhibitors for use after primary cancer therapy
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WO2018162722A1 (en) 2017-03-09 2018-09-13 Deutsches Institut Für Ernährungsforschung Potsdam-Rehbrücke Dpp-4 inhibitors for use in treating bone fractures
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CN108047257B (zh) * 2017-12-17 2020-03-13 沧州普瑞东方科技有限公司 一种手性n-boc-吡咯烷-2-硼酸的制备工艺
WO2019163738A1 (en) * 2018-02-20 2019-08-29 Otsuka Pharmaceutical Co., Ltd. Method of 4-boronophenylalanine production
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CA2080474A1 (en) * 1990-04-14 1991-10-15 William W. Bachovchin Inhibitors of dipeptidyl-aminopeptidase type iv
GB9017694D0 (en) * 1990-08-13 1990-09-26 Sandoz Ltd Improvements in or relating to organic chemistry

Also Published As

Publication number Publication date
FI942345A0 (fi) 1994-05-20
JPH07501078A (ja) 1995-02-02
TW232697B (enrdf_load_stackoverflow) 1994-10-21
MX9206628A (es) 1993-05-01
NO941905D0 (no) 1994-05-20
HU9401350D0 (en) 1994-08-29
SK59294A3 (en) 1995-02-08
AU661362B2 (en) 1995-07-20
HUT67937A (en) 1995-05-29
CZ124494A3 (en) 1995-07-12
IL103817A0 (en) 1993-04-04
PT101079A (pt) 1994-02-28
NZ245207A (en) 1994-07-26
WO1993010127A1 (en) 1993-05-27
NO941905L (no) 1994-07-14
CN1073946A (zh) 1993-07-07
CA2123128A1 (en) 1993-05-27
AU3136893A (en) 1993-06-15
FI942345A7 (fi) 1994-05-20
EP0641347A1 (en) 1995-03-08

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