SI9111779B - Lhrh-antagonists. - Google Patents

Lhrh-antagonists. Download PDF

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Publication number
SI9111779B
SI9111779B SI9111779A SI9111779A SI9111779B SI 9111779 B SI9111779 B SI 9111779B SI 9111779 A SI9111779 A SI 9111779A SI 9111779 A SI9111779 A SI 9111779A SI 9111779 B SI9111779 B SI 9111779B
Authority
SI
Slovenia
Prior art keywords
leu7
pro1
nac
ser4
arg8
Prior art date
Application number
SI9111779A
Other languages
English (en)
Slovenian (sl)
Other versions
SI9111779A (en
Inventor
Shaobo Xiao
Original Assignee
Tianjin Municipal Res Inst For
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tianjin Municipal Res Inst For filed Critical Tianjin Municipal Res Inst For
Publication of SI9111779A publication Critical patent/SI9111779A/sl
Publication of SI9111779B publication Critical patent/SI9111779B/sl

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Endocrinology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Medicinal Preparation (AREA)
SI9111779A 1990-11-10 1991-11-08 Lhrh-antagonists. SI9111779B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN90108955A CN1036343C (zh) 1990-11-10 1990-11-10 新促黄体生成素释放激素拮抗类似物的制备方法
YU177991A YU48831B (sh) 1990-11-10 1991-11-08 Lhrh - antagonisti i postupak za njihovu proizvodnju

Publications (2)

Publication Number Publication Date
SI9111779A SI9111779A (en) 1997-04-30
SI9111779B true SI9111779B (en) 2001-12-31

Family

ID=4881223

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9111779A SI9111779B (en) 1990-11-10 1991-11-08 Lhrh-antagonists.

Country Status (29)

Country Link
EP (1) EP0564466B1 (cs)
KR (1) KR100244624B1 (cs)
CN (1) CN1036343C (cs)
AT (1) ATE149520T1 (cs)
AU (1) AU662496B2 (cs)
CA (1) CA2095932C (cs)
CZ (1) CZ284168B6 (cs)
DE (1) DE69125024T2 (cs)
DK (1) DK0564466T3 (cs)
EE (1) EE03141B1 (cs)
ES (1) ES2100965T3 (cs)
FI (1) FI933156A7 (cs)
GR (1) GR3023389T3 (cs)
HR (1) HRP920585B1 (cs)
IE (1) IE913915A1 (cs)
LT (1) LT3971B (cs)
LV (1) LV10106B (cs)
NO (1) NO931697L (cs)
NZ (1) NZ240505A (cs)
PH (1) PH31178A (cs)
PL (1) PL170564B1 (cs)
PT (1) PT99458B (cs)
RU (1) RU2123499C1 (cs)
SI (1) SI9111779B (cs)
SK (1) SK281319B6 (cs)
UA (1) UA41300C2 (cs)
WO (1) WO1992008733A1 (cs)
YU (1) YU48831B (cs)
ZA (1) ZA918847B (cs)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2164096T3 (es) * 1992-12-18 2002-02-16 Abbott Lab Antagonistas de lhrh que comprenden restos de aminoacilo modificados en posicion 5 y 6.
US6828415B2 (en) 1993-02-19 2004-12-07 Zentaris Gmbh Oligopeptide lyophilisate, their preparation and use
DE4305225A1 (de) * 1993-02-19 1994-08-25 Asta Medica Ag Neues Herstellverfahren für Cetrorelix Lyophilisat
DE4338015A1 (de) * 1993-11-08 1995-05-11 Asta Medica Ag Verwendung von D-glucopyranuronsäuren und deren Derivaten zum Einbau in pharmakologisch wirksame Peptide und deren Salze
US5843901A (en) * 1995-06-07 1998-12-01 Advanced Research & Technology Institute LHRH antagonist peptides
DE19544212A1 (de) * 1995-11-28 1997-06-05 Asta Medica Ag Neue LH-RH-Antagonisten mit verbesserter Wirkung
US5968547A (en) 1997-02-24 1999-10-19 Euro-Celtique, S.A. Method of providing sustained analgesia with buprenorphine
DE19911771B4 (de) * 1999-03-17 2006-03-30 Zentaris Gmbh LHRH-Antagonist, Verfahren zu seiner Herstellung und seiner Verwendung
CN101037472B (zh) * 2006-03-14 2013-03-27 中国人民解放军军事医学科学院毒物药物研究所 具有低组胺释放作用的促黄体生成素释放激素拮抗剂
CN102675418B (zh) * 2011-03-15 2016-04-20 中国人民解放军军事医学科学院毒物药物研究所 Lhrh拮抗剂衍生物、其制备方法及用途
CN103524599B (zh) * 2012-07-05 2016-04-20 中国人民解放军军事医学科学院毒物药物研究所 环肽lhrh拮抗剂衍生物及其药物用途
CN104418936B (zh) * 2013-08-20 2018-06-05 中国人民解放军军事医学科学院毒物药物研究所 Lhrh拮抗剂衍生物及其药物用途

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4801577A (en) * 1987-02-05 1989-01-31 Syntex (U.S.A.) Inc. Nonapeptide and decapeptide analogs of LHRH useful as LHRH antagonists
US4851385A (en) * 1987-07-15 1989-07-25 Indiana University Foundation LHRH antagonist analogs having low histamine-release activity

Also Published As

Publication number Publication date
SK281319B6 (sk) 2001-02-12
ZA918847B (en) 1992-08-26
YU177991A (sh) 1994-06-24
KR930703353A (ko) 1993-11-29
AU8861291A (en) 1992-06-11
CN1061605A (zh) 1992-06-03
SK45393A3 (en) 1993-10-06
NO931697L (no) 1993-07-07
LT3971B (en) 1996-05-27
LV10106B (en) 1995-04-20
PT99458A (pt) 1992-10-30
CA2095932C (en) 2003-02-25
ES2100965T3 (es) 1997-07-01
PL295427A1 (en) 1993-09-06
AU662496B2 (en) 1995-09-07
EP0564466A1 (en) 1993-10-13
DE69125024D1 (de) 1997-04-10
GR3023389T3 (en) 1997-08-29
SI9111779A (en) 1997-04-30
ATE149520T1 (de) 1997-03-15
CZ84893A3 (en) 1994-02-16
NO931697D0 (no) 1993-05-10
NZ240505A (en) 1993-04-28
EP0564466B1 (en) 1997-03-05
PL170564B1 (pl) 1996-12-31
CN1036343C (zh) 1997-11-05
CA2095932A1 (en) 1992-05-11
YU48831B (sh) 2002-03-18
WO1992008733A1 (en) 1992-05-29
HRP920585B1 (en) 2000-08-31
DE69125024T2 (de) 1997-07-17
FI933156A0 (fi) 1993-07-09
UA41300C2 (uk) 2001-09-17
LTIP1513A (en) 1995-06-26
LV10106A (lv) 1994-05-10
IE913915A1 (en) 1992-05-20
RU2123499C1 (ru) 1998-12-20
FI933156A7 (fi) 1993-07-09
PT99458B (pt) 1999-02-26
EE03141B1 (et) 1998-12-15
CZ284168B6 (cs) 1998-09-16
PH31178A (en) 1998-03-20
DK0564466T3 (da) 1997-08-25
HRP920585A2 (en) 1997-04-30
KR100244624B1 (ko) 2000-02-15

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Effective date: 20090616