SI1100781T1 - High affinity ligands for nociceptin receptor orl-1 - Google Patents
High affinity ligands for nociceptin receptor orl-1Info
- Publication number
- SI1100781T1 SI1100781T1 SI9930667T SI9930667T SI1100781T1 SI 1100781 T1 SI1100781 T1 SI 1100781T1 SI 9930667 T SI9930667 T SI 9930667T SI 9930667 T SI9930667 T SI 9930667T SI 1100781 T1 SI1100781 T1 SI 1100781T1
- Authority
- SI
- Slovenia
- Prior art keywords
- high affinity
- affinity ligands
- nociceptin receptor
- receptor orl
- orl
- Prior art date
Links
- 102100028646 Nociceptin receptor Human genes 0.000 title 1
- 239000003446 ligand Substances 0.000 title 1
- 108010020615 nociceptin receptor Proteins 0.000 title 1
Classifications
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- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/20—Spiro-condensed ring systems
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/14—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/10—Spiro-condensed systems
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Pulmonology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Epidemiology (AREA)
- Anesthesiology (AREA)
- Diabetes (AREA)
- Rheumatology (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Incineration Of Waste (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US12287898A | 1998-07-27 | 1998-07-27 | |
| EP99937174A EP1100781B1 (en) | 1998-07-27 | 1999-07-26 | High affinity ligands for nociceptin receptor orl-1 |
| PCT/US1999/014165 WO2000006545A1 (en) | 1998-07-27 | 1999-07-26 | High affinity ligands for nociceptin receptor orl-1 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SI1100781T1 true SI1100781T1 (en) | 2005-02-28 |
Family
ID=22405371
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SI9930667T SI1100781T1 (en) | 1998-07-27 | 1999-07-26 | High affinity ligands for nociceptin receptor orl-1 |
Country Status (33)
| Country | Link |
|---|---|
| EP (2) | EP1100781B1 (cs) |
| JP (1) | JP3881516B2 (cs) |
| KR (1) | KR100462074B1 (cs) |
| CN (1) | CN1231467C (cs) |
| AR (2) | AR019478A1 (cs) |
| AT (1) | ATE277013T1 (cs) |
| AU (1) | AU768607C (cs) |
| BR (1) | BR9912495B1 (cs) |
| CA (1) | CA2338206C (cs) |
| CL (1) | CL2009002184A1 (cs) |
| CO (1) | CO5080744A1 (cs) |
| CZ (1) | CZ302533B6 (cs) |
| DE (1) | DE69920476T2 (cs) |
| DK (1) | DK1100781T3 (cs) |
| ES (1) | ES2229750T3 (cs) |
| HK (1) | HK1047544A1 (cs) |
| HU (1) | HUP0103840A3 (cs) |
| ID (1) | ID29137A (cs) |
| IL (1) | IL140449A0 (cs) |
| MY (1) | MY140505A (cs) |
| NO (1) | NO319772B1 (cs) |
| NZ (1) | NZ509033A (cs) |
| PE (1) | PE20000941A1 (cs) |
| PL (1) | PL195633B1 (cs) |
| PT (1) | PT1100781E (cs) |
| RU (1) | RU2237060C2 (cs) |
| SA (1) | SA99200540B1 (cs) |
| SI (1) | SI1100781T1 (cs) |
| SK (1) | SK287678B6 (cs) |
| TR (1) | TR200100241T2 (cs) |
| TW (1) | TW502021B (cs) |
| WO (1) | WO2000006545A1 (cs) |
| ZA (1) | ZA200100150B (cs) |
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1999
- 1999-06-26 ID IDW20010226A patent/ID29137A/id unknown
- 1999-07-26 EP EP99937174A patent/EP1100781B1/en not_active Expired - Lifetime
- 1999-07-26 DK DK99937174T patent/DK1100781T3/da active
- 1999-07-26 CN CNB998092215A patent/CN1231467C/zh not_active Expired - Fee Related
- 1999-07-26 BR BRPI9912495-5B1A patent/BR9912495B1/pt not_active IP Right Cessation
- 1999-07-26 HU HU0103840A patent/HUP0103840A3/hu unknown
- 1999-07-26 AU AU52056/99A patent/AU768607C/en not_active Ceased
- 1999-07-26 TW TW088112624A patent/TW502021B/zh not_active IP Right Cessation
- 1999-07-26 CA CA002338206A patent/CA2338206C/en not_active Expired - Fee Related
- 1999-07-26 ES ES99937174T patent/ES2229750T3/es not_active Expired - Lifetime
- 1999-07-26 PT PT99937174T patent/PT1100781E/pt unknown
- 1999-07-26 SI SI9930667T patent/SI1100781T1/xx unknown
- 1999-07-26 MY MYPI99003144A patent/MY140505A/en unknown
- 1999-07-26 TR TR2001/00241T patent/TR200100241T2/xx unknown
- 1999-07-26 WO PCT/US1999/014165 patent/WO2000006545A1/en not_active Ceased
- 1999-07-26 CZ CZ20010282A patent/CZ302533B6/cs not_active IP Right Cessation
- 1999-07-26 AR ARP990103672A patent/AR019478A1/es active IP Right Grant
- 1999-07-26 PL PL99345671A patent/PL195633B1/pl not_active IP Right Cessation
- 1999-07-26 CO CO99047011A patent/CO5080744A1/es unknown
- 1999-07-26 NZ NZ509033A patent/NZ509033A/en not_active IP Right Cessation
- 1999-07-26 JP JP2000562351A patent/JP3881516B2/ja not_active Expired - Fee Related
- 1999-07-26 IL IL14044999A patent/IL140449A0/xx not_active IP Right Cessation
- 1999-07-26 RU RU2001105910/04A patent/RU2237060C2/ru not_active IP Right Cessation
- 1999-07-26 EP EP02018161A patent/EP1258244A1/en not_active Withdrawn
- 1999-07-26 DE DE69920476T patent/DE69920476T2/de not_active Expired - Lifetime
- 1999-07-26 AT AT99937174T patent/ATE277013T1/de active
- 1999-07-26 KR KR10-2001-7000750A patent/KR100462074B1/ko not_active Expired - Fee Related
- 1999-07-26 SK SK96-2001A patent/SK287678B6/sk not_active IP Right Cessation
- 1999-07-27 PE PE1999000761A patent/PE20000941A1/es not_active Application Discontinuation
- 1999-09-05 SA SA99200540A patent/SA99200540B1/ar unknown
-
2001
- 2001-01-05 ZA ZA200100150A patent/ZA200100150B/en unknown
- 2001-01-26 NO NO20010467A patent/NO319772B1/no not_active IP Right Cessation
- 2001-05-25 HK HK02109089.1A patent/HK1047544A1/en unknown
-
2008
- 2008-10-08 AR ARP080104397A patent/AR068757A2/es unknown
-
2009
- 2009-12-17 CL CL2009002184A patent/CL2009002184A1/es unknown
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