SE432596B - Forfarande for framstellning av 6-piperidino-2,4-diaminopyrimidin-3-oxid - Google Patents

Forfarande for framstellning av 6-piperidino-2,4-diaminopyrimidin-3-oxid

Info

Publication number
SE432596B
SE432596B SE7908629A SE7908629A SE432596B SE 432596 B SE432596 B SE 432596B SE 7908629 A SE7908629 A SE 7908629A SE 7908629 A SE7908629 A SE 7908629A SE 432596 B SE432596 B SE 432596B
Authority
SE
Sweden
Prior art keywords
diaminopyrimidine
reacted
formula
hydroxy
oxide
Prior art date
Application number
SE7908629A
Other languages
English (en)
Swedish (sv)
Other versions
SE7908629L (sv
Inventor
A Vedres
C Szantay
G Balogh
J Horvath
T Mester
Original Assignee
Egyt Gyogyszervegyeszeti Gyar
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egyt Gyogyszervegyeszeti Gyar filed Critical Egyt Gyogyszervegyeszeti Gyar
Publication of SE7908629L publication Critical patent/SE7908629L/xx
Publication of SE432596B publication Critical patent/SE432596B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50—Three nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
SE7908629A 1978-10-27 1979-10-17 Forfarande for framstellning av 6-piperidino-2,4-diaminopyrimidin-3-oxid SE432596B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU78EE2594A HU177601B (en) 1978-10-27 1978-10-27 New process for preparing 6-piperidino-2,4-diamino-pyrimidine-3-oxide

Publications (2)

Publication Number Publication Date
SE7908629L SE7908629L (sv) 1980-04-28
SE432596B true SE432596B (sv) 1984-04-09

Family

ID=10995794

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7908629A SE432596B (sv) 1978-10-27 1979-10-17 Forfarande for framstellning av 6-piperidino-2,4-diaminopyrimidin-3-oxid

Country Status (14)

Country Link
JP (1) JPS5559172A (cs)
AT (1) AT373246B (cs)
CH (1) CH642365A5 (cs)
CS (1) CS213398B2 (cs)
DE (1) DE2943161A1 (cs)
DK (1) DK454579A (cs)
ES (1) ES485457A1 (cs)
FI (1) FI793307A7 (cs)
GB (1) GB2032434B (cs)
HU (1) HU177601B (cs)
PL (1) PL119712B1 (cs)
SE (1) SE432596B (cs)
SU (1) SU913942A3 (cs)
YU (1) YU262579A (cs)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1179344A (en) * 1981-07-15 1984-12-11 Jean-Claude Muller Process for the preparation of 6-¬3,6-dihydro-1(2h)- pyridyl| pyrimidine-3-oxides
CH649291A5 (de) * 1982-03-16 1985-05-15 Hoffmann La Roche Dicarbamate.
HU196061B (en) * 1986-07-10 1988-09-28 Richter Gedeon Vegyeszet Process for production of pirimidine-derivatives
HU196067B (en) * 1986-07-10 1988-09-28 Richter Gedeon Vegyeszet Process for production of 6-amin-1,2-dihydro-1-hydroxi-2-imino-4-piperidin-piramidin
FI864046A7 (fi) * 1986-10-07 1988-04-08 Farmos Oy Menetelmä terapeuttisesti aktiivisen yhdisteen valmistamiseksi.
LU86958A1 (fr) * 1987-07-31 1989-03-08 Oreal Sels d'acide thiamorpholinone carboxylique et de derives de diamino-2,4 pyrimidine,leur utilisation en cosmetique et pharmacie
LU86960A1 (fr) * 1987-07-31 1989-03-08 Oreal Procede de preparation de piperidino-6 diamino-2,4 pyrimidine oxyde-3 et composes nouveaux
US4959475A (en) * 1989-01-04 1990-09-25 Lonza Ltd. Process for the production of 2,4-diamino-6-piperidinyl-pyrimidine-3-N-oxide

Also Published As

Publication number Publication date
PL219242A1 (cs) 1980-06-16
CH642365A5 (de) 1984-04-13
ES485457A1 (es) 1980-10-01
PL119712B1 (en) 1982-01-30
FI793307A7 (fi) 1981-01-01
JPS5559172A (en) 1980-05-02
YU262579A (en) 1983-01-21
CS213398B2 (en) 1982-04-09
SU913942A3 (en) 1982-03-15
GB2032434B (en) 1982-11-17
DE2943161A1 (de) 1980-05-08
AT373246B (de) 1983-12-27
DK454579A (da) 1980-04-28
HU177601B (en) 1981-11-28
SE7908629L (sv) 1980-04-28
GB2032434A (en) 1980-05-08
ATA689879A (de) 1983-05-15

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