SE416303B - Analogiforfarande for framstellning av terapeutiskt verksamma fenylalkansyraderivat av imidazo/1,2-a/pyridin - Google Patents

Analogiforfarande for framstellning av terapeutiskt verksamma fenylalkansyraderivat av imidazo/1,2-a/pyridin

Info

Publication number
SE416303B
SE416303B SE7408886A SE7408886A SE416303B SE 416303 B SE416303 B SE 416303B SE 7408886 A SE7408886 A SE 7408886A SE 7408886 A SE7408886 A SE 7408886A SE 416303 B SE416303 B SE 416303B
Authority
SE
Sweden
Prior art keywords
phenylalkanic
imidazo
pyridine
preparation
therapeutically effective
Prior art date
Application number
SE7408886A
Other languages
English (en)
Other versions
SE7408886L (sv
Inventor
M Nakanishi
T Muro
T Nakao
K Ogawa
Original Assignee
Yoshitomi Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP48076944A external-priority patent/JPS5221509B2/ja
Priority claimed from JP48081380A external-priority patent/JPS5217039B2/ja
Priority claimed from JP10409473A external-priority patent/JPS5711913B2/ja
Priority claimed from JP3289874A external-priority patent/JPS5341678B2/ja
Priority claimed from JP49035007A external-priority patent/JPS5745237B2/ja
Application filed by Yoshitomi Pharmaceutical filed Critical Yoshitomi Pharmaceutical
Publication of SE7408886L publication Critical patent/SE7408886L/xx
Publication of SE416303B publication Critical patent/SE416303B/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SE7408886A 1973-07-07 1974-07-05 Analogiforfarande for framstellning av terapeutiskt verksamma fenylalkansyraderivat av imidazo/1,2-a/pyridin SE416303B (sv)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP48076944A JPS5221509B2 (sv) 1973-07-07 1973-07-07
JP48081380A JPS5217039B2 (sv) 1973-07-21 1973-07-21
JP10409473A JPS5711913B2 (sv) 1973-09-13 1973-09-13
JP3289874A JPS5341678B2 (sv) 1974-03-22 1974-03-22
JP49035007A JPS5745237B2 (sv) 1974-03-27 1974-03-27

Publications (2)

Publication Number Publication Date
SE7408886L SE7408886L (sv) 1975-01-08
SE416303B true SE416303B (sv) 1980-12-15

Family

ID=27521460

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7408886A SE416303B (sv) 1973-07-07 1974-07-05 Analogiforfarande for framstellning av terapeutiskt verksamma fenylalkansyraderivat av imidazo/1,2-a/pyridin

Country Status (7)

Country Link
US (1) US3978071A (sv)
BE (2) BE817247A (sv)
DE (1) DE2432410C2 (sv)
FR (1) FR2235675B1 (sv)
GB (1) GB1442707A (sv)
NL (1) NL7409124A (sv)
SE (1) SE416303B (sv)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4141898A (en) * 1976-08-06 1979-02-27 Pfizer Inc. Imidazo pyridinium quaternary salts as hypoglycemic agents
US4537889A (en) * 1982-12-27 1985-08-27 Eli Lilly And Company Inotropic agents
RO87859B (ro) * 1982-12-27 1985-12-31 Eli Lilly And Company Procedeu pentru prepararea unor derivati de inidazopirimidina pirezina si triazina
US4636502A (en) * 1982-12-27 1987-01-13 Eli Lilly And Company Methods of producing a positive inotropic effect or vasodilation by administration of 2-phenyl imidazo pyrimidines and pyrazines
US4791117A (en) * 1986-09-22 1988-12-13 Ortho Pharmaceutical Corporation 2- or 3-aryl substituted imidazo[1,2-a]pyridines and their use as calcium channel blockers
ES2026666T3 (es) * 1987-03-27 1992-05-01 Synthelabo Procedimiento para preparar derivados de imidazopiridinas.
US5356630A (en) * 1989-02-22 1994-10-18 Massachusetts Institute Of Technology Delivery system for controlled release of bioactive factors
US6147216A (en) * 1993-06-25 2000-11-14 Merrell Pharmaceuticals Inc. Intermediates useful for the preparation of antihistaminic piperidine derivatives
DE69431954T2 (de) 1993-06-25 2003-11-06 Merrell Pharmaceuticals Inc., Cincinnati Neue zwischenprodukte für die herstellung von antihistaminschen 4-diphenylmethyl/diphenylmethoxypiperidin-derivaten
US6689898B2 (en) 1998-07-02 2004-02-10 Aventis Pharmaceuticals Inc. Antihistaminic piperidine derivatives and intermediates for the preparation thereof
US6683094B2 (en) 1998-07-02 2004-01-27 Aventis Pharmaceuticals Inc. Antihistaminic piperidine derivatives and intermediates for the preparation thereof
DE10247271A1 (de) * 2002-10-10 2004-08-26 Grünenthal GmbH Substituierte C-Imidazo[1,2-a]pyridin-3-yle
ITMI20030311A1 (it) * 2003-02-21 2004-08-22 Chiesi Farma Spa Acidi 2-fenil-2-dialchil-acetici per il trattamento della malattia di alzheimer.
US7618981B2 (en) * 2004-05-06 2009-11-17 Cytokinetics, Inc. Imidazopyridinyl-benzamide anti-cancer agents
US7795448B2 (en) * 2004-05-06 2010-09-14 Cytokinetics, Incorporated Imidazoyl-benzamide anti-cancer agents
US7504413B2 (en) * 2004-05-06 2009-03-17 Cytokinetics, Inc. N-(4-(imidazo[1,2A]pyridin-YL)phenethyl)benzamide inhibitors of the mitotic kinesin CENP-E for treating certain cellular proliferation diseases
EP1942899A4 (en) * 2005-11-02 2010-04-28 Cytokinetics Inc INHIBITORS OF MITOTIC KINESINE
JP4738419B2 (ja) * 2005-11-30 2011-08-03 富士フイルムRiファーマ株式会社 アミロイドの凝集及び/又は沈着に起因する疾患の診断薬及び治療薬
US7868001B2 (en) * 2007-11-02 2011-01-11 Hutchison Medipharma Enterprises Limited Cytokine inhibitors
US9199959B2 (en) * 2011-10-25 2015-12-01 Shionogi & Co., Ltd. HIV replication inhibitor

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3318880A (en) * 1963-04-30 1967-05-09 Selvi & C Lab Bioterapico Novel[1, 2-alpha]imidazopyridines and a process for the manufacture thereof
BE788792A (fr) * 1971-09-30 1973-03-13 Ici Ltd Procedes et compositions a usage anti-bacterien

Also Published As

Publication number Publication date
NL7409124A (nl) 1975-01-09
FR2235675B1 (sv) 1978-07-28
SE7408886L (sv) 1975-01-08
DE2432410A1 (de) 1975-01-30
FR2235675A1 (sv) 1975-01-31
GB1442707A (en) 1976-07-14
AU7088474A (en) 1976-01-08
US3978071A (en) 1976-08-31
BE888695Q (fr) 1981-08-28
DE2432410C2 (de) 1986-04-24
BE817247A (fr) 1974-11-04

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