RU2008134314A - Твердые формы производного пирролопиримидина и их применение в качестве противоопухолевых агентов - Google Patents

Твердые формы производного пирролопиримидина и их применение в качестве противоопухолевых агентов Download PDF

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Publication number
RU2008134314A
RU2008134314A RU2008134314/04A RU2008134314A RU2008134314A RU 2008134314 A RU2008134314 A RU 2008134314A RU 2008134314/04 A RU2008134314/04 A RU 2008134314/04A RU 2008134314 A RU2008134314 A RU 2008134314A RU 2008134314 A RU2008134314 A RU 2008134314A
Authority
RU
Russia
Prior art keywords
ethylpiperazin
pyrrolo
ylmethyl
phenylethyl
phenyl
Prior art date
Application number
RU2008134314/04A
Other languages
English (en)
Russian (ru)
Inventor
Михаэль МУТЦ (DE)
Михаэль Мутц
Рето ФИШЕР (CH)
Рето ФИШЕР
Original Assignee
Новартис АГ (CH)
Новартис Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37946476&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RU2008134314(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Новартис АГ (CH), Новартис Аг filed Critical Новартис АГ (CH)
Publication of RU2008134314A publication Critical patent/RU2008134314A/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
RU2008134314/04A 2006-01-23 2007-01-19 Твердые формы производного пирролопиримидина и их применение в качестве противоопухолевых агентов RU2008134314A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76122406P 2006-01-23 2006-01-23
US60/761,224 2006-01-23

Publications (1)

Publication Number Publication Date
RU2008134314A true RU2008134314A (ru) 2010-02-27

Family

ID=37946476

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2008134314/04A RU2008134314A (ru) 2006-01-23 2007-01-19 Твердые формы производного пирролопиримидина и их применение в качестве противоопухолевых агентов

Country Status (13)

Country Link
EP (1) EP1979357A1 (ko)
JP (1) JP2009523768A (ko)
KR (1) KR20080095859A (ko)
CN (1) CN101370814A (ko)
AR (1) AR059090A1 (ko)
AU (1) AU2007206925A1 (ko)
BR (1) BRPI0706729A2 (ko)
CA (1) CA2636954A1 (ko)
PE (1) PE20071323A1 (ko)
RU (1) RU2008134314A (ko)
TN (1) TNSN08312A1 (ko)
TW (1) TW200738719A (ko)
WO (1) WO2007082946A1 (ko)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20011349A1 (es) * 2000-06-16 2002-01-19 Upjohn Co 1-aril-4-oxo-1,4-dihidro-3-quinolincarboxamidas como agentes antivirales
GB0119249D0 (en) * 2001-08-07 2001-10-03 Novartis Ag Organic compounds
US20050038048A1 (en) * 2001-10-29 2005-02-17 Ball Howard Ashley Use of 7h-pyrrollo{2,3-d}pyrimidine derivatives in the treatment of solid tumor diseases
US20080227980A1 (en) * 2005-08-05 2008-09-18 Novartis Ag Preparation of a 7H-Pyrrolo [2,3-D] Pyrimidine Derivative

Also Published As

Publication number Publication date
AR059090A1 (es) 2008-03-12
KR20080095859A (ko) 2008-10-29
BRPI0706729A2 (pt) 2011-04-05
CN101370814A (zh) 2009-02-18
TNSN08312A1 (en) 2009-12-29
CA2636954A1 (en) 2007-07-26
PE20071323A1 (es) 2008-02-15
WO2007082946A1 (en) 2007-07-26
EP1979357A1 (en) 2008-10-15
TW200738719A (en) 2007-10-16
JP2009523768A (ja) 2009-06-25
AU2007206925A1 (en) 2007-07-26

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Legal Events

Date Code Title Description
FA92 Acknowledgement of application withdrawn (lack of supplementary materials submitted)

Effective date: 20110302