RS57225B1 - Derivati pirolo[3,2-d]pirimidina za tretman viralnih infekcija i drugih bolesti - Google Patents
Derivati pirolo[3,2-d]pirimidina za tretman viralnih infekcija i drugih bolestiInfo
- Publication number
- RS57225B1 RS57225B1 RS20180577A RSP20180577A RS57225B1 RS 57225 B1 RS57225 B1 RS 57225B1 RS 20180577 A RS20180577 A RS 20180577A RS P20180577 A RSP20180577 A RS P20180577A RS 57225 B1 RS57225 B1 RS 57225B1
- Authority
- RS
- Serbia
- Prior art keywords
- pyrrolo
- diseases
- treatment
- viral infections
- pyrimidine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12187994 | 2012-10-10 | ||
| EP13779766.8A EP2906563B1 (en) | 2012-10-10 | 2013-10-09 | Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseases |
| PCT/EP2013/070990 WO2014056953A1 (en) | 2012-10-10 | 2013-10-09 | Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| RS57225B1 true RS57225B1 (sr) | 2018-07-31 |
Family
ID=47073301
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RS20180577A RS57225B1 (sr) | 2012-10-10 | 2013-10-09 | Derivati pirolo[3,2-d]pirimidina za tretman viralnih infekcija i drugih bolesti |
Country Status (32)
| Country | Link |
|---|---|
| US (3) | US9499549B2 (sr) |
| EP (1) | EP2906563B1 (sr) |
| JP (1) | JP6293765B2 (sr) |
| KR (2) | KR102280595B1 (sr) |
| CN (1) | CN104837840B (sr) |
| AU (1) | AU2013328732B2 (sr) |
| BR (1) | BR112015007586B1 (sr) |
| CA (1) | CA2884478C (sr) |
| CL (1) | CL2015000898A1 (sr) |
| CY (1) | CY1120885T1 (sr) |
| DK (1) | DK2906563T3 (sr) |
| EA (2) | EA035327B1 (sr) |
| ES (1) | ES2670513T3 (sr) |
| HK (1) | HK1209412A1 (sr) |
| HR (1) | HRP20180771T1 (sr) |
| HU (1) | HUE037064T2 (sr) |
| IL (1) | IL237761B (sr) |
| LT (1) | LT2906563T (sr) |
| MX (1) | MX365114B (sr) |
| MY (1) | MY179392A (sr) |
| NO (1) | NO2906563T3 (sr) |
| NZ (1) | NZ705589A (sr) |
| PH (1) | PH12015500758B1 (sr) |
| PL (1) | PL2906563T3 (sr) |
| PT (1) | PT2906563T (sr) |
| RS (1) | RS57225B1 (sr) |
| SG (1) | SG11201502622VA (sr) |
| SI (1) | SI2906563T1 (sr) |
| TR (1) | TR201807076T4 (sr) |
| UA (1) | UA115677C2 (sr) |
| WO (1) | WO2014056953A1 (sr) |
| ZA (1) | ZA201502383B (sr) |
Families Citing this family (143)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK2694484T3 (en) | 2011-04-08 | 2018-11-05 | Janssen Sciences Ireland Uc | PYRIMIDINE DERIVATIVES FOR TREATING VIRUS INFECTIONS |
| RS57851B1 (sr) | 2011-11-09 | 2018-12-31 | Janssen Sciences Ireland Uc | Purinski derivati za tretman viralnih infekcija |
| EA035790B1 (ru) | 2012-07-13 | 2020-08-11 | Янссен Сайенсиз Айрлэнд Юси | Макроциклические пурины для лечения вирусных инфекций |
| HUE037064T2 (hu) * | 2012-10-10 | 2018-08-28 | Janssen Sciences Ireland Uc | Pirrolo[3,2-d]-pirimidin származékok vírusos fertõzések és egyéb betegségek kezelésére |
| SG11201503042QA (en) | 2012-11-16 | 2015-06-29 | Janssen Sciences Ireland Uc | Heterocyclic substituted 2-amino-quinazoline derivatives for the treatment of viral infections |
| JP6404835B2 (ja) | 2013-02-21 | 2018-10-17 | ヤンセン・サイエンシズ・アイルランド・ユーシー | ウイルス感染の治療のための２−アミノピリミジン誘導体 |
| JP6336036B2 (ja) | 2013-03-29 | 2018-06-06 | ヤンセン・サイエンシズ・アイルランド・ユーシー | ウイルス感染治療のための大環状デアザプリノン |
| BR112015028890B1 (pt) | 2013-05-24 | 2022-09-20 | Janssen Sciences Ireland Uc | Derivados de piridona, composição farmacêutica que os compreende e uso dos mesmos |
| MX361527B (es) * | 2013-06-27 | 2018-12-07 | Janssen Sciences Ireland Uc | Derivados de pirrolo[3,2-d]pirimidina para el tratamiento de infecciones víricas y otras enfermedades. |
| WO2015014815A1 (en) | 2013-07-30 | 2015-02-05 | Janssen R&D Ireland | THIENO[3,2-d]PYRIMIDINES DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS |
| CU24401B1 (es) * | 2014-05-01 | 2019-05-03 | Novartis Ag | Compuestos derivados de metoxibencil-pirrolopirimidin-amina como agonistas del receptor tipo toll 7 (tlr7) |
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| SG11201503042QA (en) | 2012-11-16 | 2015-06-29 | Janssen Sciences Ireland Uc | Heterocyclic substituted 2-amino-quinazoline derivatives for the treatment of viral infections |
| JP6404835B2 (ja) | 2013-02-21 | 2018-10-17 | ヤンセン・サイエンシズ・アイルランド・ユーシー | ウイルス感染の治療のための２−アミノピリミジン誘導体 |
| JP6336036B2 (ja) | 2013-03-29 | 2018-06-06 | ヤンセン・サイエンシズ・アイルランド・ユーシー | ウイルス感染治療のための大環状デアザプリノン |
| WO2015014815A1 (en) | 2013-07-30 | 2015-02-05 | Janssen R&D Ireland | THIENO[3,2-d]PYRIMIDINES DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS |
| EP3166938A4 (en) | 2014-07-11 | 2018-01-17 | Northwestern University | 2-imidazolyl-pyrimidine scaffolds as potent and selective inhibitors of neuronal nitric oxide synthase |
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