PL147092B1 - Process for preparing novel n-/bicycloheterocyclo/-4-piperidinamines - Google Patents

Process for preparing novel n-/bicycloheterocyclo/-4-piperidinamines Download PDF

Info

Publication number
PL147092B1
PL147092B1 PL24297083A PL24297083A PL147092B1 PL 147092 B1 PL147092 B1 PL 147092B1 PL 24297083 A PL24297083 A PL 24297083A PL 24297083 A PL24297083 A PL 24297083A PL 147092 B1 PL147092 B1 PL 147092B1
Authority
PL
Poland
Prior art keywords
group
formula
lower alkyl
groups
radical
Prior art date
Application number
PL24297083A
Other languages
English (en)
Polish (pl)
Other versions
PL242970A1 (en
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of PL242970A1 publication Critical patent/PL242970A1/xx
Publication of PL147092B1 publication Critical patent/PL147092B1/pl

Links

Landscapes

  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PL24297083A 1982-07-12 1983-07-12 Process for preparing novel n-/bicycloheterocyclo/-4-piperidinamines PL147092B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US39762682A 1982-07-12 1982-07-12

Publications (2)

Publication Number Publication Date
PL242970A1 PL242970A1 (en) 1985-08-13
PL147092B1 true PL147092B1 (en) 1989-04-29

Family

ID=23571984

Family Applications (1)

Application Number Title Priority Date Filing Date
PL24297083A PL147092B1 (en) 1982-07-12 1983-07-12 Process for preparing novel n-/bicycloheterocyclo/-4-piperidinamines

Country Status (4)

Country Link
JP (1) JPS5921680A (fr)
IN (1) IN156065B (fr)
PL (1) PL147092B1 (fr)
ZA (1) ZA835044B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4888426A (en) * 1983-11-30 1989-12-19 Janssen Pharmaceutica N.V. 1-(5-methyl-furan-2-ylmethyl)-N-(4-piperidinyl)imidazo [4,5-6]pyridine-2-amine
ATE79620T1 (de) * 1986-02-03 1992-09-15 Janssen Pharmaceutica Nv N-heterozyklische-4-piperidinamine enthaltende anti-histaminische zusammensetzungen.
EP0650476B1 (fr) * 1993-04-07 2002-06-26 Otsuka Pharmaceutical Co., Ltd. Agents vasodilatateurs peripheriques comportant comme principe actif des derives de la piperidine 4-amino n-acylee
MY142362A (en) 2004-01-29 2010-11-30 Otsuka Pharma Co Ltd Pharmaceutical composition for promoting angiogenesis
JP5617970B2 (ja) * 2009-02-19 2014-11-05 富士通株式会社 新規化合物、並びに、結合阻害剤、抗アレルギー剤、抗喘息剤、及び抗炎症剤
JP5617969B2 (ja) * 2009-02-19 2014-11-05 富士通株式会社 新規化合物、並びに、結合阻害剤、抗アレルギー剤、抗喘息剤、及び抗炎症剤

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1140119A (fr) * 1978-04-03 1983-01-25 Joseph Torremans Nouvelles n-heterocycle-4-piperidinamines

Also Published As

Publication number Publication date
PL242970A1 (en) 1985-08-13
IN156065B (fr) 1985-05-04
ZA835044B (en) 1985-02-27
JPS5921680A (ja) 1984-02-03

Similar Documents

Publication Publication Date Title
SU1297728A3 (ru) Способ получени @ -гетероциклил-4-пиперидинаминов или их фармацевтически приемлемых солей
CN103974950B (zh) 作为ccr(4)拮抗剂的取代的苯并咪唑类和苯并吡唑类
KR870001169B1 (ko) 4-[(두고리 헤테로시클릴)-메틸 및 -헤테로] 피페리딘 유도체의 제조방법
KR100725190B1 (ko) 4-아미노피페리딘 유도체 및 그의 약제로서의 용도
US7105548B2 (en) Heteroaryl substituted triazole modulators of metabotropic glutamate receptor-5
US20060194807A1 (en) Di-aryl substituted pyrazole modulators of metabotropic glutamate receptor-5
JPS6110577A (ja) 5員複素環式環を含有するn−(二環式ヘテロシクリル)−4−ピペリジンアミン類
CS256358B2 (en) Method of n-heterocyclyl-4-piperidinamines preparation
CN102015682B (zh) 作为肾素抑制剂的3,4-取代的哌啶衍生物
TW201300360A (zh) 做為jak激酶調節劑之菸鹼醯胺
US20070082067A1 (en) Di-aryl substituted triazole modulators of metabotropic glutamate receptor-5
EP0937065A1 (fr) Agonistes et antagonistes contraints de somatostatine
PL146377B1 (en) Method of obtaining novel derivatives 4-piperidinoamine
PL147092B1 (en) Process for preparing novel n-/bicycloheterocyclo/-4-piperidinamines
WO1995016683A1 (fr) Composes de 6-(2-imidazolinylamino)quinoline utiles en tant qu'agonistes des adrenocepteurs alpha-2
AU2003267000B2 (en) 2-thio-substituted imidazole derivatives and their use in pharmaceutics
JP5872591B2 (ja) ピラゾール化合物
US5578607A (en) 6-(2-imidazolinylamino)quinoline compounds useful as alpha-2 adrenoceptor agonists
US4820822A (en) Novel N-(bicyclic heterocyclyl)-4-piperidinamines
US4760074A (en) Novel-N-(bicyclic heterocyclyl)-4-piperidinamines
USRE33833E (en) Novel N-(bicyclic heterocyclyl)-4-piperidinamines
KR880000247B1 (ko) 4-[(두고리 헤테로시클릴)-메틸 및-헤테로] 피페리딘 유도체의 제조방법
PL146228B1 (en) Method of obtaining novel n-/bicyclic heterocyclilo/-4-piperidinamines containing five-member heterocyclic rings
CZ16485A3 (cs) Způsob přípravy 4-/(bicyklyl heterocyklyl) methyl a hetero/-piperidinů
JPS60174778A (ja) N−ヘテロシクリル−4−ピペリジンアミン