NO326546B1 - Pyridinderivater, fremgangsmate for fremstilling derav samt farmasoytisk preparat omfattende en slik forbindelse - Google Patents
Pyridinderivater, fremgangsmate for fremstilling derav samt farmasoytisk preparat omfattende en slik forbindelse Download PDFInfo
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- NO326546B1 NO326546B1 NO20034122A NO20034122A NO326546B1 NO 326546 B1 NO326546 B1 NO 326546B1 NO 20034122 A NO20034122 A NO 20034122A NO 20034122 A NO20034122 A NO 20034122A NO 326546 B1 NO326546 B1 NO 326546B1
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- Prior art keywords
- compound
- hydrogen
- formula
- phenyl
- chlorophenyl
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Classifications
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pulmonology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Cardiology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
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- Immunology (AREA)
- Diabetes (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Vascular Medicine (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0107505A GB0107505D0 (en) | 2001-03-26 | 2001-03-26 | Organic compounds |
| US33828101P | 2001-12-06 | 2001-12-06 | |
| PCT/EP2002/003332 WO2002076946A2 (en) | 2001-03-26 | 2002-03-25 | Fused pyridine derivatives for use as vanilloid receptor antagonists for treating pain. |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20034122D0 NO20034122D0 (no) | 2003-09-16 |
| NO20034122L NO20034122L (no) | 2003-09-16 |
| NO326546B1 true NO326546B1 (no) | 2009-01-05 |
Family
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20034122A NO326546B1 (no) | 2001-03-26 | 2003-09-16 | Pyridinderivater, fremgangsmate for fremstilling derav samt farmasoytisk preparat omfattende en slik forbindelse |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US7915264B2 (zh) |
| EP (1) | EP1377576A2 (zh) |
| JP (1) | JP4205430B2 (zh) |
| KR (1) | KR20030083755A (zh) |
| CN (1) | CN1500089A (zh) |
| BR (1) | BR0208338A (zh) |
| CA (1) | CA2441599A1 (zh) |
| CZ (1) | CZ20032561A3 (zh) |
| HU (1) | HUP0303623A2 (zh) |
| IL (1) | IL157815A0 (zh) |
| MX (1) | MXPA03008754A (zh) |
| NO (1) | NO326546B1 (zh) |
| PE (1) | PE20021161A1 (zh) |
| PL (1) | PL363907A1 (zh) |
| RU (1) | RU2003130221A (zh) |
| SK (1) | SK11952003A3 (zh) |
| WO (1) | WO2002076946A2 (zh) |
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| ATE393141T1 (de) | 2000-08-21 | 2008-05-15 | Pacific Corp | Neue thiourea-derivate und pharmazeutische zusammensetzungen die diese enthalten |
| WO2002016319A1 (en) | 2000-08-21 | 2002-02-28 | Pacific Corporation | Novel thiourea compounds and the pharmaceutical compositions containing the same |
| MXPA04006882A (es) | 2002-01-17 | 2004-12-06 | Neurogen Corp | Analogos substituidos de quinazolin-4-ilamina como moduladores de receptores de capsaicina. |
| EP2033951A3 (en) | 2002-02-01 | 2009-12-23 | Euro-Celtique S.A. | 2-Piperazine-pyridines useful for treating pain |
| US6864261B2 (en) | 2002-05-02 | 2005-03-08 | Euro-Celtique S.A. | Therapeutic agents useful for treating pain |
| GB0229808D0 (en) * | 2002-12-20 | 2003-01-29 | Glaxo Group Ltd | Novel compositions |
| JP4909068B2 (ja) * | 2003-02-14 | 2012-04-04 | グラクソ グループ リミテッド | カルボキサミド誘導体 |
| EP2281823A3 (en) | 2003-05-20 | 2011-09-07 | Ajinomoto Co., Inc. | Anti-inflammatory and analgesic piperidine derivatives |
| GB0319150D0 (en) | 2003-08-14 | 2003-09-17 | Glaxo Group Ltd | Novel compounds |
| CA2545725A1 (en) | 2003-11-14 | 2005-06-02 | Merck Sharp & Dohme Limited | Bicyclic pyrimidin-4-(3h)-ones and analogues and derivatives thereof which modulate the function of the vanilloid-1 receptor (vr1) |
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Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2749344A (en) | 1953-01-02 | 1956-06-05 | Burroughs Wellcome Co | Pyrimidine compounds |
| US5958930A (en) * | 1991-04-08 | 1999-09-28 | Duquesne University Of The Holy Ghost | Pyrrolo pyrimidine and furo pyrimidine derivatives |
| CA2180122A1 (en) | 1994-01-03 | 1995-07-13 | Sui Xiong Cai | 8-aza, 6-aza and 6,8-diaza-1,4-dihydroquinoxaline-2,3-diones and the usethereof as antagonists for the glycine/nmda receptor |
| FR2750862B1 (fr) | 1996-07-12 | 1998-10-16 | Dupin Jean Pierre | Utilisation d'heterocycles diazotes fusionnes avec un systeme aromatique ou heteroaromatique pour le traitement des maladies thrombo-emboliques |
-
2002
- 2002-03-25 JP JP2002576207A patent/JP4205430B2/ja not_active Expired - Fee Related
- 2002-03-25 KR KR10-2003-7012460A patent/KR20030083755A/ko not_active Application Discontinuation
- 2002-03-25 RU RU2003130221/04A patent/RU2003130221A/ru not_active Application Discontinuation
- 2002-03-25 IL IL15781502A patent/IL157815A0/xx unknown
- 2002-03-25 EP EP02730062A patent/EP1377576A2/en not_active Withdrawn
- 2002-03-25 CA CA002441599A patent/CA2441599A1/en not_active Abandoned
- 2002-03-25 US US10/469,756 patent/US7915264B2/en not_active Expired - Fee Related
- 2002-03-25 PL PL02363907A patent/PL363907A1/xx not_active Application Discontinuation
- 2002-03-25 CN CNA028073495A patent/CN1500089A/zh active Pending
- 2002-03-25 HU HU0303623A patent/HUP0303623A2/hu unknown
- 2002-03-25 MX MXPA03008754A patent/MXPA03008754A/es not_active Application Discontinuation
- 2002-03-25 CZ CZ20032561A patent/CZ20032561A3/cs unknown
- 2002-03-25 SK SK1195-2003A patent/SK11952003A3/sk unknown
- 2002-03-25 WO PCT/EP2002/003332 patent/WO2002076946A2/en not_active Application Discontinuation
- 2002-03-25 BR BR0208338-8A patent/BR0208338A/pt not_active IP Right Cessation
- 2002-03-26 PE PE2002000241A patent/PE20021161A1/es not_active Application Discontinuation
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2003
- 2003-09-16 NO NO20034122A patent/NO326546B1/no not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| SK11952003A3 (sk) | 2004-03-02 |
| NO20034122D0 (no) | 2003-09-16 |
| WO2002076946A3 (en) | 2002-12-27 |
| US20040138454A1 (en) | 2004-07-15 |
| JP4205430B2 (ja) | 2009-01-07 |
| BR0208338A (pt) | 2004-03-09 |
| PE20021161A1 (es) | 2003-02-21 |
| IL157815A0 (en) | 2004-03-28 |
| US7915264B2 (en) | 2011-03-29 |
| EP1377576A2 (en) | 2004-01-07 |
| KR20030083755A (ko) | 2003-10-30 |
| CA2441599A1 (en) | 2002-10-03 |
| CZ20032561A3 (cs) | 2003-12-17 |
| HUP0303623A2 (hu) | 2004-03-01 |
| WO2002076946A2 (en) | 2002-10-03 |
| NO20034122L (no) | 2003-09-16 |
| CN1500089A (zh) | 2004-05-26 |
| MXPA03008754A (es) | 2004-02-18 |
| PL363907A1 (en) | 2004-11-29 |
| RU2003130221A (ru) | 2005-04-10 |
| JP2004528312A (ja) | 2004-09-16 |
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