NO323597B1 - Substituerte benzimidazoler, fremgangsmate for fremstilling av samme, farmasoytisk sammensetning innbefattende samme, anvendelse av samme for fremstilling av medikament og fremgangsmate for fremstilling av farmasoytisk middel. - Google Patents

Substituerte benzimidazoler, fremgangsmate for fremstilling av samme, farmasoytisk sammensetning innbefattende samme, anvendelse av samme for fremstilling av medikament og fremgangsmate for fremstilling av farmasoytisk middel. Download PDF

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Publication number
NO323597B1
NO323597B1 NO20016154A NO20016154A NO323597B1 NO 323597 B1 NO323597 B1 NO 323597B1 NO 20016154 A NO20016154 A NO 20016154A NO 20016154 A NO20016154 A NO 20016154A NO 323597 B1 NO323597 B1 NO 323597B1
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NO
Norway
Prior art keywords
formula
compound
mmol
phenyl
solution
Prior art date
Application number
NO20016154A
Other languages
English (en)
Norwegian (no)
Other versions
NO20016154L (no
NO20016154D0 (no
Inventor
Bernhard Neises
Armin Walser
Hans-Ulrich Stilz
Olaf Ritzeler
Jr William Jerome Bock
Gary Alan Flynn
Original Assignee
Sanofi Aventis Deutschland
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE1999128424 external-priority patent/DE19928424A1/de
Priority claimed from DE2000106297 external-priority patent/DE10006297A1/de
Application filed by Sanofi Aventis Deutschland filed Critical Sanofi Aventis Deutschland
Publication of NO20016154D0 publication Critical patent/NO20016154D0/no
Publication of NO20016154L publication Critical patent/NO20016154L/no
Publication of NO323597B1 publication Critical patent/NO323597B1/no

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Psychiatry (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Vascular Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Luminescent Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
NO20016154A 1999-06-23 2001-12-17 Substituerte benzimidazoler, fremgangsmate for fremstilling av samme, farmasoytisk sammensetning innbefattende samme, anvendelse av samme for fremstilling av medikament og fremgangsmate for fremstilling av farmasoytisk middel. NO323597B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE1999128424 DE19928424A1 (de) 1999-06-23 1999-06-23 Substituierte Benzimidazole
DE2000106297 DE10006297A1 (de) 2000-02-12 2000-02-12 Substituierte Benzimidazole
PCT/EP2000/005340 WO2001000610A1 (de) 1999-06-23 2000-06-09 Substituierte benzimidazole

Publications (3)

Publication Number Publication Date
NO20016154D0 NO20016154D0 (no) 2001-12-17
NO20016154L NO20016154L (no) 2002-02-19
NO323597B1 true NO323597B1 (no) 2007-06-11

Family

ID=26004312

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20016154A NO323597B1 (no) 1999-06-23 2001-12-17 Substituerte benzimidazoler, fremgangsmate for fremstilling av samme, farmasoytisk sammensetning innbefattende samme, anvendelse av samme for fremstilling av medikament og fremgangsmate for fremstilling av farmasoytisk middel.

Country Status (29)

Country Link
US (1) US6358978B1 (cs)
EP (1) EP1194425B1 (cs)
JP (1) JP4763949B2 (cs)
KR (1) KR100718830B1 (cs)
CN (1) CN1168727C (cs)
AT (1) ATE301651T1 (cs)
AU (1) AU769350B2 (cs)
BR (1) BR0012450B1 (cs)
CA (1) CA2377085C (cs)
CZ (1) CZ302775B6 (cs)
DE (1) DE50010931D1 (cs)
DK (1) DK1194425T3 (cs)
EE (1) EE04813B1 (cs)
ES (1) ES2246240T3 (cs)
HK (1) HK1047582B (cs)
HR (1) HRP20010944B1 (cs)
HU (1) HU228466B1 (cs)
IL (1) IL147184A0 (cs)
ME (1) ME00370B (cs)
MX (1) MXPA01012283A (cs)
NO (1) NO323597B1 (cs)
NZ (1) NZ516348A (cs)
PL (1) PL206826B1 (cs)
PT (1) PT1194425E (cs)
RS (1) RS50340B (cs)
RU (1) RU2261248C2 (cs)
SI (1) SI1194425T1 (cs)
SK (1) SK286857B6 (cs)
WO (1) WO2001000610A1 (cs)

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