NO20043841L - 1-fenyl-2-heteroaryl-substituerte benzimidazolderivater, anvendelsen derav for fremstilling av legemidler benyttet i behandlingen av immunologiske sykdommer - Google Patents
1-fenyl-2-heteroaryl-substituerte benzimidazolderivater, anvendelsen derav for fremstilling av legemidler benyttet i behandlingen av immunologiske sykdommerInfo
- Publication number
- NO20043841L NO20043841L NO20043841A NO20043841A NO20043841L NO 20043841 L NO20043841 L NO 20043841L NO 20043841 A NO20043841 A NO 20043841A NO 20043841 A NO20043841 A NO 20043841A NO 20043841 L NO20043841 L NO 20043841L
- Authority
- NO
- Norway
- Prior art keywords
- benzimidazole derivatives
- preparation
- treatment
- heteroaryl
- phenyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Immunology (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pulmonology (AREA)
- Transplantation (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Det beskrives nye benzimidazolderivater, deres fremstilling og deres anvendelse for fremstilling av legemidler for behandling og forebygging av sykdommer som er assosiert med en mikroglieaktivering, og av T-celle-formidlede immunologiske sykdommer, samt farmasøytiske preparater som inneholder de nye benzimidazolderivater.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10207844A DE10207844A1 (de) | 2002-02-15 | 2002-02-15 | 1-Phenyl-2-heteroaryl-substituierte Benzimidazolderivate, deren Verwendung zur Herstellung von Arzneimitteln sowie diese Derivate enthaltende pharmazeutische Präparate |
PCT/EP2003/000462 WO2003068766A1 (de) | 2002-02-15 | 2003-01-17 | 1-phenyl-2-heteroaryl-substituierte benzimidazolderivate, deren verwendung zur herstellung von arzneimitteln zur behandlung von immunologischen erkrankungen |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20043841L true NO20043841L (no) | 2004-11-12 |
NO329667B1 NO329667B1 (no) | 2010-11-29 |
Family
ID=27674913
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20043841A NO329667B1 (no) | 2002-02-15 | 2004-09-14 | 1-fenyl-2-(pyridyl eller tienyl)-substituerte benzimidazolderivater, farmasoytiske preparater som inneholder forbindelsene og anvendelse av disse for fremstilling av legemidler benyttet for behandling av immunologiske sykdommer |
Country Status (30)
Country | Link |
---|---|
EP (1) | EP1474415B1 (no) |
JP (1) | JP4739675B2 (no) |
KR (1) | KR101027556B1 (no) |
CN (1) | CN1317274C (no) |
AR (1) | AR038492A1 (no) |
AT (1) | ATE517881T1 (no) |
AU (1) | AU2003205624B2 (no) |
BR (1) | BR0307723A (no) |
CA (1) | CA2475780C (no) |
CR (1) | CR7442A (no) |
CY (1) | CY1113230T1 (no) |
DE (1) | DE10207844A1 (no) |
DK (1) | DK1474415T3 (no) |
EC (1) | ECSP045296A (no) |
ES (1) | ES2369662T3 (no) |
IL (1) | IL163431A (no) |
MX (1) | MXPA04007949A (no) |
NO (1) | NO329667B1 (no) |
NZ (1) | NZ534660A (no) |
PE (1) | PE20030941A1 (no) |
PL (1) | PL216233B1 (no) |
PT (1) | PT1474415E (no) |
RS (1) | RS51831B (no) |
RU (1) | RU2325384C2 (no) |
SI (1) | SI1474415T1 (no) |
TW (1) | TWI328583B (no) |
UA (1) | UA81243C2 (no) |
UY (1) | UY27661A1 (no) |
WO (1) | WO2003068766A1 (no) |
ZA (1) | ZA200407381B (no) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1956004B1 (en) | 2002-03-27 | 2012-06-13 | Glaxo Group Limited | Quinoline derivatives and their use as 5-HT6 ligands |
CA2524054C (en) * | 2003-05-19 | 2012-04-24 | Irm Llc | Immunosuppressant compounds and compositions |
WO2014044611A1 (en) | 2012-09-20 | 2014-03-27 | Bayer Pharma Aktiengesellschaft | 1-aryl-2-heteroaryl benzimidazoles for the induction of neuronal regeneration |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE4330959A1 (de) * | 1993-09-09 | 1995-03-16 | Schering Ag | Neue Benzimidazolderivate, Verfahren zu ihrer Herstellung und ihre pharmazeutische Verwendung |
DK1246808T3 (da) * | 2000-01-14 | 2011-12-05 | Bayer Pharma AG | 1,2-diarylbenzimidazoler til behandling af sygdomme, som er associeret med en mikroglia-aktivering |
US7115645B2 (en) * | 2000-01-14 | 2006-10-03 | Schering Aktiengesellschaft | 1,2 diarylbenzimidazoles and their pharmaceutical use |
DE10207843A1 (de) * | 2002-02-15 | 2003-09-04 | Schering Ag | Mikrolia-Inhibitoren zur Unterbrechung von Interleukin 12 und IFN-gamma vermittelten Immunreaktionen |
-
2002
- 2002-02-15 DE DE10207844A patent/DE10207844A1/de not_active Ceased
-
2003
- 2003-01-17 WO PCT/EP2003/000462 patent/WO2003068766A1/de active Application Filing
- 2003-01-17 AT AT03702464T patent/ATE517881T1/de active
- 2003-01-17 KR KR1020047012576A patent/KR101027556B1/ko not_active IP Right Cessation
- 2003-01-17 SI SI200332061T patent/SI1474415T1/sl unknown
- 2003-01-17 RS YU71404A patent/RS51831B/en unknown
- 2003-01-17 AU AU2003205624A patent/AU2003205624B2/en not_active Ceased
- 2003-01-17 CA CA2475780A patent/CA2475780C/en not_active Expired - Fee Related
- 2003-01-17 DK DK03702464.3T patent/DK1474415T3/da active
- 2003-01-17 BR BR0307723-3A patent/BR0307723A/pt not_active IP Right Cessation
- 2003-01-17 RU RU2004127678/04A patent/RU2325384C2/ru not_active IP Right Cessation
- 2003-01-17 EP EP03702464A patent/EP1474415B1/de not_active Expired - Lifetime
- 2003-01-17 PT PT03702464T patent/PT1474415E/pt unknown
- 2003-01-17 PL PL371269A patent/PL216233B1/pl unknown
- 2003-01-17 UA UA20040907405A patent/UA81243C2/uk unknown
- 2003-01-17 ES ES03702464T patent/ES2369662T3/es not_active Expired - Lifetime
- 2003-01-17 NZ NZ534660A patent/NZ534660A/en not_active IP Right Cessation
- 2003-01-17 CN CNB038039974A patent/CN1317274C/zh not_active Expired - Fee Related
- 2003-01-17 MX MXPA04007949A patent/MXPA04007949A/es active IP Right Grant
- 2003-01-17 JP JP2003567893A patent/JP4739675B2/ja not_active Expired - Fee Related
- 2003-01-31 PE PE2003000110A patent/PE20030941A1/es not_active Application Discontinuation
- 2003-02-11 UY UY27661A patent/UY27661A1/es not_active Application Discontinuation
- 2003-02-12 AR ARP030100437A patent/AR038492A1/es not_active Application Discontinuation
- 2003-02-14 TW TW092103073A patent/TWI328583B/zh not_active IP Right Cessation
-
2004
- 2004-08-10 IL IL163431A patent/IL163431A/en not_active IP Right Cessation
- 2004-09-01 CR CR7442A patent/CR7442A/es not_active Application Discontinuation
- 2004-09-14 NO NO20043841A patent/NO329667B1/no not_active IP Right Cessation
- 2004-09-14 EC EC2004005296A patent/ECSP045296A/es unknown
- 2004-09-14 ZA ZA2004/07381A patent/ZA200407381B/en unknown
-
2011
- 2011-10-26 CY CY20111101016T patent/CY1113230T1/el unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
CHAD | Change of the owner's name or address (par. 44 patent law, par. patentforskriften) |
Owner name: BAYER INTELLECTUAL PROPERTY GMBH, DE |
|
MM1K | Lapsed by not paying the annual fees |