NO174775C - Analogifremgangsmåte til fremstilling av modifiserte gangliosider og deres funksjonelle derivater - Google Patents
Analogifremgangsmåte til fremstilling av modifiserte gangliosider og deres funksjonelle derivaterInfo
- Publication number
- NO174775C NO174775C NO904921A NO904921A NO174775C NO 174775 C NO174775 C NO 174775C NO 904921 A NO904921 A NO 904921A NO 904921 A NO904921 A NO 904921A NO 174775 C NO174775 C NO 174775C
- Authority
- NO
- Norway
- Prior art keywords
- preparation
- functional derivatives
- analogous procedure
- gangliosides
- modified gangliosides
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07G—COMPOUNDS OF UNKNOWN CONSTITUTION
- C07G99/00—Subject matter not provided for in other groups of this subclass
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
- C07H15/10—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical containing unsaturated carbon-to-carbon bonds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Molecular Biology (AREA)
- Crystallography & Structural Chemistry (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Hospice & Palliative Care (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT04855489A IT1238346B (it) | 1989-11-14 | 1989-11-14 | Gangliosidi modificati e loro derivati funzionali. |
Publications (4)
Publication Number | Publication Date |
---|---|
NO904921D0 NO904921D0 (no) | 1990-11-13 |
NO904921L NO904921L (no) | 1991-05-15 |
NO174775B NO174775B (no) | 1994-03-28 |
NO174775C true NO174775C (no) | 1994-07-06 |
Family
ID=11267289
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO904921A NO174775C (no) | 1989-11-14 | 1990-11-13 | Analogifremgangsmåte til fremstilling av modifiserte gangliosider og deres funksjonelle derivater |
Country Status (19)
Country | Link |
---|---|
US (2) | US5264424A (pt) |
EP (1) | EP0433112B1 (pt) |
JP (1) | JPH03170491A (pt) |
KR (1) | KR910009716A (pt) |
CN (1) | CN1033031C (pt) |
AR (1) | AR246527A1 (pt) |
AT (1) | ATE172737T1 (pt) |
AU (1) | AU645766B2 (pt) |
BR (1) | BR9005758A (pt) |
CA (1) | CA2029974A1 (pt) |
DE (1) | DE69032722T2 (pt) |
ES (1) | ES2124214T3 (pt) |
FI (1) | FI905628A0 (pt) |
HU (1) | HU210744B (pt) |
IL (1) | IL96344A0 (pt) |
IT (1) | IT1238346B (pt) |
NO (1) | NO174775C (pt) |
NZ (1) | NZ236057A (pt) |
PL (1) | PL287756A1 (pt) |
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5824662A (en) | 1996-09-27 | 1998-10-20 | Guilford Pharmaceuticals Inc. | Treatment of global and focal ischemia using naaladase inhibitors |
US6017903A (en) | 1996-09-27 | 2000-01-25 | Guilford Pharmaceuticals Inc. | Pharmaceutical compositions and methods of treating a glutamate abnormality and effecting a neuronal activity in an animal using NAALADase inhibitors |
US6413948B1 (en) | 1996-09-27 | 2002-07-02 | Guilford Pharmaceuticals Inc. | Pharmaceutical compositions and methods of effecting a neuronal activity in an animal using naaladase inhibitors |
Families Citing this family (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6407072B1 (en) * | 1988-12-02 | 2002-06-18 | Fidia S.P.A. | Lysoganglioside derivatives |
IT1232176B (it) * | 1989-07-27 | 1992-01-25 | Fidia Farmaceutici | Derivati di-lisogangliosidi |
IT1239060B (it) * | 1990-05-04 | 1993-09-20 | Fidia Spa | Processo per la modulazione selettiva dell'espressione e della funzione di un determinante sulla superficie cellulare attraverso appropriati agenti chimici |
IT1253832B (it) * | 1991-08-01 | 1995-08-29 | Fidia Spa | Derivati di gangliosidi |
IT1267955B1 (it) * | 1993-03-04 | 1997-02-18 | Fidia S P A In Amministrazione | Derivati solfatati dei lisogangliosidi |
US5849717A (en) * | 1993-03-04 | 1998-12-15 | Fidia S.P.A. | O-sulfated gangliosides and lyso-ganglioside derivatives |
IT1267956B1 (it) * | 1993-03-04 | 1997-02-18 | Fidia S P A In Amministrazione | Derivati o-solfatati di gangliosidi e lisogangliosidi |
US5973128A (en) * | 1996-11-22 | 1999-10-26 | The Hospital For Sick Children Research And Development Lp | Glycolipid mimics and methods of use thereof |
US7057057B2 (en) | 2002-05-22 | 2006-06-06 | Errant Gene Therapeutics, Llc | Histone deacetylase inhibitors based on alpha-ketoepoxide compounds |
US7312247B2 (en) | 2001-03-27 | 2007-12-25 | Errant Gene Therapeutics, Llc | Histone deacetylase inhibitors |
US8026280B2 (en) | 2001-03-27 | 2011-09-27 | Errant Gene Therapeutics, Llc | Histone deacetylase inhibitors |
US7842727B2 (en) | 2001-03-27 | 2010-11-30 | Errant Gene Therapeutics, Llc | Histone deacetylase inhibitors |
US6495719B2 (en) | 2001-03-27 | 2002-12-17 | Circagen Pharmaceutical | Histone deacetylase inhibitors |
NZ531139A (en) * | 2001-08-29 | 2007-09-28 | Neose Technologies Inc | Synthetic ganglioside derivatives and compositions thereof |
WO2004046104A2 (en) | 2002-11-20 | 2004-06-03 | Errant Gene Therapeutics, Llc | Treatment of lung cells with histone deacetylase inhibitors |
NZ542148A (en) * | 2003-03-06 | 2008-05-30 | Neose Technologies Inc | Methods and compositions for the enzymatic synthesis of gangliosides |
WO2005033700A1 (ja) * | 2003-10-03 | 2005-04-14 | Takeda Pharmaceutical Company Limited | インスリン抵抗性改善剤のスクリーニング方法 |
CN102151897B (zh) * | 2004-04-15 | 2013-06-19 | 密尔沃基电动工具公司 | 动力工具 |
US7932236B2 (en) * | 2004-11-09 | 2011-04-26 | Seneb Biosciences, Inc. | Glycolipids |
WO2009006591A1 (en) | 2007-07-03 | 2009-01-08 | Children's Hospital & Research Center At Oakland | Inhibitors of polysialic acid de-n-acetylase and methods for using the same |
EP2183261A4 (en) * | 2007-07-03 | 2010-09-15 | Childrens Hosp & Res Ct Oak | POLYSIALYLIC ACID DERIVATIVES, MANUFACTURING METHODS AND APPLICATIONS FOR INCREASING THE PRODUCTION AND TARGETING OF CANCER ANIMALS |
WO2009006620A1 (en) | 2007-07-03 | 2009-01-08 | Children's Hospital & Research Center At Oakland | Oligosialic acid derivatives, methods of manufacture, and immunological uses |
EP3175857A1 (en) | 2009-03-25 | 2017-06-07 | Seneb Biosciences Inc. | Glycolipids as treatment for disease |
CN109721632B (zh) * | 2017-10-27 | 2023-10-31 | 齐鲁制药有限公司 | 一种高纯度神经节苷脂gm1及其制备方法 |
US20210353659A1 (en) * | 2018-08-24 | 2021-11-18 | Industry-Academic Cooperation Foundation, Yonsei University | Composition for preventing or treating muscular diseases, or for improving muscular functions, containing gagnlioside |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1046051B (it) * | 1975-08-13 | 1980-06-30 | Fidia Spa | Nuova applicazione terapeutica dei gangliosidi e procedimento per la loro estrazione |
IT1171432B (it) * | 1981-08-03 | 1987-06-10 | Fidia Farmaceutici | Amidi organiche derivate da lipidi azotati utilizzabili come farmaci |
US4476119A (en) * | 1981-08-04 | 1984-10-09 | Fidia S.P.A. | Method for preparing ganglioside derivatives and use thereof in pharmaceutical compositions |
US4716223A (en) * | 1981-08-04 | 1987-12-29 | Fidia, S.P.A. | Method for preparing ganglioside derivatives and use thereof in pharmaceutical compositions |
US4593091A (en) * | 1981-08-04 | 1986-06-03 | Fidia, S.P.A. | Method for preparing ganglioside derivatives and use thereof in pharmaceutical compositions |
IT1199116B (it) * | 1984-07-03 | 1988-12-30 | Fidia Farmaceutici | Derivati di gangliosidi |
IT1182209B (it) * | 1985-02-18 | 1987-09-30 | Fidia Farmaceutici | Uso terapeutico del monosialoganglioside gm1 e dei suoi derivati in gravi patologie di infarti cerebrali |
IT1235161B (it) * | 1988-12-02 | 1992-06-22 | Fidia Farmaceutici | Derivati di lisogangliosidi |
IT1232176B (it) * | 1989-07-27 | 1992-01-25 | Fidia Farmaceutici | Derivati di-lisogangliosidi |
-
1989
- 1989-11-14 IT IT04855489A patent/IT1238346B/it active IP Right Grant
-
1990
- 1990-11-13 NO NO904921A patent/NO174775C/no unknown
- 1990-11-13 BR BR909005758A patent/BR9005758A/pt not_active Application Discontinuation
- 1990-11-13 US US07/611,700 patent/US5264424A/en not_active Expired - Fee Related
- 1990-11-13 NZ NZ236057A patent/NZ236057A/en unknown
- 1990-11-14 AU AU66624/90A patent/AU645766B2/en not_active Ceased
- 1990-11-14 FI FI905628A patent/FI905628A0/fi not_active Application Discontinuation
- 1990-11-14 DE DE69032722T patent/DE69032722T2/de not_active Expired - Fee Related
- 1990-11-14 KR KR1019900018389A patent/KR910009716A/ko not_active Application Discontinuation
- 1990-11-14 JP JP2310149A patent/JPH03170491A/ja active Pending
- 1990-11-14 CN CN90109290A patent/CN1033031C/zh not_active Expired - Fee Related
- 1990-11-14 AR AR90318382A patent/AR246527A1/es active
- 1990-11-14 PL PL28775690A patent/PL287756A1/xx unknown
- 1990-11-14 IL IL96344A patent/IL96344A0/xx unknown
- 1990-11-14 ES ES90403220T patent/ES2124214T3/es not_active Expired - Lifetime
- 1990-11-14 HU HU907124A patent/HU210744B/hu not_active IP Right Cessation
- 1990-11-14 CA CA002029974A patent/CA2029974A1/en not_active Abandoned
- 1990-11-14 AT AT90403220T patent/ATE172737T1/de not_active IP Right Cessation
- 1990-11-14 EP EP90403220A patent/EP0433112B1/en not_active Expired - Lifetime
-
1993
- 1993-10-20 US US08/138,184 patent/US5424294A/en not_active Expired - Fee Related
Cited By (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5824662A (en) | 1996-09-27 | 1998-10-20 | Guilford Pharmaceuticals Inc. | Treatment of global and focal ischemia using naaladase inhibitors |
US5985855A (en) | 1996-09-27 | 1999-11-16 | Guilford Pharmaceuticals Inc. | Treatment of global and focal ischemia using NAALADase inhibitors |
US6004946A (en) | 1996-09-27 | 1999-12-21 | Guilford Pharmaceuticals Inc. | Treatment of global and focal ischemia using naaladase inhibitors |
US6017903A (en) | 1996-09-27 | 2000-01-25 | Guilford Pharmaceuticals Inc. | Pharmaceutical compositions and methods of treating a glutamate abnormality and effecting a neuronal activity in an animal using NAALADase inhibitors |
US6413948B1 (en) | 1996-09-27 | 2002-07-02 | Guilford Pharmaceuticals Inc. | Pharmaceutical compositions and methods of effecting a neuronal activity in an animal using naaladase inhibitors |
Also Published As
Publication number | Publication date |
---|---|
DE69032722T2 (de) | 1999-07-08 |
ATE172737T1 (de) | 1998-11-15 |
PL287756A1 (en) | 1991-12-02 |
JPH03170491A (ja) | 1991-07-24 |
NO904921D0 (no) | 1990-11-13 |
EP0433112A1 (en) | 1991-06-19 |
US5264424A (en) | 1993-11-23 |
HU210744B (en) | 1995-07-28 |
BR9005758A (pt) | 1991-09-24 |
DE69032722D1 (de) | 1998-12-03 |
HUT55403A (en) | 1991-05-28 |
US5424294A (en) | 1995-06-13 |
CN1033031C (zh) | 1996-10-16 |
KR910009716A (ko) | 1991-06-28 |
AU645766B2 (en) | 1994-01-27 |
IL96344A0 (en) | 1991-08-16 |
ES2124214T3 (es) | 1999-02-01 |
CA2029974A1 (en) | 1991-05-15 |
NO174775B (no) | 1994-03-28 |
IT8948554A0 (it) | 1989-11-14 |
NO904921L (no) | 1991-05-15 |
NZ236057A (en) | 1994-09-27 |
IT1238346B (it) | 1993-07-13 |
FI905628A0 (fi) | 1990-11-14 |
CN1051912A (zh) | 1991-06-05 |
IT8948554A1 (it) | 1991-05-14 |
EP0433112B1 (en) | 1998-10-28 |
AU6662490A (en) | 1991-05-23 |
AR246527A1 (es) | 1994-08-31 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NO174775C (no) | Analogifremgangsmåte til fremstilling av modifiserte gangliosider og deres funksjonelle derivater | |
DK166084C (da) | Imidazoquinolinyletherderivater og fremgangsmaade til deres fremstilling | |
NO881344D0 (no) | Fremgangsmaate til fremstilling av kvaternaere esteraminer og deres anvendelse. | |
DK195587D0 (da) | Phenylpiperazinderivater og deres anvendelse til fremstilling af antiarrytmi-laegemidler | |
NO167092C (no) | Fremgangsmaate og sukrosederivat til fremstilling av sukrose-6-acylater. | |
MX9101793A (es) | Derivados de tiazolidindiona y procedimiento para su preparacion | |
NO171208C (no) | Fremgangsmaate for fremstilling av eventuelt kvaterniserteestere og deres anvendelse | |
DK397388A (da) | Derivater af n-aminobutyl-n-phenylarylamider til terapeutisk anvendelse samt fremgangsmaade til fremstilling af saadanne derivater | |
DK631587D0 (da) | Imidazolderivater og fremgangsmaade til deres fremstilling | |
NO173604C (no) | Analogifremgangsmaate til fremstilling av bis-dioksopiperazinderivater | |
NO882940D0 (no) | Fremgangsmaate for fremstilling av castanosperminestere og glycosider. | |
NO900643D0 (no) | Fremgangsmaate for fremstilling og anvendelse av 2,3,23-trihydroksi-urs-12-ener og deres derivater. | |
NO894185D0 (no) | Fremgangsmaate for fremstilling av 1-buten- og/eller heksener. | |
NO891985D0 (no) | Fremgangsmaate for fremstilling av dibenzotiofen- og tioxanten-derivater. | |
NO904805D0 (no) | Fremgangsmaate for fremstilling av antihypertensive og antiarytmiske pyridinderivater. | |
MX9100367A (es) | Derivados de heteroarilcetona y procedimiento para su preparacion | |
NO905543D0 (no) | Fremgangsmaate for fremstilling og anvendelse av aminopyridinylmetanoler og aminometylpyridinaminer. | |
NO901732D0 (no) | Fremgangsmaate for fremstilling av 4-alkoksyalkyl-4-aminofenylpiperidiner og derivater derav. | |
NO921168L (no) | Fremgangsmaate og anordning for fremstilling av elementaertjod i ren form | |
NO904588L (no) | Fremgangsmaate til fremstilling av diazinylpiperidin-derivater | |
MX9100388A (es) | Derivados de carboximetilciclopropano y procedimiento para su preparacion | |
MX19566A (es) | Nuevos derivados de 1-arilsulfonil-pirrolidin-2-tiona o de 1-arilsulfonil-piperidin-2-tiona y procedimiento para su preparacion | |
MX17198A (es) | Derivados de benzazola y procedimiento para su preparacion | |
NO921313D0 (no) | Derivater av 2-spirocyklopropylcefalosporinsulfoner og deres fremstilling | |
MX6550A (es) | Derivados de tetrahidronaftalina e indeno y procedimiento para su preparacion. |