NL8800998A - Werkwijze voor het bereiden van een al of niet gesubstitueerd 4(5)-(omega-aminoalkyl) imidazool. - Google Patents

Werkwijze voor het bereiden van een al of niet gesubstitueerd 4(5)-(omega-aminoalkyl) imidazool. Download PDF

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Publication number
NL8800998A
NL8800998A NL8800998A NL8800998A NL8800998A NL 8800998 A NL8800998 A NL 8800998A NL 8800998 A NL8800998 A NL 8800998A NL 8800998 A NL8800998 A NL 8800998A NL 8800998 A NL8800998 A NL 8800998A
Authority
NL
Netherlands
Prior art keywords
ppm
singlet
filtered
imidazole
concentrated
Prior art date
Application number
NL8800998A
Other languages
English (en)
Dutch (nl)
Original Assignee
Cedona Pharm Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cedona Pharm Bv filed Critical Cedona Pharm Bv
Priority to NL8800998A priority Critical patent/NL8800998A/nl
Priority to PCT/NL1989/000019 priority patent/WO1989010360A1/en
Priority to AU34308/89A priority patent/AU632044B2/en
Priority to JP1504592A priority patent/JPH03504853A/ja
Priority to HU892601A priority patent/HU206088B/hu
Priority to US07/573,015 priority patent/US5190589A/en
Priority to EP89904857A priority patent/EP0415948A1/en
Publication of NL8800998A publication Critical patent/NL8800998A/nl
Priority to NO90904486A priority patent/NO904486L/no
Priority to FI905127A priority patent/FI905127A0/fi
Priority to DK250290A priority patent/DK250290A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NL8800998A 1988-04-18 1988-04-18 Werkwijze voor het bereiden van een al of niet gesubstitueerd 4(5)-(omega-aminoalkyl) imidazool. NL8800998A (nl)

Priority Applications (10)

Application Number Priority Date Filing Date Title
NL8800998A NL8800998A (nl) 1988-04-18 1988-04-18 Werkwijze voor het bereiden van een al of niet gesubstitueerd 4(5)-(omega-aminoalkyl) imidazool.
PCT/NL1989/000019 WO1989010360A1 (en) 1988-04-18 1989-04-05 PROCESS FOR PREPARING A SUBSTITUTED OR AN UNSUBSTITUTED 4(5)-(omega-AMINOALKYL)IMIDAZOLE
AU34308/89A AU632044B2 (en) 1988-04-18 1989-04-05 Process for preparing a substituted or an unsubstituted 4(5)-(omega-aminoalkyl)imidazole
JP1504592A JPH03504853A (ja) 1988-04-18 1989-04-05 置換または未置換4(5)―(ω―アミノアルキル)イミダゾールの製造方法
HU892601A HU206088B (en) 1988-04-18 1989-04-05 Process for produicng 4(5)-(aminoalkyl)-imidazole derivatives
US07/573,015 US5190589A (en) 1988-04-18 1989-04-05 Compounds and process preparing a substituted or an unsubstituted 4(5)-(ω-aminoalkyl)imidazole
EP89904857A EP0415948A1 (en) 1988-04-18 1989-04-05 PROCESS FOR PREPARING A SUBSTITUTED OR AN UNSUBSTITUTED 4(5)-($g(v)-AMINOALKYL)IMIDAZOLE
NO90904486A NO904486L (no) 1988-04-18 1990-10-17 Fremgangsmaate til fremstilling av en substituert eller enusubstituert 4(5)-(omega-aminoalkyl)imidazol.
FI905127A FI905127A0 (fi) 1988-04-18 1990-10-17 Foerfarande foer framstaellning av en substituerad eller osubstituerad 4(5)-(omega-aminoalkyl)imidazol.
DK250290A DK250290A (da) 1988-04-18 1990-10-17 Substituerede eller usubstituerede 4(5)-(omega-aminoalkyl)imidazoler, fremgangsmaade til fremstilling heraf og farmaceutiske praeparater indeholdende disse forbindelser

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
NL8800998A NL8800998A (nl) 1988-04-18 1988-04-18 Werkwijze voor het bereiden van een al of niet gesubstitueerd 4(5)-(omega-aminoalkyl) imidazool.
NL8800998 1988-04-18

Publications (1)

Publication Number Publication Date
NL8800998A true NL8800998A (nl) 1989-11-16

Family

ID=19852148

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8800998A NL8800998A (nl) 1988-04-18 1988-04-18 Werkwijze voor het bereiden van een al of niet gesubstitueerd 4(5)-(omega-aminoalkyl) imidazool.

Country Status (9)

Country Link
US (1) US5190589A (da)
EP (1) EP0415948A1 (da)
JP (1) JPH03504853A (da)
AU (1) AU632044B2 (da)
DK (1) DK250290A (da)
FI (1) FI905127A0 (da)
HU (1) HU206088B (da)
NL (1) NL8800998A (da)
WO (1) WO1989010360A1 (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL9000132A (nl) * 1990-01-19 1991-08-16 Cedona Pharm Bv Nieuwe thiazoolderivaten.
US5159083A (en) * 1990-12-28 1992-10-27 Neurogen Corporation Certain aminomethyl phenylimidazole derivatives; a class of dopamine receptor subtype specific ligands
US5646281A (en) * 1990-12-28 1997-07-08 Neurogen Corporation Certain 4-piperidino- and piperazinomethyl-2-phenyl imidazole derivatives; dopamine receptor subtype specific ligands
FR2686084B1 (fr) * 1992-01-10 1995-12-22 Bioprojet Soc Civ Nouveaux derives de l'imidazole, leur preparation et leurs applications therapeutiques.
USRE37303E1 (en) * 1992-01-10 2001-07-31 Institut National Del La Sante Et De La Recherche Medicale Imidazole compounds and their therapeutic applications
US5971979A (en) * 1997-12-02 1999-10-26 Odyssey Technologies, Inc. Method for cryogenic inhibition of hyperplasia
WO2000039098A1 (en) 1998-12-23 2000-07-06 Maxim Pharmaceuticals, Inc. Synthesis of histamine dihydrochloride
EP1741709A1 (en) * 2005-06-28 2007-01-10 Sanofi-Aventis Deutschland GmbH Heteroaryl-substituted amides comprising a saturated linker group, and their use as pharmaceuticals
JP5463055B2 (ja) * 2009-02-27 2014-04-09 公益財団法人相模中央化学研究所 フタルイミド誘導体及びそれらの製造方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE758146A (fr) * 1969-10-29 1971-04-28 Smith Kline French Lab Derives de l'amidine
GB1570212A (en) * 1975-10-29 1980-06-25 Smithkline Corp Imidazoles

Also Published As

Publication number Publication date
WO1989010360A1 (en) 1989-11-02
FI905127A0 (fi) 1990-10-17
AU3430889A (en) 1989-11-24
AU632044B2 (en) 1992-12-17
US5190589A (en) 1993-03-02
HU206088B (en) 1992-08-28
DK250290A (da) 1990-12-04
HU892601D0 (en) 1991-05-28
HUT55762A (en) 1991-06-28
JPH03504853A (ja) 1991-10-24
EP0415948A1 (en) 1991-03-13
DK250290D0 (da) 1990-10-17

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BV The patent application has lapsed