NL194240C - Lincomycine en clindamycine-analoga. - Google Patents

Lincomycine en clindamycine-analoga. Download PDF

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Publication number
NL194240C
NL194240C NL8006229A NL8006229A NL194240C NL 194240 C NL194240 C NL 194240C NL 8006229 A NL8006229 A NL 8006229A NL 8006229 A NL8006229 A NL 8006229A NL 194240 C NL194240 C NL 194240C
Authority
NL
Netherlands
Prior art keywords
formula
group
substituted
acid
compound
Prior art date
Application number
NL8006229A
Other languages
English (en)
Dutch (nl)
Other versions
NL194240B (nl
NL8006229A (nl
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of NL8006229A publication Critical patent/NL8006229A/nl
Publication of NL194240B publication Critical patent/NL194240B/xx
Application granted granted Critical
Publication of NL194240C publication Critical patent/NL194240C/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
    • C07H15/06—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical being a hydroxyalkyl group esterified by a fatty acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
    • C07H15/16—Lincomycin; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
NL8006229A 1979-11-23 1980-11-14 Lincomycine en clindamycine-analoga. NL194240C (nl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US9665279A 1979-11-23 1979-11-23
US9665279 1979-11-23
US14805680 1980-05-19
US06/148,056 US4278789A (en) 1979-11-23 1980-05-19 Lincomycin compounds

Publications (3)

Publication Number Publication Date
NL8006229A NL8006229A (nl) 1981-06-16
NL194240B NL194240B (nl) 2001-06-01
NL194240C true NL194240C (nl) 2001-10-02

Family

ID=26791923

Family Applications (2)

Application Number Title Priority Date Filing Date
NL8006229A NL194240C (nl) 1979-11-23 1980-11-14 Lincomycine en clindamycine-analoga.
NL300064C NL300064I2 (nl) 1979-11-23 2001-10-02 Lincomycine en clindamycine-analoga.

Family Applications After (1)

Application Number Title Priority Date Filing Date
NL300064C NL300064I2 (nl) 1979-11-23 2001-10-02 Lincomycine en clindamycine-analoga.

Country Status (16)

Country Link
US (1) US4278789A (de)
KR (1) KR850000065B1 (de)
AU (1) AU535986B2 (de)
CA (1) CA1165315A (de)
CH (1) CH647244A5 (de)
DE (1) DE3043502A1 (de)
ES (1) ES8204442A1 (de)
FR (4) FR2470134B1 (de)
GB (1) GB2063252B (de)
HU (2) HU190437B (de)
IL (1) IL61245A (de)
IT (1) IT1134065B (de)
NL (2) NL194240C (de)
PL (2) PL228054A1 (de)
SE (1) SE447260B (de)
SU (1) SU1169543A3 (de)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4383109A (en) * 1981-04-20 1983-05-10 The Upjohn Company Lincomycin nucleotides
US4368193A (en) * 1981-04-20 1983-01-11 The Upjohn Company Process for treating malaria
US4393054A (en) * 1982-05-19 1983-07-12 The Upjohn Company Method of treating cardiac arrhythmia
US4430495A (en) 1982-09-17 1984-02-07 The Upjohn Company Process for preparing lincomycin and clindamycin ribonucleotides
ATE69142T1 (de) * 1987-05-19 1991-11-15 Upjohn Co Pirlimycin wachstumsteigerndes mittel fuer fleischproduzierende tiere.
TW282399B (de) * 1990-05-25 1996-08-01 Takeda Pharm Industry Co Ltd
CN100350036C (zh) * 2001-04-27 2007-11-21 宝洁公司 用于控制生物膜的装置和方法
US7049339B2 (en) * 2001-06-15 2006-05-23 Forty Eight Shelf (80) Limited Composition for the treatment of diseases which affect animals' hooves
ES2243763T3 (es) * 2001-08-28 2005-12-01 Pharmacia Corporation Base libre de clindamicina cristalina.
US7199105B2 (en) * 2002-08-15 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
KR20050056195A (ko) * 2002-08-15 2005-06-14 비큐론 파마슈티컬스 인코포레이티드 항박테리아 작용을 갖는 링코마이신 유도체
US7199106B2 (en) 2003-06-17 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antimicrobial activity
CA2528592A1 (en) * 2003-06-17 2005-02-10 Vicuron Pharmaceuticals Inc. Novel lincomycin derivatives possessing antimicrobial activity
US7256177B2 (en) 2003-06-17 2007-08-14 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
US7361743B2 (en) * 2004-02-11 2008-04-22 Pfizer Inc Lincomycin derivatives possessing antibacterial activity
CN100404543C (zh) * 2006-09-21 2008-07-23 浙江海正药业股份有限公司 一种合成吡利霉素的中间体及其制备方法和用途
CA2871766C (en) * 2011-12-08 2020-06-16 The Board Of Regents Of The University Of Texas System Piperidine-based small molecule 5-hydroxytryptamine 2c receptor (5-ht2cr) allosteric modulators

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3086912A (en) * 1961-07-03 1963-04-23 Upjohn Co Antibiotic lincolnensin and method of production
US3496163A (en) * 1965-02-08 1970-02-17 Upjohn Co 7-halo-7-deoxylincomycins and process for preparing the same
US3758454A (en) * 1971-03-12 1973-09-11 Upjohn Co Lincomycin type compounds and process for making them
US3853843A (en) * 1972-12-13 1974-12-10 Upjohn Co Derivatives of thiolincosaminide compounds

Also Published As

Publication number Publication date
NL300064I1 (nl) 2001-12-01
NL300064I2 (nl) 2002-01-02
AU6344380A (en) 1981-05-28
PL228054A1 (en) 1983-05-09
FR2487358A1 (fr) 1982-01-29
AU535986B2 (en) 1984-04-12
ES496988A0 (es) 1982-05-01
CA1165315A (en) 1984-04-10
SU1169543A3 (ru) 1985-07-23
HU190437B (en) 1986-09-29
KR830004332A (ko) 1983-07-09
FR2493852B1 (fr) 1985-08-16
CH647244A5 (de) 1985-01-15
GB2063252B (en) 1983-05-18
FR2491072A1 (fr) 1982-04-02
NL194240B (nl) 2001-06-01
IT8025607A0 (it) 1980-10-27
FR2470134B1 (fr) 1985-07-26
US4278789A (en) 1981-07-14
FR2493852A1 (fr) 1982-05-14
PL233258A1 (en) 1983-05-09
FR2470134A1 (fr) 1981-05-29
KR850000065B1 (ko) 1985-02-15
GB2063252A (en) 1981-06-03
IT1134065B (it) 1986-07-24
IL61245A0 (en) 1980-12-31
SE447260B (sv) 1986-11-03
IL61245A (en) 1986-07-31
ES8204442A1 (es) 1982-05-01
DE3043502A1 (de) 1981-06-04
DE3043502C2 (de) 1989-05-11
NL8006229A (nl) 1981-06-16
HU187281B (en) 1985-12-28
SE8008181L (sv) 1981-05-24
PL132002B1 (en) 1985-01-31

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
DNT Communications of changes of names of applicants whose applications have been laid open to public inspection

Free format text: PHARMACIA & UPJOHN COMPANY

AC1 Application for a supplementary protection certificate

Free format text: 300064, 20011002

V4 Discontinued because of reaching the maximum lifetime of a patent

Free format text: 20011002

KC1 Grant of a supplementary protection certificate

Free format text: 300064, 20001114, EXPIRES: 20051113