NI200600306A - Derivados de sulfamida y sulfamato para el tratamiento de la epilepsia y trastornos relacionados - Google Patents
Derivados de sulfamida y sulfamato para el tratamiento de la epilepsia y trastornos relacionadosInfo
- Publication number
- NI200600306A NI200600306A NI200600306A NI200600306A NI200600306A NI 200600306 A NI200600306 A NI 200600306A NI 200600306 A NI200600306 A NI 200600306A NI 200600306 A NI200600306 A NI 200600306A NI 200600306 A NI200600306 A NI 200600306A
- Authority
- NI
- Nicaragua
- Prior art keywords
- epilepsy
- treatment
- sulfamide
- related disorders
- sulfamate derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
- C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
- C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D319/20—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
- C07D317/58—Radicals substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D321/00—Heterocyclic compounds containing rings having two oxygen atoms as the only ring hetero atoms, not provided for by groups C07D317/00 - C07D319/00
- C07D321/02—Seven-membered rings
- C07D321/10—Seven-membered rings condensed with carbocyclic rings or ring systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrane Compounds (AREA)
Abstract
La presente invención está dirigida a nuevos derivados de sulfamida y sulfamato, composiciones farmacéuticas que las contienen y sus usos en el tratamiento de la epilepsia y trastornos relacionados.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US58017804P | 2004-06-16 | 2004-06-16 |
Publications (1)
Publication Number | Publication Date |
---|---|
NI200600306A true NI200600306A (es) | 2007-11-27 |
Family
ID=34972935
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NI200600306A NI200600306A (es) | 2004-06-16 | 2006-12-15 | Derivados de sulfamida y sulfamato para el tratamiento de la epilepsia y trastornos relacionados |
Country Status (22)
Country | Link |
---|---|
US (1) | US8084490B2 (es) |
EP (1) | EP1768970B1 (es) |
JP (2) | JP4884378B2 (es) |
CN (1) | CN101006072B (es) |
AR (2) | AR049398A1 (es) |
AU (1) | AU2005262496B2 (es) |
BR (1) | BRPI0512242A (es) |
CA (1) | CA2570606C (es) |
CR (1) | CR8858A (es) |
EA (1) | EA013685B1 (es) |
EC (1) | ECSP067093A (es) |
ES (1) | ES2573844T3 (es) |
IL (1) | IL180108A (es) |
MX (1) | MXPA06014934A (es) |
MY (1) | MY147767A (es) |
NI (1) | NI200600306A (es) |
NO (1) | NO20070081L (es) |
NZ (1) | NZ552056A (es) |
TW (1) | TWI361691B (es) |
UA (1) | UA91680C2 (es) |
WO (1) | WO2006007435A1 (es) |
ZA (1) | ZA200700430B (es) |
Families Citing this family (33)
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TW200612905A (en) * | 2004-06-16 | 2006-05-01 | Janssen Pharmaceutica Nv | Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders |
MY147767A (en) * | 2004-06-16 | 2013-01-31 | Janssen Pharmaceutica Nv | Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders |
ES2310366T3 (es) * | 2004-08-24 | 2009-01-01 | Janssen Pharmaceutica Nv | Nuevos derivados de heteroaril sulfonamida benzo-condensada utiles como agentes anticonvulsivos. |
CA2609185A1 (en) * | 2005-05-20 | 2006-11-30 | Ahmed F. Abdel-Magid | Process for preparation of sulfamide derivatives |
US8691867B2 (en) | 2005-12-19 | 2014-04-08 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction |
US8497298B2 (en) * | 2005-12-19 | 2013-07-30 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels |
US8716231B2 (en) * | 2005-12-19 | 2014-05-06 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain |
US20070155827A1 (en) * | 2005-12-19 | 2007-07-05 | Smith-Swintosky Virginia L | Use of benzo-fused heterocycle sulfamide derivatives for the treatment of depression |
US8937096B2 (en) | 2005-12-19 | 2015-01-20 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder |
AR058389A1 (es) * | 2005-12-19 | 2008-01-30 | Janssen Pharmaceutica Nv | Uso de derivados heterociclicos benzo-fusionados de sulfamida para el tratamiento de la obesidad |
US20070155824A1 (en) * | 2005-12-19 | 2007-07-05 | Smith-Swintosky Virginia L | Use of benzo-fused heterocycle sulfamide derivatives for disease modification / epileptogenesis |
TWI398248B (zh) * | 2005-12-19 | 2013-06-11 | Janssen Pharmaceutica Nv | 苯并稠合雜環磺醯胺衍生物於保護及恢復性治療/癲癇產生之用途 |
US20070191474A1 (en) * | 2006-02-15 | 2007-08-16 | Smith-Swintosky Virginia L | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of migraine |
EA200870556A1 (ru) * | 2006-05-19 | 2009-06-30 | Янссен Фармацевтика Н.В. | Комбинированная терапия в лечении эпилепсии и родственных расстройств |
WO2009089210A1 (en) * | 2008-01-07 | 2009-07-16 | Janssen Pharmaceutica N. V. | Preparation of sulfamide derivatives |
EP2280950A1 (en) * | 2008-03-26 | 2011-02-09 | Janssen Pharmaceutica, N.V. | Process for the preparation of benzo-fused heteroaryl sulfamates and crystalline form of n- ( ( (2s) -6-chloro-2,3-dihydro-l,4-benzodioxin-2-yl) methyl-sulfamide |
CN101981023A (zh) * | 2008-03-26 | 2011-02-23 | 詹森药业有限公司 | 用于制备苯并稠合二噁英衍生物的方法 |
US20090247616A1 (en) * | 2008-03-26 | 2009-10-01 | Smith-Swintosky Virginia L | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of anxiety |
US20090247617A1 (en) * | 2008-03-26 | 2009-10-01 | Abdel-Magid Ahmed F | Process for the preparation of benzo-fused heteroaryl sulfamates |
CN102015674B (zh) * | 2008-04-29 | 2014-10-29 | Nsab神经研究瑞典公司分公司 | 多巴胺神经传递调节剂 |
AU2009242092A1 (en) * | 2008-04-29 | 2009-11-05 | Nsab, Filial Af Neurosearch Sweden Ab, Sverige | Modulators of dopamine neurotransmission |
JP2011519839A (ja) * | 2008-04-29 | 2011-07-14 | エヌエスエイビー、フィリアル アヴ ノイロサーチ スウェーデン エービー、スヴェーリエ | ドーパミン神経伝達のモジュレーター |
WO2010008776A2 (en) * | 2008-06-23 | 2010-01-21 | Janssen Pharmaceutica Nv | Disposable patch and reusable sensor assembly for use in medical device localization and mapping systems |
US8815939B2 (en) * | 2008-07-22 | 2014-08-26 | Janssen Pharmaceutica Nv | Substituted sulfamide derivatives |
US20120263714A1 (en) * | 2009-10-21 | 2012-10-18 | Bayer Intellectual Property Gmbh | Substituted halophenoxybenzamide derivatives |
US8609849B1 (en) | 2010-11-30 | 2013-12-17 | Fox Chase Chemical Diversity Center, Inc. | Hydroxylated sulfamides exhibiting neuroprotective action and their method of use |
CA2850015A1 (en) * | 2011-09-29 | 2013-04-04 | Janssen Pharmaceutica Nv | Improved process for the preparation of sulfamide derivatives |
CA2850513A1 (en) | 2011-09-29 | 2013-04-04 | Janssen Pharmaceutica Nv | Process for the preparation of sulfamide derivatives |
WO2014140220A1 (en) | 2013-03-13 | 2014-09-18 | Janssen Pharmaceutica, N.V. | Process for the preparation of (2,3-dihydro-benzo[b][1,4]dioxin-2-yl) methanol derivatives |
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2005
- 2005-06-14 MY MYPI20052699A patent/MY147767A/en unknown
- 2005-06-15 AR ARP050102445A patent/AR049398A1/es active IP Right Grant
- 2005-06-15 TW TW094119737A patent/TWI361691B/zh not_active IP Right Cessation
- 2005-06-16 ES ES05763399.2T patent/ES2573844T3/es active Active
- 2005-06-16 BR BRPI0512242-2A patent/BRPI0512242A/pt active Search and Examination
- 2005-06-16 EP EP05763399.2A patent/EP1768970B1/en active Active
- 2005-06-16 EA EA200700035A patent/EA013685B1/ru not_active IP Right Cessation
- 2005-06-16 CN CN2005800274918A patent/CN101006072B/zh not_active Expired - Fee Related
- 2005-06-16 CA CA2570606A patent/CA2570606C/en not_active Expired - Fee Related
- 2005-06-16 WO PCT/US2005/021513 patent/WO2006007435A1/en active Application Filing
- 2005-06-16 UA UAA200613517A patent/UA91680C2/ru unknown
- 2005-06-16 JP JP2007516788A patent/JP4884378B2/ja not_active Expired - Fee Related
- 2005-06-16 US US11/154,443 patent/US8084490B2/en not_active Expired - Fee Related
- 2005-06-16 AU AU2005262496A patent/AU2005262496B2/en not_active Ceased
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- 2005-06-16 MX MXPA06014934A patent/MXPA06014934A/es active IP Right Grant
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- 2006-12-14 IL IL180108A patent/IL180108A/en not_active IP Right Cessation
- 2006-12-15 NI NI200600306A patent/NI200600306A/es unknown
- 2006-12-18 EC EC2006007093A patent/ECSP067093A/es unknown
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2007
- 2007-01-05 NO NO20070081A patent/NO20070081L/no not_active Application Discontinuation
- 2007-01-15 CR CR8858A patent/CR8858A/es not_active Application Discontinuation
- 2007-01-15 ZA ZA200700430A patent/ZA200700430B/en unknown
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Also Published As
Publication number | Publication date |
---|---|
ZA200700430B (en) | 2008-07-30 |
WO2006007435A1 (en) | 2006-01-19 |
TWI361691B (en) | 2012-04-11 |
AR049398A1 (es) | 2006-07-26 |
CN101006072A (zh) | 2007-07-25 |
CA2570606C (en) | 2013-04-30 |
NZ552056A (en) | 2010-08-27 |
TW200611702A (en) | 2006-04-16 |
ES2573844T3 (es) | 2016-06-10 |
EA200700035A1 (ru) | 2007-06-29 |
JP2008503487A (ja) | 2008-02-07 |
BRPI0512242A (pt) | 2008-02-19 |
CN101006072B (zh) | 2011-10-19 |
IL180108A0 (en) | 2007-05-15 |
AU2005262496A1 (en) | 2006-01-19 |
EP1768970B1 (en) | 2016-03-09 |
EP1768970A1 (en) | 2007-04-04 |
AU2005262496B2 (en) | 2011-10-20 |
UA91680C2 (ru) | 2010-08-25 |
EA013685B1 (ru) | 2010-06-30 |
CR8858A (es) | 2009-01-14 |
CA2570606A1 (en) | 2006-01-19 |
JP5416740B2 (ja) | 2014-02-12 |
MY147767A (en) | 2013-01-31 |
AR091400A2 (es) | 2015-02-04 |
JP2011246472A (ja) | 2011-12-08 |
US20060041008A1 (en) | 2006-02-23 |
ECSP067093A (es) | 2007-01-26 |
IL180108A (en) | 2015-10-29 |
US8084490B2 (en) | 2011-12-27 |
NO20070081L (no) | 2007-02-26 |
MXPA06014934A (es) | 2007-08-21 |
JP4884378B2 (ja) | 2012-02-29 |
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