MY137045A - Medicaments comprising steroids and a novel anticholinergic - Google Patents

Medicaments comprising steroids and a novel anticholinergic

Info

Publication number
MY137045A
MY137045A MYPI20031320A MYPI20031320A MY137045A MY 137045 A MY137045 A MY 137045A MY PI20031320 A MYPI20031320 A MY PI20031320A MY PI20031320 A MYPI20031320 A MY PI20031320A MY 137045 A MY137045 A MY 137045A
Authority
MY
Malaysia
Prior art keywords
steroids
medicaments
pharmaceutical compositions
novel pharmaceutical
present
Prior art date
Application number
MYPI20031320A
Inventor
Rolf Dr Banholzer
Helmut Meissner
Gerd Morschhaeuser
Michael P Dr Pieper
Gerald Dr Pohl
Richard Dr Reichl
Georg Dr Speck
Christopher John Montague Dr Meade
Michel Dr Pairet
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of MY137045A publication Critical patent/MY137045A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/468-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4738Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/12Aerosols; Foams
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/16Central respiratory analeptics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/06Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Emergency Medicine (AREA)
  • Dispersion Chemistry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

THE PRESENT INVENTION RELATES TO NOVEL PHARMACEUTICAL COMPOSITIONS COMPRISING STEROIDS WITH A LONG-LASTING EFFECT AND COMPRISING SALTS OF A NEW ANTICHOLINERGIC OF FORMULA 1.WHEREINX -DENOTES AN ANION WITH A SINGLE NEGATIVE CHARGE, PREFERABLY AN ANION SELECTED FROM THE GROUP CONSISTING OF CHLORIDE, BROMIDE, IODIDE, SULPHATE, PHOSPHATE, METHANESULPHONATE, NITRATE, MALEATE, ACETATE, CITRATE, FUMARATE, TARTRATE, OXALATE, SUCCINATE, BENZOATE AND P-TOLUENESULPHONATE. THE PRESENT INVENTION FURTHER RELATES TO PROCESSES FOR PREPARING THESE NOVEL PHARMACEUTICAL COMPOSITIONS AND THEIR USE IN THE TREATMENT OF RESPIRATORY COMPLAINTS, IN PARTICULAR ASTHMA AND COPD.
MYPI20031320A 2002-04-12 2003-04-10 Medicaments comprising steroids and a novel anticholinergic MY137045A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10216429A DE10216429A1 (en) 2002-04-12 2002-04-12 Synergistic medicaments for treating inflammatory or obstructive respiratory tract diseases, containing quaternized scopine ester anticholinergic agent and steroid, e.g. budesonide

Publications (1)

Publication Number Publication Date
MY137045A true MY137045A (en) 2008-12-31

Family

ID=28458802

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI20031320A MY137045A (en) 2002-04-12 2003-04-10 Medicaments comprising steroids and a novel anticholinergic

Country Status (29)

Country Link
EP (2) EP1496902B1 (en)
JP (1) JP4559086B2 (en)
KR (1) KR101010869B1 (en)
CN (1) CN1646126A (en)
AR (1) AR039275A1 (en)
AT (1) ATE312607T1 (en)
AU (1) AU2003216921B2 (en)
BR (1) BR0309085A (en)
CA (1) CA2481268C (en)
DE (2) DE10216429A1 (en)
DK (1) DK1496902T3 (en)
EA (1) EA008386B1 (en)
EC (1) ECSP045355A (en)
ES (1) ES2254917T3 (en)
HR (1) HRP20040943B1 (en)
IL (2) IL164391A0 (en)
ME (1) MEP54208A (en)
MX (1) MXPA04009917A (en)
MY (1) MY137045A (en)
NO (1) NO20044097L (en)
NZ (1) NZ536284A (en)
PE (1) PE20040326A1 (en)
PL (1) PL211227B1 (en)
RS (1) RS50776B (en)
TW (1) TWI311055B (en)
UA (1) UA80125C2 (en)
UY (1) UY27758A1 (en)
WO (1) WO2003086399A1 (en)
ZA (1) ZA200406751B (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2165768B1 (en) 1999-07-14 2003-04-01 Almirall Prodesfarma Sa NEW DERIVATIVES OF QUINUCLIDINE AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM.
GB2389530B (en) 2002-06-14 2007-01-10 Cipla Ltd Pharmaceutical compositions
CN100569235C (en) 2004-02-06 2009-12-16 Meda制药有限及两合公司 Be used for the anticholinergic of asthma and COPD long-term treatment and the combination of glucocorticoid
EP2100598A1 (en) 2008-03-13 2009-09-16 Laboratorios Almirall, S.A. Inhalation composition containing aclidinium for treatment of asthma and chronic obstructive pulmonary disease
EP2100599A1 (en) 2008-03-13 2009-09-16 Laboratorios Almirall, S.A. Inhalation composition containing aclidinium for treatment of asthma and chronic obstructive pulmonary disease
US8815258B2 (en) 2009-05-29 2014-08-26 Pearl Therapeutics, Inc. Compositions, methods and systems for respiratory delivery of two or more active agents
ES2774391T3 (en) 2009-05-29 2020-07-20 Pearl Therapeutics Inc Compositions, methods and systems for the respiratory administration of two or more active agents
EP2510928A1 (en) 2011-04-15 2012-10-17 Almirall, S.A. Aclidinium for use in improving the quality of sleep in respiratory patients
BR112015022784B1 (en) 2013-03-15 2023-02-14 Pearl Therapeutics, Inc MICRONIZED CRYSTALLINE MATERIAL CONDITIONING METHOD AND CONDITIONING SYSTEMS
CN115282411A (en) * 2022-01-14 2022-11-04 温州医科大学 Delivery system for delivering drugs into the brain using the nasal olfactory region and method of use thereof

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4570630A (en) 1983-08-03 1986-02-18 Miles Laboratories, Inc. Medicament inhalation device
DK163640C (en) 1985-07-30 1992-08-17 Glaxo Group Ltd DEVICE FOR ADMINISTRATING MEDICINES
SG45171A1 (en) 1990-03-21 1998-01-16 Boehringer Ingelheim Int Atomising devices and methods
DE4108393A1 (en) 1991-03-15 1992-09-17 Boehringer Ingelheim Kg NEW ESTERS BI-AND TRICYCLIC AMINO ALCOHOLS, THEIR PREPARATION AND THEIR USE IN MEDICINAL PRODUCTS
IL107120A (en) 1992-09-29 1997-09-30 Boehringer Ingelheim Int Atomising nozzle and filter and spray generating device
DE4318455A1 (en) 1993-06-03 1994-12-08 Boehringer Ingelheim Kg Capsule holder
DE69632728T2 (en) * 1995-04-28 2004-10-14 Banyu Pharmaceutical Co., Ltd. 1,4-DISUBSTITUTED PIPERID DERIVATIVES
DE19536902A1 (en) 1995-10-04 1997-04-10 Boehringer Ingelheim Int Miniature fluid pressure generating device
DE19536903C2 (en) 1995-10-04 1998-09-10 Boehringer Ingelheim Int Device for holding a fluidic component
DE19545226C1 (en) 1995-12-05 1997-06-19 Boehringer Ingelheim Int Locking mechanism for a spring-operated output
GB0009591D0 (en) * 2000-04-18 2000-06-07 Glaxo Group Ltd Medical combinations
DE10050994A1 (en) * 2000-10-14 2002-04-18 Boehringer Ingelheim Pharma New diphenylalkanoic acid azabicyclooctane ester quaternary salts useful as anticholinergic agents, especially in treatment of asthma and chronic obstructive pulmonary disease
MXPA03003751A (en) * 2000-10-31 2004-10-15 Boehringer Ingelheim Pharma Novel medicament compositions based on anticholinergics and corticosteroids.

Also Published As

Publication number Publication date
EA008386B1 (en) 2007-04-27
TW200403062A (en) 2004-03-01
NO20044097L (en) 2004-11-04
ES2254917T3 (en) 2006-06-16
HRP20040943A2 (en) 2005-04-30
BR0309085A (en) 2005-02-09
KR101010869B1 (en) 2011-01-26
AR039275A1 (en) 2005-02-16
RS50776B (en) 2010-08-31
CA2481268A1 (en) 2003-10-23
EP1621197A3 (en) 2010-01-06
PE20040326A1 (en) 2004-07-13
CA2481268C (en) 2011-07-12
AU2003216921A1 (en) 2003-10-27
IL164391A0 (en) 2005-12-18
RS89904A (en) 2006-10-27
KR20050000391A (en) 2005-01-03
IL164391A (en) 2010-11-30
UA80125C2 (en) 2007-08-27
EP1621197A2 (en) 2006-02-01
ATE312607T1 (en) 2005-12-15
HRP20040943B1 (en) 2013-05-31
UY27758A1 (en) 2003-11-28
TWI311055B (en) 2009-06-21
JP2005529105A (en) 2005-09-29
JP4559086B2 (en) 2010-10-06
AU2003216921B2 (en) 2008-03-13
ZA200406751B (en) 2006-12-27
PL211227B1 (en) 2012-04-30
DE10216429A1 (en) 2003-10-23
NZ536284A (en) 2006-11-30
ECSP045355A (en) 2005-01-28
CN1646126A (en) 2005-07-27
MXPA04009917A (en) 2004-12-07
DE50301934D1 (en) 2006-01-19
EP1496902B1 (en) 2005-12-14
MEP54208A (en) 2011-05-10
WO2003086399A1 (en) 2003-10-23
EP1496902A1 (en) 2005-01-19
PL371561A1 (en) 2005-06-27
EA200401303A1 (en) 2005-04-28
DK1496902T3 (en) 2006-05-08

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