MA52754A - Composés hétérocycliques tricycliques en tant qu'activateurs de sting - Google Patents

Composés hétérocycliques tricycliques en tant qu'activateurs de sting

Info

Publication number
MA52754A
MA52754A MA052754A MA52754A MA52754A MA 52754 A MA52754 A MA 52754A MA 052754 A MA052754 A MA 052754A MA 52754 A MA52754 A MA 52754A MA 52754 A MA52754 A MA 52754A
Authority
MA
Morocco
Prior art keywords
tricyclic compounds
sting activators
heterocyclic tricyclic
heterocyclic
sting
Prior art date
Application number
MA052754A
Other languages
English (en)
French (fr)
Inventor
Neil Lajkiewicz
Zhenwu Li
Liangxing Wu
Wenqing Yao
Yingda Ye
Original Assignee
Incyte Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Incyte Corp filed Critical Incyte Corp
Publication of MA52754A publication Critical patent/MA52754A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
MA052754A 2018-05-25 2019-05-24 Composés hétérocycliques tricycliques en tant qu'activateurs de sting MA52754A (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862676810P 2018-05-25 2018-05-25
US201862730610P 2018-09-13 2018-09-13
US201962841587P 2019-05-01 2019-05-01

Publications (1)

Publication Number Publication Date
MA52754A true MA52754A (fr) 2021-04-14

Family

ID=66912949

Family Applications (1)

Application Number Title Priority Date Filing Date
MA052754A MA52754A (fr) 2018-05-25 2019-05-24 Composés hétérocycliques tricycliques en tant qu'activateurs de sting

Country Status (7)

Country Link
US (2) US10947227B2 (https=)
EP (1) EP3802534B1 (https=)
JP (2) JP7570235B2 (https=)
CA (1) CA3101368A1 (https=)
ES (1) ES2929415T3 (https=)
MA (1) MA52754A (https=)
WO (1) WO2019227007A1 (https=)

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Also Published As

Publication number Publication date
WO2019227007A1 (en) 2019-11-28
JP2021525706A (ja) 2021-09-27
JP2024133472A (ja) 2024-10-02
CA3101368A1 (en) 2019-11-28
US11713317B2 (en) 2023-08-01
JP7570235B2 (ja) 2024-10-21
US20190359608A1 (en) 2019-11-28
US20220073509A1 (en) 2022-03-10
US10947227B2 (en) 2021-03-16
EP3802534B1 (en) 2022-07-13
EP3802534A1 (en) 2021-04-14
ES2929415T3 (es) 2022-11-29

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