KR940003071B1 - 벤즈옥사진 유도체 및 이의 제조방법 - Google Patents

벤즈옥사진 유도체 및 이의 제조방법 Download PDF

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Publication number
KR940003071B1
KR940003071B1 KR1019880002851A KR880002851A KR940003071B1 KR 940003071 B1 KR940003071 B1 KR 940003071B1 KR 1019880002851 A KR1019880002851 A KR 1019880002851A KR 880002851 A KR880002851 A KR 880002851A KR 940003071 B1 KR940003071 B1 KR 940003071B1
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KR
South Korea
Prior art keywords
group
formula
compound
hydrogen atom
pharmaceutically acceptable
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
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KR1019880002851A
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English (en)
Korean (ko)
Other versions
KR880011154A (ko
Inventor
이쿠오 이이지마
마사카쓰 오오제키
쿠니히토 오쿠무라
마사노리 이나마스
Original Assignee
타나베세이야꾸가부시끼가이샤
아다찌 케이지로
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Publication of KR880011154A publication Critical patent/KR880011154A/ko
Application granted granted Critical
Publication of KR940003071B1 publication Critical patent/KR940003071B1/ko
Anticipated expiration legal-status Critical
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
KR1019880002851A 1987-03-18 1988-03-18 벤즈옥사진 유도체 및 이의 제조방법 Expired - Fee Related KR940003071B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP65360/87 1987-03-18
JP62065360A JPS63230689A (ja) 1987-03-18 1987-03-18 ベンゾオキサジン誘導体
JP62-65360 1987-03-18

Publications (2)

Publication Number Publication Date
KR880011154A KR880011154A (ko) 1988-10-26
KR940003071B1 true KR940003071B1 (ko) 1994-04-13

Family

ID=13284716

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019880002851A Expired - Fee Related KR940003071B1 (ko) 1987-03-18 1988-03-18 벤즈옥사진 유도체 및 이의 제조방법

Country Status (16)

Country Link
US (1) US4824833A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (1) EP0283036B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JPS63230689A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (1) KR940003071B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CN (1) CN1019911C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AT (1) ATE67199T1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA1305706C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE3864707D1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (1) DK147588A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (1) ES2038710T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (1) FI91870C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR2612517B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GR (1) GR3002692T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HU (2) HU203548B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IE (1) IE60522B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL85768A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995018805A1 (en) * 1992-09-21 1995-07-13 Senju Pharmaceutical Co., Ltd. 1,4-benzoxazine-2-acetic acid compound, process for producing the same, and use thereof
US5332733A (en) * 1990-11-24 1994-07-26 Kali-Chemie Pharma Gmbh Heterocyclically substituted piperazinoakylbenzoxazine and piperazinoalkylbenzothiazine compounds, processes for preparing them, and medicaments containing them
US5635505A (en) * 1994-01-06 1997-06-03 Senju Pharmaceutical Co., Ltd. 1,4-benzoxazine-2-acetic acid compound, method for production thereof and use thereof
CA2384194A1 (en) 1999-08-31 2001-03-08 David P. M. Pleynet Benzylidene-thiazolidinediones and analogues and their use in the treatment of inflammation
CA2473156A1 (en) * 2001-03-08 2002-09-19 Incyte San Diego, Inc. Rxr activating molecules
US7102000B2 (en) * 2002-03-08 2006-09-05 Incyte San Diego Inc. Heterocyclic amide derivatives for the treatment of diabetes and other diseases
EP1549644A1 (en) 2002-07-10 2005-07-06 Applied Research Systems ARS Holding N.V. Azolidinone-vinyl fused-benzene derivatives
BR0316386A (pt) * 2002-12-06 2005-09-27 Warner Lambert Co Benzoxazin-3-onas e seus derivados como inibidores de p13k
ES2393197T3 (es) * 2004-09-28 2012-12-19 Otsuka Pharmaceutical Co., Ltd. Compuesto de carbostirilo
CN100455573C (zh) * 2005-11-11 2009-01-28 华东理工大学 一种制备1,4-苯并噁唑嗪-3-酮化合物的微波合成方法
CA2898482A1 (en) * 2013-02-22 2014-08-28 Linda L. Brockunier Antidiabetic bicyclic compounds
US10968193B2 (en) 2014-08-08 2021-04-06 Merck Sharp & Dohme Corp. Antidiabetic bicyclic compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5522636A (en) * 1978-08-04 1980-02-18 Takeda Chem Ind Ltd Thiazoliding derivative
US4619687A (en) * 1984-09-27 1986-10-28 Sumitomo Chemical Company, Limited Triazolopyridazines and their use as herbicides
CN1003445B (zh) * 1984-10-03 1989-03-01 武田药品工业株式会社 噻唑烷二酮衍生物，其制备方法和用途
WO1986007056A1 (en) * 1985-05-21 1986-12-04 Pfizer Inc. Hypoglycemic thiazolidinediones
JPH06779B2 (ja) * 1985-06-10 1994-01-05 武田薬品工業株式会社 チアゾリジオン誘導体およびそれを含んでなる医薬組成物
JPS6314782A (ja) * 1986-07-07 1988-01-21 Nippon Tokushu Noyaku Seizo Kk 新規ジアルキルマレインイミド類及び除草剤
US4734124A (en) * 1987-01-15 1988-03-29 Fmc Corporation Tetrazolinone herbicides
FI91869C (fi) * 1987-03-18 1994-08-25 Tanabe Seiyaku Co Menetelmä antidiabeettisena aineena käytettävien bensoksatsolijohdannaisten valmistamiseksi

Also Published As

Publication number Publication date
EP0283036A1 (en) 1988-09-21
FI91870C (fi) 1994-08-25
DK147588A (da) 1988-09-19
ATE67199T1 (de) 1991-09-15
CN1019911C (zh) 1993-02-17
HUT50337A (en) 1990-01-29
IL85768A0 (en) 1988-09-30
IL85768A (en) 1993-02-21
HU211596A9 (en) 1995-12-28
DK147588D0 (da) 1988-03-17
ES2038710T3 (es) 1993-08-01
CN88101541A (zh) 1988-10-05
FI881104L (fi) 1988-09-19
JPH0460597B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1992-09-28
HU203548B (en) 1991-08-28
CA1305706C (en) 1992-07-28
KR880011154A (ko) 1988-10-26
DE3864707D1 (de) 1991-10-17
GR3002692T3 (en) 1993-01-25
IE60522B1 (en) 1994-07-27
FI91870B (fi) 1994-05-13
FR2612517B1 (fr) 1992-11-13
IE880772L (en) 1988-09-18
AU1317688A (en) 1988-09-22
FR2612517A1 (fr) 1988-09-23
EP0283036B1 (en) 1991-09-11
US4824833A (en) 1989-04-25
FI881104A0 (fi) 1988-03-09
JPS63230689A (ja) 1988-09-27
AU601029B2 (en) 1990-08-30

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