KR900005021B1 - 1-펜옥시-3-히드록시 인돌릴 알킬아미노-3-프로판올류 및 그 제조방법 - Google Patents

1-펜옥시-3-히드록시 인돌릴 알킬아미노-3-프로판올류 및 그 제조방법 Download PDF

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Publication number
KR900005021B1
KR900005021B1 KR1019840003251A KR840003251A KR900005021B1 KR 900005021 B1 KR900005021 B1 KR 900005021B1 KR 1019840003251 A KR1019840003251 A KR 1019840003251A KR 840003251 A KR840003251 A KR 840003251A KR 900005021 B1 KR900005021 B1 KR 900005021B1
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KR
South Korea
Prior art keywords
compound
formula
hydrogen
hydroxy
alkyl
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Expired
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KR1019840003251A
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English (en)
Korean (ko)
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KR850000396A (ko
Inventor
이이. 크라이그바움 윌리암
Original Assignee
브리스톨-마이어즈 스퀴브 컴페니
아이삭 자아코브스키
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Publication of KR850000396A publication Critical patent/KR850000396A/ko
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Publication of KR900005021B1 publication Critical patent/KR900005021B1/ko
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D303/00Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02Compounds containing oxirane rings
    • C07D303/12Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
    • C07D303/18Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by etherified hydroxyl radicals
    • C07D303/20Ethers with hydroxy compounds containing no oxirane rings
    • C07D303/22Ethers with hydroxy compounds containing no oxirane rings with monohydroxy compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1019840003251A 1983-06-10 1984-06-09 1-펜옥시-3-히드록시 인돌릴 알킬아미노-3-프로판올류 및 그 제조방법 Expired KR900005021B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US50290183A 1983-06-10 1983-06-10
US502901 1983-06-10

Publications (2)

Publication Number Publication Date
KR850000396A KR850000396A (ko) 1985-02-27
KR900005021B1 true KR900005021B1 (ko) 1990-07-18

Family

ID=23999880

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019840003251A Expired KR900005021B1 (ko) 1983-06-10 1984-06-09 1-펜옥시-3-히드록시 인돌릴 알킬아미노-3-프로판올류 및 그 제조방법

Country Status (29)

Country Link
JP (1) JPS608262A (enrdf_load_html_response)
KR (1) KR900005021B1 (enrdf_load_html_response)
AT (1) AT381492B (enrdf_load_html_response)
AU (1) AU569303B2 (enrdf_load_html_response)
BE (1) BE899875A (enrdf_load_html_response)
CA (1) CA1217496A (enrdf_load_html_response)
CH (1) CH662561A5 (enrdf_load_html_response)
CY (1) CY1518A (enrdf_load_html_response)
DE (1) DE3421252A1 (enrdf_load_html_response)
DK (1) DK162089C (enrdf_load_html_response)
ES (1) ES533185A0 (enrdf_load_html_response)
FI (1) FI78291C (enrdf_load_html_response)
FR (1) FR2549054B1 (enrdf_load_html_response)
GB (1) GB2141121B (enrdf_load_html_response)
GR (1) GR82208B (enrdf_load_html_response)
HK (1) HK14690A (enrdf_load_html_response)
HU (1) HU191670B (enrdf_load_html_response)
IE (1) IE57682B1 (enrdf_load_html_response)
IL (1) IL72008A (enrdf_load_html_response)
IT (1) IT1206705B (enrdf_load_html_response)
LU (1) LU85410A1 (enrdf_load_html_response)
MY (1) MY102077A (enrdf_load_html_response)
NL (1) NL8401840A (enrdf_load_html_response)
NO (1) NO164471C (enrdf_load_html_response)
NZ (1) NZ208337A (enrdf_load_html_response)
SE (1) SE455865B (enrdf_load_html_response)
SG (1) SG1090G (enrdf_load_html_response)
YU (1) YU44873B (enrdf_load_html_response)
ZA (1) ZA844277B (enrdf_load_html_response)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2601008B1 (fr) * 1986-07-03 1990-03-30 Sanofi Sa Procede de synthese stereospecifique de derives de l'indole
KR101986648B1 (ko) 2018-04-06 2019-06-07 (유)로뎀건설 강관작업구 굴착장치

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES259580A1 (es) * 1959-07-13 1961-01-16 Philips Nv Procedimiento para la preparacion de nuevas indolietilaminas farmacologicamente activas
NL300886A (enrdf_load_html_response) * 1962-11-23
CA1116598A (en) * 1977-07-13 1982-01-19 William T. Comer 3-indolyl-tertiary butylaminopropanols
US4314943A (en) * 1977-07-13 1982-02-09 Mead Johnson & Company Heterocyclic substituted aryloxy 3-indolyl-tertiary butylaminopropanols
US4234595A (en) * 1977-07-13 1980-11-18 Mead Johnson & Company 3-Indolyl-tertiary butylaminopropanols
FR2463765A1 (fr) * 1979-08-17 1981-02-27 Clin Midy Nouveaux derives de l'indole actifs sur le systeme cardiovasculaire

Also Published As

Publication number Publication date
NO164471B (no) 1990-07-02
JPS608262A (ja) 1985-01-17
CY1518A (en) 1990-11-16
IT8421330A0 (it) 1984-06-08
HUT34445A (en) 1985-03-28
GB2141121B (en) 1987-01-07
FI842316L (fi) 1984-12-11
DK284184D0 (da) 1984-06-08
NL8401840A (nl) 1985-01-02
GB8414652D0 (en) 1984-07-11
FI78291B (fi) 1989-03-31
FR2549054B1 (fr) 1988-03-04
NZ208337A (en) 1988-10-28
ES8507490A1 (es) 1985-09-16
DK284184A (da) 1984-12-11
FI842316A0 (fi) 1984-06-07
KR850000396A (ko) 1985-02-27
ZA844277B (en) 1985-03-27
IT1206705B (it) 1989-04-27
AU569303B2 (en) 1988-01-28
MY102077A (en) 1992-03-31
CA1217496A (en) 1987-02-03
GR82208B (enrdf_load_html_response) 1984-12-13
FR2549054A1 (fr) 1985-01-18
FI78291C (fi) 1989-07-10
NO164471C (no) 1990-10-10
DK162089B (da) 1991-09-16
AT381492B (de) 1986-10-27
CH662561A5 (de) 1987-10-15
SE8403112L (sv) 1984-12-11
YU99784A (en) 1986-10-31
IL72008A0 (en) 1984-10-31
ATA186784A (de) 1986-03-15
SE455865B (sv) 1988-08-15
JPH0587503B2 (enrdf_load_html_response) 1993-12-16
LU85410A1 (fr) 1985-03-26
IL72008A (en) 1988-05-31
AU2923884A (en) 1984-12-13
DE3421252A1 (de) 1984-12-13
NO842279L (no) 1984-12-11
SG1090G (en) 1990-07-06
IE57682B1 (en) 1993-02-24
GB2141121A (en) 1984-12-12
IE841441L (en) 1984-12-10
BE899875A (fr) 1984-12-10
DK162089C (da) 1992-02-24
YU44873B (en) 1991-04-30
HK14690A (en) 1990-03-02
HU191670B (en) 1987-03-30
SE8403112D0 (sv) 1984-06-08
ES533185A0 (es) 1985-09-16

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