KR890003380A - 피부에 축적하는 외용의 항 바이러스성 약학적 조성물 및 그 제조방법 - Google Patents
피부에 축적하는 외용의 항 바이러스성 약학적 조성물 및 그 제조방법 Download PDFInfo
- Publication number
- KR890003380A KR890003380A KR1019880008222A KR880008222A KR890003380A KR 890003380 A KR890003380 A KR 890003380A KR 1019880008222 A KR1019880008222 A KR 1019880008222A KR 880008222 A KR880008222 A KR 880008222A KR 890003380 A KR890003380 A KR 890003380A
- Authority
- KR
- South Korea
- Prior art keywords
- pharmaceutical composition
- external
- skin
- manufacturing
- antiviral pharmaceutical
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/06—Pyrimidine radicals
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biotechnology (AREA)
- Ophthalmology & Optometry (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Dermatology (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
내용 없음
Description
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음
제1도는 사이민, EDU 및 IPDU의 사이민 포릴라제에 의한 분해율을 나타낸 것이며, 제2도는 IPDU(I)로 처리한 마우스의 뇨증에서 확인된 대사생성물을 나타낸 것이다.
Claims (3)
- 5-이소프로필-2'-β-데옥시유리딘 0.02-5%(W)을 외용의 약학적 조성물의 제조에 통상으로 사용되는 담체, 희석제 및/또는 기타 첨가제와 혼합하여 이루어진 피부에 축적하는 외용의 항 바이러스성 약학적 조성물.
- 5-이소프로필-2'-β-데옥시유리딘 0.1-1%(W)를 외용의 약학적 조성물의 제조에 통상으로 사용되는 담체, 희석제 및/또는 기타 첨가제와 혼합하여 이루어진 안과용 항 바이러스성 약학적 조성물.
- 5-이소프로필-2'-β-데옥시유리딘 0.2-5%(W)를 외용의 약학적 조성물의 제조에 사용되는 담체, 희석제 및/또는 기타 첨가제와 함께 혼합하고 통상의 방법으로 연고, 유제, 현탁제, 겔, 액제, 분무제, 점착제, 등과 같은 약학적 조성물로 성형함을 특징으로 하는 피부에 축적하는 외용의 항 바이러스성 약학적 조성물을 제조하는 방법.※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HU873596A HU196038B (en) | 1987-08-07 | 1987-08-07 | Process for producing antiherpetic pharmaceutics for external use, containing 5-isopropyl-2'-beta-deoxy-uridine |
HU3596/87 | 1987-08-07 |
Publications (2)
Publication Number | Publication Date |
---|---|
KR890003380A true KR890003380A (ko) | 1989-04-14 |
KR960015953B1 KR960015953B1 (ko) | 1996-11-25 |
Family
ID=10964716
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR1019880008222A KR960015953B1 (ko) | 1987-08-07 | 1988-07-02 | 피부에 축적하는 외용의 항바이러스성 약학적 조성물 및 그 제조방법 |
Country Status (25)
Country | Link |
---|---|
US (2) | US4880785A (ko) |
JP (1) | JPS6442437A (ko) |
KR (1) | KR960015953B1 (ko) |
CN (1) | CN1034133A (ko) |
AU (1) | AU605875B2 (ko) |
BE (1) | BE1001774A4 (ko) |
CA (1) | CA1286227C (ko) |
CH (1) | CH675538A5 (ko) |
CS (1) | CS276467B6 (ko) |
CY (1) | CY1655A (ko) |
DD (1) | DD270656A5 (ko) |
DE (1) | DE3820270A1 (ko) |
DK (1) | DK299088A (ko) |
ES (1) | ES2010559A6 (ko) |
FI (1) | FI883692A (ko) |
FR (1) | FR2619010B1 (ko) |
GB (1) | GB2207864B (ko) |
GR (1) | GR1000139B (ko) |
HU (1) | HU196038B (ko) |
IT (1) | IT1217789B (ko) |
NL (1) | NL8801411A (ko) |
NO (1) | NO882491L (ko) |
RU (1) | RU2035180C1 (ko) |
SE (1) | SE503261C2 (ko) |
SG (1) | SG42292G (ko) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8904855D0 (en) * | 1989-03-03 | 1989-04-12 | Beecham Group Plc | Pharmaceutical treatment |
ZA927277B (en) * | 1991-10-02 | 1993-05-19 | Boston Ocular Res | Dry eye treatment process and solution. |
HUP9602024A3 (en) * | 1996-07-25 | 1999-05-28 | Toth Sandor | Pharmaceutical composition containing aminoacid for external use |
MY136633A (en) * | 2001-01-17 | 2008-11-28 | Berlin Chemie Ag | Stabilized brivudine topical formulations |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2918260A1 (de) * | 1979-05-07 | 1980-11-27 | Robugen Gmbh | Anwendung von 5-alkyl-2'-desoxyuridinen |
DE3010397A1 (de) * | 1980-03-18 | 1981-10-29 | Robugen Gmbh Pharmazeutische Fabrik Esslingen A.N., 7300 Esslingen | Verwendung von 5-alkyl-pyrimidinnukleosiden als cytostatika |
WO1983000436A1 (en) * | 1981-08-04 | 1983-02-17 | Gauri, Kailash, Kumar | Combined preparation with synergic effect |
HU198393B (en) * | 1984-03-06 | 1989-10-30 | Sloan Kettering Inst Cancer | Process for production of medical composition suitable for treatment of hepatitis containing as active substance derivatives of piramidin-nucleoside |
HU197837B (en) * | 1984-12-29 | 1989-06-28 | Mta Koezponti Kemiai Kutato In | Composition with skin cleaning effect, particularly for treating pimpled skin of face |
-
1987
- 1987-08-07 HU HU873596A patent/HU196038B/hu not_active IP Right Cessation
-
1988
- 1988-06-02 DK DK299088A patent/DK299088A/da not_active Application Discontinuation
- 1988-06-02 NL NL8801411A patent/NL8801411A/nl active Search and Examination
- 1988-06-02 FR FR888807341A patent/FR2619010B1/fr not_active Expired - Lifetime
- 1988-06-06 IT IT20871/88A patent/IT1217789B/it active
- 1988-06-06 NO NO88882491A patent/NO882491L/no unknown
- 1988-06-06 AU AU17413/88A patent/AU605875B2/en not_active Ceased
- 1988-06-07 GB GB8813392A patent/GB2207864B/en not_active Expired - Lifetime
- 1988-06-08 BE BE8800651A patent/BE1001774A4/fr not_active IP Right Cessation
- 1988-06-09 CA CA000569083A patent/CA1286227C/en not_active Expired - Lifetime
- 1988-06-10 US US07/204,724 patent/US4880785A/en not_active Expired - Lifetime
- 1988-06-10 DD DD88316660A patent/DD270656A5/de not_active IP Right Cessation
- 1988-06-13 SE SE8802193A patent/SE503261C2/sv not_active IP Right Cessation
- 1988-06-14 DE DE3820270A patent/DE3820270A1/de not_active Ceased
- 1988-06-18 JP JP63149285A patent/JPS6442437A/ja active Granted
- 1988-06-22 CH CH2399/88A patent/CH675538A5/de not_active IP Right Cessation
- 1988-06-23 CS CS884413A patent/CS276467B6/cs not_active IP Right Cessation
- 1988-06-24 GR GR880100417A patent/GR1000139B/el not_active IP Right Cessation
- 1988-06-29 ES ES8802036A patent/ES2010559A6/es not_active Expired
- 1988-07-02 KR KR1019880008222A patent/KR960015953B1/ko not_active IP Right Cessation
- 1988-08-05 RU SU884356280A patent/RU2035180C1/ru active
- 1988-08-06 CN CN88104902A patent/CN1034133A/zh active Pending
- 1988-08-08 FI FI883692A patent/FI883692A/fi not_active Application Discontinuation
-
1989
- 1989-05-16 US US07/352,420 patent/US4937233A/en not_active Expired - Lifetime
-
1992
- 1992-04-16 SG SG422/92A patent/SG42292G/en unknown
-
1993
- 1993-05-14 CY CY1655A patent/CY1655A/xx unknown
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