KR850005422A - 트리아졸 유도체의 제조방법 - Google Patents
트리아졸 유도체의 제조방법 Download PDFInfo
- Publication number
- KR850005422A KR850005422A KR1019850000417A KR850000417A KR850005422A KR 850005422 A KR850005422 A KR 850005422A KR 1019850000417 A KR1019850000417 A KR 1019850000417A KR 850000417 A KR850000417 A KR 850000417A KR 850005422 A KR850005422 A KR 850005422A
- Authority
- KR
- South Korea
- Prior art keywords
- fluorophenyl
- formula
- difluorophenyl
- independently
- compound
- Prior art date
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
- A01N43/647—Triazoles; Hydrogenated triazoles
- A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
- C07C45/46—Friedel-Crafts reactions
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
- C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
내용 없음
Description
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음
Claims (8)
- 다음 일반식(Ⅱ)화합물을 다음 일반식(Ⅲ)의 케톤과 반응시킨 다음, 생성물을 0-에스테르 또는 0-에테르로 전환시키는 공정 및 약학적으로 또는 농업적으로 허용되는 염으로 전환시키는 공정중의 하나 또는 두 공정을 임의로 수행함을 특징으로하여 다음 일반식(Ⅰ)의 트리아졸 또는 이의 0-에스테르, 0-에테르 또는 약학적으로 또는 농업적으로 허용되는 염을 제조하는 방법.상기식에서, R 및 R¹은 상기 독립적으로 F, Cl, Br, I, CF₃,C₁-C₄알킬 및 C₁-C₄알콕시 중에서 각기 독립적으로 선택된 1내지 3개의 치환체로 임의 치환된 페닐 그룹이고, R²는 H,CH₃또는 F이고, R₃는 H또는 CH₃이며, 단, R²및 R³중 하나는 H가 아니다.
- 제1항에 있어서, R 및 R¹이 각기 독립적으로, F,Cl,Br,I및 CF₃중에서 각기 독립적으로 선택된 1내지 3개의 치환체로 치환된 페닐임을 특징으로 하는 방법.
- 제2항에 있어서, R 및 R¹이 각기 독립적으로 4-플루오로페닐, 4-클로로페닐, 4-트리플루오로틸페닐, 2-플루오로페닐, 2,4-디클로로페닐, 2,4-디플루오로페닐, 4-클로로-2-플루오로페닐, 2-클로로-4-플루오로페닐, 2,5-디플루오로페닐, 2,4,6-트리플루오로페닐 또는 4-브로모-2,5-디플루오로페닐임을 특징으로 하는 방법.
- 제3항에 있어서, R및 R¹이 각기 독립적으로 4-클로로페닐, 4-플루오로페닐, 2,4-디콜로로페닐 또는 2,4-디플루오로페닐임을 특징으로하는 방법.
- 제1항에 있어서, R²가 F이고 R³가 CH₃임을 특징으로하는 방법.
- 제1항에 있어서, R²가 H,CH₃또는 F이고 R³가 CH₃임을 특징으로 하는 방법.
- 다음 일반식(Ⅳ)의 화합물을 2당량이상의 다음 일반식(Ⅲ)화합물과 반응시킨 다음 임의로 생성물을 0-에스테르 또는 0-에테르로 전환시키고/시키거나, 약학적으로 또는 농업적으로 허용되는 염으로 전환시킴을 특징으로하여 R 및 R¹이 동일하고 R²및 R³가 모두 CH₃인 일반식(Ⅰ)의 트리아졸을 제조하는 방법.상기식에서, R 및 R¹이 동일하며, F,Cl,Br,I,CF3, C1-C4알킬 및 C₁-C₄알콕시중에서 각기 독립적으로 선택된 1내지 3개의 치환체로 임의 치환된 페닐그룹이다.
- 제7항에 있어서, R 및 R¹이 동일하게 4-페플루오로닐, 4-클로로페닐, 4-트리플루오로메틸페닐, 2-플루오로페닐, 2,4-디클로로페닐, 2,4-디플루오로페닐, 4-클로로-2-플루오로페닐, 2-클로로-4-플루오로페닐, 2,5-디플루오로페닐, 2,4,6-트리플루오로페닐 또는 4-부로모-2,5-디플루오로페닐인 방법.※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB????8401738? | 1984-01-24 | ||
GB848401738A GB8401738D0 (en) | 1984-01-24 | 1984-01-24 | Triazole antifungal agents |
GB848420583A GB8420583D0 (en) | 1984-08-14 | 1984-08-14 | Triazole antifungal agents |
GB8420583? | 1984-08-14 |
Publications (1)
Publication Number | Publication Date |
---|---|
KR850005422A true KR850005422A (ko) | 1985-08-26 |
Family
ID=26287218
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR1019850000417A KR850005422A (ko) | 1984-01-24 | 1985-01-23 | 트리아졸 유도체의 제조방법 |
Country Status (13)
Country | Link |
---|---|
EP (1) | EP0153803A3 (ko) |
KR (1) | KR850005422A (ko) |
AU (1) | AU3799085A (ko) |
DK (1) | DK30085A (ko) |
ES (2) | ES8604901A1 (ko) |
FI (1) | FI850295L (ko) |
GR (1) | GR850159B (ko) |
HU (1) | HU192296B (ko) |
IL (1) | IL74121A0 (ko) |
PH (1) | PH20855A (ko) |
PL (1) | PL251640A1 (ko) |
PT (1) | PT79852B (ko) |
YU (1) | YU9385A (ko) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB2156807A (en) * | 1984-04-05 | 1985-10-16 | Ici Plc | Azolyl propanols |
EP0228995A1 (de) * | 1985-12-20 | 1987-07-15 | Ciba-Geigy Ag | Mikrobizide |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1529818A (en) * | 1975-12-03 | 1978-10-25 | Ici Ltd | 1,2,4-triazolyl alkanols and their use as pesticides |
US4413003A (en) * | 1977-07-29 | 1983-11-01 | Rohm And Haas Company | β-Hydroxyarylethylimidazoles |
DE3010093A1 (de) * | 1980-03-15 | 1981-10-01 | Basf Ag, 6700 Ludwigshafen | 1,1-diphenyl-2-(1.2.4-triazol-1-yl)-aethan-1-ole, verfahren zu ihrer herstellung und diese enthaltende therapeutische mittel |
-
1985
- 1985-01-15 PH PH31720A patent/PH20855A/en unknown
- 1985-01-21 PT PT79852A patent/PT79852B/pt unknown
- 1985-01-21 ES ES539723A patent/ES8604901A1/es not_active Expired
- 1985-01-21 GR GR850159A patent/GR850159B/el unknown
- 1985-01-22 PL PL25164085A patent/PL251640A1/xx unknown
- 1985-01-22 IL IL74121A patent/IL74121A0/xx unknown
- 1985-01-22 EP EP85300401A patent/EP0153803A3/en not_active Withdrawn
- 1985-01-23 DK DK30085A patent/DK30085A/da not_active Application Discontinuation
- 1985-01-23 AU AU37990/85A patent/AU3799085A/en not_active Abandoned
- 1985-01-23 KR KR1019850000417A patent/KR850005422A/ko not_active Application Discontinuation
- 1985-01-23 YU YU00093/85A patent/YU9385A/xx unknown
- 1985-01-23 FI FI850295A patent/FI850295L/fi not_active Application Discontinuation
- 1985-01-23 HU HU85268A patent/HU192296B/hu unknown
- 1985-10-29 ES ES548322A patent/ES8606300A1/es not_active Expired
Also Published As
Publication number | Publication date |
---|---|
PT79852A (en) | 1985-02-01 |
EP0153803A2 (en) | 1985-09-04 |
FI850295L (fi) | 1985-07-25 |
ES8604901A1 (es) | 1986-03-01 |
HUT38325A (en) | 1986-05-28 |
PH20855A (en) | 1987-05-19 |
FI850295A0 (fi) | 1985-01-23 |
ES539723A0 (es) | 1986-03-01 |
HU192296B (en) | 1987-05-28 |
ES8606300A1 (es) | 1986-04-16 |
PT79852B (en) | 1986-12-18 |
DK30085A (da) | 1985-07-25 |
IL74121A0 (en) | 1985-04-30 |
YU9385A (en) | 1987-06-30 |
PL251640A1 (en) | 1985-10-08 |
EP0153803A3 (en) | 1986-09-03 |
AU3799085A (en) | 1985-08-01 |
ES548322A0 (es) | 1986-04-16 |
DK30085D0 (da) | 1985-01-23 |
GR850159B (ko) | 1985-05-23 |
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E902 | Notification of reason for refusal | ||
E601 | Decision to refuse application |