JPWO2023126436A5 - - Google Patents

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Publication number
JPWO2023126436A5
JPWO2023126436A5 JP2024539928A JP2024539928A JPWO2023126436A5 JP WO2023126436 A5 JPWO2023126436 A5 JP WO2023126436A5 JP 2024539928 A JP2024539928 A JP 2024539928A JP 2024539928 A JP2024539928 A JP 2024539928A JP WO2023126436 A5 JPWO2023126436 A5 JP WO2023126436A5
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JP
Japan
Prior art keywords
formula
crystalline form
monohydrate
compound
alpha
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024539928A
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English (en)
Japanese (ja)
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JP2025502842A5 (https=
JP2025502842A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2022/087952 external-priority patent/WO2023126436A1/en
Publication of JP2025502842A publication Critical patent/JP2025502842A/ja
Publication of JP2025502842A5 publication Critical patent/JP2025502842A5/ja
Publication of JPWO2023126436A5 publication Critical patent/JPWO2023126436A5/ja
Pending legal-status Critical Current

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JP2024539928A 2021-12-29 2022-12-28 薬学的に活性な化合物としての使用のための(5s)-{[2-(4-カルボキシフェニル)エチル][2-(2-{[3-クロロ-4’-(トリフルオロメチル)ビフェニル-4-イル]メトキシ}フェニル)エチル]アミノ}-5,6,7,8-テトラヒドロキノリン-2-カルボン酸及びその結晶形態を調製するための方法 Pending JP2025502842A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP21218163.0 2021-12-29
EP21218163 2021-12-29
PCT/EP2022/087952 WO2023126436A1 (en) 2021-12-29 2022-12-28 Process for preparing (5s)-{[2-(4-carboxyphenyl)ethyl] |2-(2-{|3-chloro-4'-(trifluoromethyl)biphenyl-4- yl]methoxy}phenyl)ethyl]aminol-5,6,7,8-tetrahydroquinoline-2-carboxylic acid and its crystalline forms for use as pharmaceutically active compound

Publications (3)

Publication Number Publication Date
JP2025502842A JP2025502842A (ja) 2025-01-28
JP2025502842A5 JP2025502842A5 (https=) 2026-01-09
JPWO2023126436A5 true JPWO2023126436A5 (https=) 2026-01-09

Family

ID=79185525

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024539928A Pending JP2025502842A (ja) 2021-12-29 2022-12-28 薬学的に活性な化合物としての使用のための(5s)-{[2-(4-カルボキシフェニル)エチル][2-(2-{[3-クロロ-4’-(トリフルオロメチル)ビフェニル-4-イル]メトキシ}フェニル)エチル]アミノ}-5,6,7,8-テトラヒドロキノリン-2-カルボン酸及びその結晶形態を調製するための方法

Country Status (12)

Country Link
US (2) US12202805B2 (https=)
EP (1) EP4457215A1 (https=)
JP (1) JP2025502842A (https=)
KR (1) KR20240144177A (https=)
CN (1) CN118765272A (https=)
AR (1) AR128147A1 (https=)
AU (1) AU2022429647A1 (https=)
CA (1) CA3244893A1 (https=)
IL (1) IL313922A (https=)
MX (1) MX2024008172A (https=)
TW (1) TW202342012A (https=)
WO (1) WO2023126436A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN118765199A (zh) 2021-12-29 2024-10-11 拜耳股份公司 心肺病症的治疗
TW202342012A (zh) 2021-12-29 2023-11-01 德商拜耳廠股份有限公司 製備用作醫藥活性化合物的(5s)-{[2-(4-羧基苯基)乙基][2-(2-{[3-氯-4'-(三氟甲基)聯苯-4-基]甲氧基}苯基)乙基]胺基}-5,6,7,8-四氫喹啉-2-羧酸及其結晶形式之方法

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CN118765199A (zh) 2021-12-29 2024-10-11 拜耳股份公司 心肺病症的治疗
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