JPWO2023084206A5 - - Google Patents

Info

Publication number
JPWO2023084206A5
JPWO2023084206A5 JP2024526654A JP2024526654A JPWO2023084206A5 JP WO2023084206 A5 JPWO2023084206 A5 JP WO2023084206A5 JP 2024526654 A JP2024526654 A JP 2024526654A JP 2024526654 A JP2024526654 A JP 2024526654A JP WO2023084206 A5 JPWO2023084206 A5 JP WO2023084206A5
Authority
JP
Japan
Prior art keywords
cyclohexyl
carboxamide
methyl
imidazol
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024526654A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024540318A (ja
JP2024540318A5 (https=
Publication date
Application filed filed Critical
Priority claimed from PCT/GB2022/052833 external-priority patent/WO2023084206A1/en
Publication of JP2024540318A publication Critical patent/JP2024540318A/ja
Publication of JPWO2023084206A5 publication Critical patent/JPWO2023084206A5/ja
Publication of JP2024540318A5 publication Critical patent/JP2024540318A5/ja
Pending legal-status Critical Current

Links

JP2024526654A 2021-11-09 2022-11-09 Cd38阻害剤としてのn-(4-アミノシクロヘキシル)ピリミジン-4-カルボキサミド誘導体 Pending JP2024540318A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB202116077 2021-11-09
GB2116077.5 2021-11-09
PCT/GB2022/052833 WO2023084206A1 (en) 2021-11-09 2022-11-09 N-(4-aminocyclohexyl)pyrimidine-4-carboxamide derivatives as cd38 inhibitors

Publications (3)

Publication Number Publication Date
JP2024540318A JP2024540318A (ja) 2024-10-31
JPWO2023084206A5 true JPWO2023084206A5 (https=) 2025-11-18
JP2024540318A5 JP2024540318A5 (https=) 2025-11-18

Family

ID=84360092

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024526654A Pending JP2024540318A (ja) 2021-11-09 2022-11-09 Cd38阻害剤としてのn-(4-アミノシクロヘキシル)ピリミジン-4-カルボキサミド誘導体

Country Status (6)

Country Link
US (1) US20250019369A1 (https=)
EP (1) EP4430034A1 (https=)
JP (1) JP2024540318A (https=)
CN (1) CN118317955A (https=)
CA (1) CA3236793A1 (https=)
WO (1) WO2023084206A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023235880A1 (en) * 2022-06-02 2023-12-07 Aeovian Pharmaceuticals, Inc. Cd38 modulators and uses thereof
AU2024285368A1 (en) * 2023-06-07 2025-12-18 Flagship Pioneering Innovations Vi, Llc Condensed azines as inhibitors of cyclic adp ribose hydrolase
WO2026000074A1 (en) * 2024-06-25 2026-01-02 Welnx Company Inc. Use of cd38 inhibitors for reducing th2 inflammation
WO2026075971A1 (en) 2024-10-01 2026-04-09 Neolaia Inc. Combination therapy for treatment of metabolic disorders and inflamation related disorders using incretin compounds and cd38 inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021021986A1 (en) 2019-07-31 2021-02-04 Ribon Therapeutics, Inc. Heterobicyclic amides as inhibitors of cd38
BR112022020291A2 (pt) * 2020-04-07 2022-12-06 Mitobridge Inc Inibidores de cd38
US20240254113A1 (en) * 2021-04-30 2024-08-01 Nanjing Immunophage Biotech Co., Ltd. Compounds and their uses as cd38 inhibitors

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