JPWO2022256680A5 - - Google Patents

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Publication number
JPWO2022256680A5
JPWO2022256680A5 JP2024518956A JP2024518956A JPWO2022256680A5 JP WO2022256680 A5 JPWO2022256680 A5 JP WO2022256680A5 JP 2024518956 A JP2024518956 A JP 2024518956A JP 2024518956 A JP2024518956 A JP 2024518956A JP WO2022256680 A5 JPWO2022256680 A5 JP WO2022256680A5
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JP
Japan
Prior art keywords
cancer
compound
alkyl
tumor
formula
Prior art date
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Pending
Application number
JP2024518956A
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English (en)
Japanese (ja)
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JP2024522304A5 (https=
JP2024522304A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/032203 external-priority patent/WO2022256680A1/en
Publication of JP2024522304A publication Critical patent/JP2024522304A/ja
Publication of JP2024522304A5 publication Critical patent/JP2024522304A5/ja
Publication of JPWO2022256680A5 publication Critical patent/JPWO2022256680A5/ja
Pending legal-status Critical Current

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JP2024518956A 2021-06-04 2022-06-03 Wee1キナーゼ阻害剤として有用なピリドピリミジン誘導体 Pending JP2024522304A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163196744P 2021-06-04 2021-06-04
US63/196,744 2021-06-04
PCT/US2022/032203 WO2022256680A1 (en) 2021-06-04 2022-06-03 Pyridopyrimidine derivatives useful as wee1 kinase inhibitors

Publications (3)

Publication Number Publication Date
JP2024522304A JP2024522304A (ja) 2024-06-13
JP2024522304A5 JP2024522304A5 (https=) 2025-06-10
JPWO2022256680A5 true JPWO2022256680A5 (https=) 2025-06-10

Family

ID=82321319

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024518956A Pending JP2024522304A (ja) 2021-06-04 2022-06-03 Wee1キナーゼ阻害剤として有用なピリドピリミジン誘導体

Country Status (10)

Country Link
US (1) US20240254123A1 (https=)
EP (1) EP4347592A1 (https=)
JP (1) JP2024522304A (https=)
KR (1) KR20240044409A (https=)
CN (1) CN117794932A (https=)
AU (2) AU2022287033B2 (https=)
CA (1) CA3225152A1 (https=)
IL (1) IL309037A (https=)
MX (1) MX2023014466A (https=)
WO (1) WO2022256680A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL315441A (en) 2022-03-07 2024-11-01 Debiopharm Int Sa Treatment methods for small cell lung cancer
IL326854A (en) 2023-09-14 2026-04-01 Debiopharm Int Sa Combination of WEE1 inhibitor and PKMYT1 inhibitor
CN120189510A (zh) * 2023-12-21 2025-06-24 北京哲源科技有限责任公司 一种并环化合物的应用
TW202541810A (zh) 2023-12-22 2025-11-01 瑞士商德彪製藥國際公司 治療實體腫瘤之方法
WO2025186213A1 (en) 2024-03-04 2025-09-12 Debiopharm International S.A. Combination of a wee1 inhibitor and a topoisomerase 1 inhibitor

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002098370A2 (en) 2001-03-02 2002-12-12 Medimmune, Inc. Methods of administering/dosing cd2 antagonists for the prevention and treatment of autoimmune disorders or inflammatory disorders
AR060635A1 (es) * 2006-04-27 2008-07-02 Banyu Pharma Co Ltd Derivados de 1,2-dihidro-3h-pirazolo[3,4-d]pirimidin-3-ona, composiciones farmaceuticas que los comprenden y su uso en el tratamiento del cancer
CN104271576A (zh) * 2012-02-23 2015-01-07 艾伯维公司 激酶的吡啶并嘧啶酮抑制剂
GB201306610D0 (en) * 2013-04-11 2013-05-29 Almac Discovery Ltd Pharmaceutical compounds
GB201612095D0 (en) * 2016-07-12 2016-08-24 Almac Discovery Ltd Pharmaceutical compounds
CA3071405A1 (en) * 2017-08-01 2019-02-07 Recurium Ip Holdings, Llc 1, 2 - dihydro- 3h- pyrazolo [3, 4 - d] pyrimidin -3 - one analogs
GB201800378D0 (en) * 2018-01-10 2018-02-21 Almac Discovery Ltd Pharmaceutical compounds

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