JPWO2022117477A5 - - Google Patents

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Publication number
JPWO2022117477A5
JPWO2022117477A5 JP2023527318A JP2023527318A JPWO2022117477A5 JP WO2022117477 A5 JPWO2022117477 A5 JP WO2022117477A5 JP 2023527318 A JP2023527318 A JP 2023527318A JP 2023527318 A JP2023527318 A JP 2023527318A JP WO2022117477 A5 JPWO2022117477 A5 JP WO2022117477A5
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JP
Japan
Prior art keywords
methyl
compound according
hydroxymethyl
indazol
thiazol
Prior art date
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Application number
JP2023527318A
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English (en)
Japanese (ja)
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JP2023550902A5 (https=
JP7840327B2 (ja
JP2023550902A (ja
Publication date
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Priority claimed from PCT/EP2021/083279 external-priority patent/WO2022117477A1/en
Publication of JP2023550902A publication Critical patent/JP2023550902A/ja
Publication of JP2023550902A5 publication Critical patent/JP2023550902A5/ja
Publication of JPWO2022117477A5 publication Critical patent/JPWO2022117477A5/ja
Application granted granted Critical
Publication of JP7840327B2 publication Critical patent/JP7840327B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2023527318A 2020-12-01 2021-11-29 新規インダゾールアセチレン誘導体 Active JP7840327B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP20210859 2020-12-01
EP20210859.3 2020-12-01
PCT/EP2021/083279 WO2022117477A1 (en) 2020-12-01 2021-11-29 New indazole acetylene derivatives

Publications (4)

Publication Number Publication Date
JP2023550902A JP2023550902A (ja) 2023-12-06
JP2023550902A5 JP2023550902A5 (https=) 2024-12-04
JPWO2022117477A5 true JPWO2022117477A5 (https=) 2024-12-04
JP7840327B2 JP7840327B2 (ja) 2026-04-03

Family

ID=73654642

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023527318A Active JP7840327B2 (ja) 2020-12-01 2021-11-29 新規インダゾールアセチレン誘導体

Country Status (15)

Country Link
US (1) US20240002390A1 (https=)
EP (1) EP4255908A1 (https=)
JP (1) JP7840327B2 (https=)
KR (1) KR20230116799A (https=)
CN (1) CN116490182A (https=)
AR (1) AR124170A1 (https=)
AU (1) AU2021393722A1 (https=)
CA (1) CA3197659A1 (https=)
CL (1) CL2023001440A1 (https=)
CO (1) CO2023006912A2 (https=)
CR (1) CR20230218A (https=)
IL (1) IL303064A (https=)
MX (1) MX2023006176A (https=)
PE (1) PE20240099A1 (https=)
WO (1) WO2022117477A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114008049B (zh) 2019-06-21 2024-07-05 豪夫迈·罗氏有限公司 用于癌症治疗的egfr抑制剂
JP7840324B2 (ja) 2020-12-01 2026-04-03 エフ・ホフマン-ラ・ロシュ・アクチェンゲゼルシャフト 新規インダゾール誘導体
JP2025516543A (ja) * 2022-05-13 2025-05-30 エフ・ホフマン-ラ・ロシュ・アクチェンゲゼルシャフト がんの治療のためのアロステリックおよびオルソステリックegfr阻害剤の組み合わせ

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2987914C (en) * 2015-06-30 2022-09-13 Dana-Farber Cancer Institute, Inc. Inhibitors of egfr and methods of use thereof
TW201834651A (zh) * 2016-12-22 2018-10-01 瑞士商赫孚孟拉羅股份公司 化合物
WO2018220149A1 (en) * 2017-06-02 2018-12-06 F. Hoffmann-La Roche Ag Compounds
SG11202011818YA (en) * 2018-06-29 2020-12-30 Hoffmann La Roche Compounds
CN113993591A (zh) * 2019-06-21 2022-01-28 豪夫迈·罗氏有限公司 新egfr抑制剂

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