JPWO2022040293A5 - - Google Patents

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Publication number
JPWO2022040293A5
JPWO2022040293A5 JP2023512161A JP2023512161A JPWO2022040293A5 JP WO2022040293 A5 JPWO2022040293 A5 JP WO2022040293A5 JP 2023512161 A JP2023512161 A JP 2023512161A JP 2023512161 A JP2023512161 A JP 2023512161A JP WO2022040293 A5 JPWO2022040293 A5 JP WO2022040293A5
Authority
JP
Japan
Prior art keywords
phenyl
methyl
pyrrolo
pyridine
methylsulfonyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023512161A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023539136A (ja
JP2023539136A5 (https=
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/046475 external-priority patent/WO2022040293A1/en
Publication of JP2023539136A publication Critical patent/JP2023539136A/ja
Publication of JP2023539136A5 publication Critical patent/JP2023539136A5/ja
Publication of JPWO2022040293A5 publication Critical patent/JPWO2022040293A5/ja
Pending legal-status Critical Current

Links

JP2023512161A 2020-08-19 2021-08-18 Tlr9阻害剤として有用な置換ヘテロアリール化合物 Pending JP2023539136A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063067389P 2020-08-19 2020-08-19
US63/067,389 2020-08-19
PCT/US2021/046475 WO2022040293A1 (en) 2020-08-19 2021-08-18 Substituted heteroaryl compounds useful as inhibitors of tlr9

Publications (3)

Publication Number Publication Date
JP2023539136A JP2023539136A (ja) 2023-09-13
JP2023539136A5 JP2023539136A5 (https=) 2024-08-26
JPWO2022040293A5 true JPWO2022040293A5 (https=) 2024-08-26

Family

ID=77726550

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023512161A Pending JP2023539136A (ja) 2020-08-19 2021-08-18 Tlr9阻害剤として有用な置換ヘテロアリール化合物

Country Status (16)

Country Link
US (1) US20230322770A1 (https=)
EP (1) EP4200015B1 (https=)
JP (1) JP2023539136A (https=)
KR (1) KR20230052930A (https=)
CN (1) CN115956077A (https=)
AR (1) AR123284A1 (https=)
AU (1) AU2021328362A1 (https=)
BR (1) BR112023002662A2 (https=)
CA (1) CA3189816A1 (https=)
CL (1) CL2023000428A1 (https=)
CO (1) CO2023001670A2 (https=)
IL (1) IL300696A (https=)
MX (1) MX2023001883A (https=)
PE (1) PE20231318A1 (https=)
TW (1) TW202227431A (https=)
WO (1) WO2022040293A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022140325A1 (en) * 2020-12-22 2022-06-30 Gilead Sciences, Inc. 6-substituted indole compounds
TWI838670B (zh) * 2020-12-22 2024-04-11 美商基利科學股份有限公司 經取代之吲哚化合物
CR20230478A (es) 2021-04-16 2023-11-30 Gilead Sciences Inc Compuestos de tienopirrol.
KR20240056747A (ko) 2021-09-10 2024-04-30 길리애드 사이언시즈, 인코포레이티드 티에노피롤 화합물
MX2024009441A (es) * 2022-02-18 2024-08-14 Bristol Myers Squibb Co Compuestos de imidazopiridinilo sustituidos utiles como inhibidores del receptor tipo toll 9 (tlr9).
WO2024102886A1 (en) * 2022-11-10 2024-05-16 Bristol-Myers Squibb Company Substituted benzimidazole compounds useful as inhibitors of tlr9
KR20250094727A (ko) * 2022-11-10 2025-06-25 브리스톨-마이어스 스큅 컴퍼니 Tlr9의 억제제로서 유용한 치환된 퀴놀론 화합물

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013092467A1 (en) * 2011-12-20 2013-06-27 F. Hoffmann-La Roche Ag 7-azaindole inhibitors of crac
CN105992766A (zh) * 2013-12-13 2016-10-05 武田药品工业株式会社 作为tlr抑制剂的吡咯并[3,2-c]吡啶衍生物
TW201630907A (zh) * 2014-12-22 2016-09-01 必治妥美雅史谷比公司 TGFβR拮抗劑
EA202091484A1 (ru) * 2017-12-18 2021-03-25 Бристол-Маерс Сквибб Компани 4-азаиндольные соединения
JP7304352B2 (ja) * 2017-12-19 2023-07-06 ブリストル-マイヤーズ スクイブ カンパニー 6-アザインドール化合物
KR102730859B1 (ko) * 2017-12-20 2024-11-15 브리스톨-마이어스 스큅 컴퍼니 아릴 및 헤테로아릴 치환된 인돌 화합물

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