JPWO2022040293A5 - - Google Patents
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- Publication number
- JPWO2022040293A5 JPWO2022040293A5 JP2023512161A JP2023512161A JPWO2022040293A5 JP WO2022040293 A5 JPWO2022040293 A5 JP WO2022040293A5 JP 2023512161 A JP2023512161 A JP 2023512161A JP 2023512161 A JP2023512161 A JP 2023512161A JP WO2022040293 A5 JPWO2022040293 A5 JP WO2022040293A5
- Authority
- JP
- Japan
- Prior art keywords
- phenyl
- methyl
- pyrrolo
- pyridine
- methylsulfonyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202063067389P | 2020-08-19 | 2020-08-19 | |
| US63/067,389 | 2020-08-19 | ||
| PCT/US2021/046475 WO2022040293A1 (en) | 2020-08-19 | 2021-08-18 | Substituted heteroaryl compounds useful as inhibitors of tlr9 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023539136A JP2023539136A (ja) | 2023-09-13 |
| JP2023539136A5 JP2023539136A5 (https=) | 2024-08-26 |
| JPWO2022040293A5 true JPWO2022040293A5 (https=) | 2024-08-26 |
Family
ID=77726550
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023512161A Pending JP2023539136A (ja) | 2020-08-19 | 2021-08-18 | Tlr9阻害剤として有用な置換ヘテロアリール化合物 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20230322770A1 (https=) |
| EP (1) | EP4200015B1 (https=) |
| JP (1) | JP2023539136A (https=) |
| KR (1) | KR20230052930A (https=) |
| CN (1) | CN115956077A (https=) |
| AR (1) | AR123284A1 (https=) |
| AU (1) | AU2021328362A1 (https=) |
| BR (1) | BR112023002662A2 (https=) |
| CA (1) | CA3189816A1 (https=) |
| CL (1) | CL2023000428A1 (https=) |
| CO (1) | CO2023001670A2 (https=) |
| IL (1) | IL300696A (https=) |
| MX (1) | MX2023001883A (https=) |
| PE (1) | PE20231318A1 (https=) |
| TW (1) | TW202227431A (https=) |
| WO (1) | WO2022040293A1 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2022140325A1 (en) * | 2020-12-22 | 2022-06-30 | Gilead Sciences, Inc. | 6-substituted indole compounds |
| TWI838670B (zh) * | 2020-12-22 | 2024-04-11 | 美商基利科學股份有限公司 | 經取代之吲哚化合物 |
| CR20230478A (es) | 2021-04-16 | 2023-11-30 | Gilead Sciences Inc | Compuestos de tienopirrol. |
| KR20240056747A (ko) | 2021-09-10 | 2024-04-30 | 길리애드 사이언시즈, 인코포레이티드 | 티에노피롤 화합물 |
| MX2024009441A (es) * | 2022-02-18 | 2024-08-14 | Bristol Myers Squibb Co | Compuestos de imidazopiridinilo sustituidos utiles como inhibidores del receptor tipo toll 9 (tlr9). |
| WO2024102886A1 (en) * | 2022-11-10 | 2024-05-16 | Bristol-Myers Squibb Company | Substituted benzimidazole compounds useful as inhibitors of tlr9 |
| KR20250094727A (ko) * | 2022-11-10 | 2025-06-25 | 브리스톨-마이어스 스큅 컴퍼니 | Tlr9의 억제제로서 유용한 치환된 퀴놀론 화합물 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2013092467A1 (en) * | 2011-12-20 | 2013-06-27 | F. Hoffmann-La Roche Ag | 7-azaindole inhibitors of crac |
| CN105992766A (zh) * | 2013-12-13 | 2016-10-05 | 武田药品工业株式会社 | 作为tlr抑制剂的吡咯并[3,2-c]吡啶衍生物 |
| TW201630907A (zh) * | 2014-12-22 | 2016-09-01 | 必治妥美雅史谷比公司 | TGFβR拮抗劑 |
| EA202091484A1 (ru) * | 2017-12-18 | 2021-03-25 | Бристол-Маерс Сквибб Компани | 4-азаиндольные соединения |
| JP7304352B2 (ja) * | 2017-12-19 | 2023-07-06 | ブリストル-マイヤーズ スクイブ カンパニー | 6-アザインドール化合物 |
| KR102730859B1 (ko) * | 2017-12-20 | 2024-11-15 | 브리스톨-마이어스 스큅 컴퍼니 | 아릴 및 헤테로아릴 치환된 인돌 화합물 |
-
2021
- 2021-08-18 WO PCT/US2021/046475 patent/WO2022040293A1/en not_active Ceased
- 2021-08-18 PE PE2023000276A patent/PE20231318A1/es unknown
- 2021-08-18 BR BR112023002662A patent/BR112023002662A2/pt unknown
- 2021-08-18 KR KR1020237009018A patent/KR20230052930A/ko active Pending
- 2021-08-18 JP JP2023512161A patent/JP2023539136A/ja active Pending
- 2021-08-18 MX MX2023001883A patent/MX2023001883A/es unknown
- 2021-08-18 TW TW110130426A patent/TW202227431A/zh unknown
- 2021-08-18 US US18/042,018 patent/US20230322770A1/en active Pending
- 2021-08-18 AR ARP210102328A patent/AR123284A1/es not_active Application Discontinuation
- 2021-08-18 AU AU2021328362A patent/AU2021328362A1/en not_active Abandoned
- 2021-08-18 CA CA3189816A patent/CA3189816A1/en active Pending
- 2021-08-18 EP EP21769573.3A patent/EP4200015B1/en active Active
- 2021-08-18 CN CN202180050343.7A patent/CN115956077A/zh active Pending
- 2021-08-18 IL IL300696A patent/IL300696A/en unknown
-
2023
- 2023-02-10 CL CL2023000428A patent/CL2023000428A1/es unknown
- 2023-02-15 CO CONC2023/0001670A patent/CO2023001670A2/es unknown
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