JPWO2021099518A5 - - Google Patents
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- Publication number
- JPWO2021099518A5 JPWO2021099518A5 JP2022554964A JP2022554964A JPWO2021099518A5 JP WO2021099518 A5 JPWO2021099518 A5 JP WO2021099518A5 JP 2022554964 A JP2022554964 A JP 2022554964A JP 2022554964 A JP2022554964 A JP 2022554964A JP WO2021099518 A5 JPWO2021099518 A5 JP WO2021099518A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- compound
- compound according
- solvate
- salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP19210073 | 2019-11-19 | ||
| EP19210073.3 | 2019-11-19 | ||
| PCT/EP2020/082778 WO2021099518A1 (en) | 2019-11-19 | 2020-11-19 | Novel compounds for the diagnosis, treatment and prevention of diseases associated with the aggregation of alpha-synuclein |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2023502794A JP2023502794A (ja) | 2023-01-25 |
| JPWO2021099518A5 true JPWO2021099518A5 (https=) | 2023-04-04 |
| JP2023502794A5 JP2023502794A5 (https=) | 2023-04-04 |
| JP7652791B2 JP7652791B2 (ja) | 2025-03-27 |
Family
ID=68834924
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022554964A Active JP7652791B2 (ja) | 2019-11-19 | 2020-11-19 | α－シヌクレインの凝集に関連する疾患の診断、治療および予防のための新規な化合物 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20230067910A1 (https=) |
| EP (2) | EP4061807A1 (https=) |
| JP (1) | JP7652791B2 (https=) |
| KR (1) | KR20220104000A (https=) |
| CN (1) | CN114728927B (https=) |
| AU (2) | AU2020386151B2 (https=) |
| BR (1) | BR112022008195A2 (https=) |
| CA (1) | CA3160364C (https=) |
| CL (1) | CL2022001302A1 (https=) |
| IL (1) | IL292919B1 (https=) |
| MX (1) | MX2022005914A (https=) |
| PH (1) | PH12022551224A1 (https=) |
| WO (1) | WO2021099518A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20210061202A (ko) | 2019-11-19 | 2021-05-27 | 일동제약(주) | 벤조나이트릴이 치환된 축합 피리미딘 유도체 및 그의 의약 용도 |
Family Cites Families (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3773919A (en) | 1969-10-23 | 1973-11-20 | Du Pont | Polylactide-drug mixtures |
| US4263428A (en) | 1978-03-24 | 1981-04-21 | The Regents Of The University Of California | Bis-anthracycline nucleic acid function inhibitors and improved method for administering the same |
| EP0052322B1 (de) | 1980-11-10 | 1985-03-27 | Gersonde, Klaus, Prof. Dr. | Verfahren zur Herstellung von Lipid-Vesikeln durch Ultraschallbehandlung, Anwendung des Verfahrens und Vorrichtung zur Durchführung des Verfahrens |
| IE52535B1 (en) | 1981-02-16 | 1987-12-09 | Ici Plc | Continuous release pharmaceutical compositions |
| US4485045A (en) | 1981-07-06 | 1984-11-27 | Research Corporation | Synthetic phosphatidyl cholines useful in forming liposomes |
| DE3374837D1 (en) | 1982-02-17 | 1988-01-21 | Ciba Geigy Ag | Lipids in the aqueous phase |
| DE3218121A1 (de) | 1982-05-14 | 1983-11-17 | Leskovar, Peter, Dr.-Ing., 8000 München | Arzneimittel zur tumorbehandlung |
| EP0102324A3 (de) | 1982-07-29 | 1984-11-07 | Ciba-Geigy Ag | Lipide und Tenside in wässriger Phase |
| US4544545A (en) | 1983-06-20 | 1985-10-01 | Trustees University Of Massachusetts | Liposomes containing modified cholesterol for organ targeting |
| HUT35524A (en) | 1983-08-02 | 1985-07-29 | Hoechst Ag | Process for preparing pharmaceutical compositions containing regulatory /regulative/ peptides providing for the retarded release of the active substance |
| DE3483949D1 (de) | 1983-09-26 | 1991-02-21 | Udo Dr Med Ehrenfeld | Mittel und erzeugnis fuer die diagnose und therapie von tumoren sowie zur behandlung von schwaechen der zelligen und humoralen immunabwehr. |
| EP0143949B1 (en) | 1983-11-01 | 1988-10-12 | TERUMO KABUSHIKI KAISHA trading as TERUMO CORPORATION | Pharmaceutical composition containing urokinase |
| AU2935200A (en) | 1999-04-30 | 2000-11-17 | Pfizer Products Inc. | Compounds for the treatment of obesity |
| US6660753B2 (en) * | 1999-08-19 | 2003-12-09 | Nps Pharmaceuticals, Inc. | Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
| US8829198B2 (en) * | 2007-10-31 | 2014-09-09 | Proteotech Inc | Compounds, compositions and methods for the treatment of beta-amyloid diseases and synucleinopathies |
| US20050075375A1 (en) * | 2003-05-14 | 2005-04-07 | Anadys Pharmaceuticals, Inc. | Heterocyclic compounds for treating hepatitis C virus |
| DE102008020113A1 (de) * | 2008-04-23 | 2009-10-29 | Bayer Schering Pharma Aktiengesellschaft | Substituierte Dihydropyrazolone und ihre Verwendung |
| PL2004155T3 (pl) * | 2006-03-29 | 2018-08-31 | Wista Laboratories Ltd. | Inhibitory agregacji białek |
| US20110201686A1 (en) * | 2006-06-23 | 2011-08-18 | Yousef Al-Abed | Inhibitors of ASS and Synuclein Aggregation |
| JP4616237B2 (ja) | 2006-11-07 | 2011-01-19 | 日本電信電話株式会社 | シリコン化合物薄膜の形成方法 |
| CN102047061A (zh) * | 2008-05-30 | 2011-05-04 | 福斯特韦勒能源股份公司 | 通过氧化燃料燃烧发电的方法和系统 |
| US20110293520A1 (en) * | 2008-06-09 | 2011-12-01 | Max-Planck-Gesellschaft Zur Forderung Der Wissenschaften E.V. | New drug for inhibiting aggregation of proteins involved in diseases linked to protein aggregation and/or neurodegenerative diseases |
| TW201120016A (en) | 2009-12-08 | 2011-06-16 | Abbott Lab | Novel oxadiazole compounds |
| PL3390412T3 (pl) * | 2015-12-14 | 2021-10-25 | MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. | Rozpuszczalne w wodzie pochodne związków 3,5-difenylodiazolowych |
| NZ746901A (en) * | 2016-03-11 | 2023-06-30 | Ac Immune Sa | Bicyclic compounds for diagnosis and therapy |
| WO2019208509A1 (en) | 2018-04-23 | 2019-10-31 | Shionogi & Co., Ltd. | Bicyclic heterocycle derivatives having selective bace1 inhibitory activity |
-
2020
- 2020-11-19 MX MX2022005914A patent/MX2022005914A/es unknown
- 2020-11-19 EP EP20810960.3A patent/EP4061807A1/en active Pending
- 2020-11-19 BR BR112022008195A patent/BR112022008195A2/pt unknown
- 2020-11-19 WO PCT/EP2020/082778 patent/WO2021099518A1/en not_active Ceased
- 2020-11-19 CN CN202080080990.8A patent/CN114728927B/zh active Active
- 2020-11-19 EP EP24166495.2A patent/EP4368184A3/en active Pending
- 2020-11-19 CA CA3160364A patent/CA3160364C/en active Active
- 2020-11-19 JP JP2022554964A patent/JP7652791B2/ja active Active
- 2020-11-19 US US17/777,571 patent/US20230067910A1/en active Pending
- 2020-11-19 PH PH1/2022/551224A patent/PH12022551224A1/en unknown
- 2020-11-19 AU AU2020386151A patent/AU2020386151B2/en active Active
- 2020-11-19 KR KR1020227020703A patent/KR20220104000A/ko not_active Ceased
-
2022
- 2022-05-10 IL IL292919A patent/IL292919B1/en unknown
- 2022-05-18 CL CL2022001302A patent/CL2022001302A1/es unknown
-
2023
- 2023-12-19 AU AU2023285721A patent/AU2023285721B2/en active Active
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