JPWO2021087113A5 - - Google Patents

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Publication number
JPWO2021087113A5
JPWO2021087113A5 JP2022525711A JP2022525711A JPWO2021087113A5 JP WO2021087113 A5 JPWO2021087113 A5 JP WO2021087113A5 JP 2022525711 A JP2022525711 A JP 2022525711A JP 2022525711 A JP2022525711 A JP 2022525711A JP WO2021087113 A5 JPWO2021087113 A5 JP WO2021087113A5
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JP
Japan
Prior art keywords
substituted
unsubstituted alkyl
unsubstituted
compound
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2022525711A
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English (en)
Japanese (ja)
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JP2023500682A5 (https=
JP2023500682A (ja
JP7803855B2 (ja
Publication date
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Priority claimed from PCT/US2020/057963 external-priority patent/WO2021087113A1/en
Publication of JP2023500682A publication Critical patent/JP2023500682A/ja
Publication of JP2023500682A5 publication Critical patent/JP2023500682A5/ja
Publication of JPWO2021087113A5 publication Critical patent/JPWO2021087113A5/ja
Priority to JP2025135404A priority Critical patent/JP2026004274A/ja
Application granted granted Critical
Publication of JP7803855B2 publication Critical patent/JP7803855B2/ja
Active legal-status Critical Current
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JP2022525711A 2019-10-30 2020-10-29 選択的な感覚神経の遮断のある局所麻酔薬 Active JP7803855B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025135404A JP2026004274A (ja) 2019-10-30 2025-08-15 選択的な感覚神経の遮断のある局所麻酔薬

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201962928177P 2019-10-30 2019-10-30
US62/928,177 2019-10-30
US201962941624P 2019-11-27 2019-11-27
US62/941,624 2019-11-27
PCT/US2020/057963 WO2021087113A1 (en) 2019-10-30 2020-10-29 Local anesthetics with selective-sensory nerve blockade

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025135404A Division JP2026004274A (ja) 2019-10-30 2025-08-15 選択的な感覚神経の遮断のある局所麻酔薬

Publications (4)

Publication Number Publication Date
JP2023500682A JP2023500682A (ja) 2023-01-10
JP2023500682A5 JP2023500682A5 (https=) 2023-11-08
JPWO2021087113A5 true JPWO2021087113A5 (https=) 2023-11-08
JP7803855B2 JP7803855B2 (ja) 2026-01-21

Family

ID=75714697

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022525711A Active JP7803855B2 (ja) 2019-10-30 2020-10-29 選択的な感覚神経の遮断のある局所麻酔薬
JP2025135404A Pending JP2026004274A (ja) 2019-10-30 2025-08-15 選択的な感覚神経の遮断のある局所麻酔薬

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025135404A Pending JP2026004274A (ja) 2019-10-30 2025-08-15 選択的な感覚神経の遮断のある局所麻酔薬

Country Status (6)

Country Link
US (1) US12454509B2 (https=)
EP (1) EP4051254A4 (https=)
JP (2) JP7803855B2 (https=)
AU (1) AU2020373030A1 (https=)
CA (1) CA3159752A1 (https=)
WO (1) WO2021087113A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116023322B (zh) * 2022-01-05 2025-10-31 天津键凯科技有限公司 一种n-乙酰苯胺类阳离子化合物及其制备方法和应用

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3050559A (en) 1962-08-21 Substituted phenylcyclopropylamjnes
GB866604A (en) 1958-05-31 1961-04-26 T & H Smith Ltd New quaternary salts
US3255207A (en) * 1962-02-09 1966-06-07 Astra Ab Quaternary ammonium salts containing anilido groups
US3998815A (en) 1974-06-24 1976-12-21 Interx Research Corporation 1-hydrocarbonoyloxymethyl-3-carbamoyl or 3-carboethoxy-pyridinium salts
CH618842A5 (en) 1975-09-30 1980-08-29 Ciba Geigy Ag Pesticides
WO1998024428A1 (en) 1996-12-02 1998-06-11 Brigham & Women's Hospital, Inc. Long-acting local anesthetics
CN103601650B (zh) * 2013-01-16 2014-08-06 四川大学华西医院 N-二乙氨基乙酰-2,6-二甲基苯胺衍生物、制备方法及用途
CN105315170B (zh) 2014-08-01 2017-08-25 四川大学华西医院 二甲基苯铵类长链化合物、制备、自组装结构及用途
CA3039767C (en) * 2015-12-22 2023-11-14 Arizona Board Of Regents On Behalf Of The University Of Arizona Compositions and methods for treatment, amelioration, and prevention of anesthesia-induced hypothermia
CN106928126B (zh) 2015-12-31 2019-12-20 四川海思科制药有限公司 一种酰胺衍生物及其制备方法和在药学上的应用
TWI833741B (zh) 2018-03-30 2024-03-01 日商樂敦製藥股份有限公司 外用油性固形組成物

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