JPWO2020010058A5 - - Google Patents

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Publication number
JPWO2020010058A5
JPWO2020010058A5 JP2021500178A JP2021500178A JPWO2020010058A5 JP WO2020010058 A5 JPWO2020010058 A5 JP WO2020010058A5 JP 2021500178 A JP2021500178 A JP 2021500178A JP 2021500178 A JP2021500178 A JP 2021500178A JP WO2020010058 A5 JPWO2020010058 A5 JP WO2020010058A5
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JP
Japan
Prior art keywords
ivosidenib
solid
powder
ray diffraction
diffraction pattern
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021500178A
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English (en)
Japanese (ja)
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JP2021529805A (ja
JP7621242B2 (ja
JP2021529805A5 (https=
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/040257 external-priority patent/WO2020010058A1/en
Publication of JP2021529805A publication Critical patent/JP2021529805A/ja
Publication of JPWO2020010058A5 publication Critical patent/JPWO2020010058A5/ja
Publication of JP2021529805A5 publication Critical patent/JP2021529805A5/ja
Priority to JP2024131926A priority Critical patent/JP2024150784A/ja
Application granted granted Critical
Publication of JP7621242B2 publication Critical patent/JP7621242B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021500178A 2018-07-06 2019-07-02 イボシデニブ形態および医薬組成物 Active JP7621242B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024131926A JP2024150784A (ja) 2018-07-06 2024-08-08 イボシデニブ形態および医薬組成物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862694596P 2018-07-06 2018-07-06
US62/694,596 2018-07-06
PCT/US2019/040257 WO2020010058A1 (en) 2018-07-06 2019-07-02 Ivosidenib forms and pharmaceutical compositions

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024131926A Division JP2024150784A (ja) 2018-07-06 2024-08-08 イボシデニブ形態および医薬組成物

Publications (4)

Publication Number Publication Date
JP2021529805A JP2021529805A (ja) 2021-11-04
JPWO2020010058A5 true JPWO2020010058A5 (https=) 2022-07-12
JP2021529805A5 JP2021529805A5 (https=) 2022-07-12
JP7621242B2 JP7621242B2 (ja) 2025-01-24

Family

ID=69059942

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021500178A Active JP7621242B2 (ja) 2018-07-06 2019-07-02 イボシデニブ形態および医薬組成物
JP2024131926A Withdrawn JP2024150784A (ja) 2018-07-06 2024-08-08 イボシデニブ形態および医薬組成物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024131926A Withdrawn JP2024150784A (ja) 2018-07-06 2024-08-08 イボシデニブ形態および医薬組成物

Country Status (18)

Country Link
US (1) US12264148B2 (https=)
EP (2) EP3817744A4 (https=)
JP (2) JP7621242B2 (https=)
KR (2) KR102919157B1 (https=)
CN (1) CN112367995A (https=)
AU (2) AU2019299352B2 (https=)
BR (1) BR112021000156A2 (https=)
CA (1) CA3103498A1 (https=)
EA (1) EA202190217A1 (https=)
IL (2) IL315423B1 (https=)
MA (1) MA53099A (https=)
MX (2) MX2021000068A (https=)
PH (1) PH12021550017A1 (https=)
SG (1) SG11202012763TA (https=)
TW (2) TWI902665B (https=)
UA (1) UA129800C2 (https=)
WO (1) WO2020010058A1 (https=)
ZA (1) ZA202008034B (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT4010331T (pt) 2019-08-08 2024-01-08 Servier Lab Um método de preparação do ivosidenib e de um seu intermediário
GB201912411D0 (en) * 2019-08-29 2019-10-16 Johnson Matthey Plc Crystalline forms of ivosidenib
AR133410A1 (es) 2023-08-01 2025-09-24 Servier Lab Cocristal de un inhibidor de idh1, proceso de preparación del mismo, composiciones farmacéuticas del mismo, y métodos de tratamiento que implican el mismo

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2010223919B2 (en) 2009-03-13 2016-03-31 Les Laboratoires Servier Methods and compositions for cell-proliferation-related disorders
EP3561077B1 (en) 2009-10-21 2022-12-21 Les Laboratoires Servier Methods for cell-proliferation-related disorders
RU2013144975A (ru) * 2011-04-08 2015-05-20 Пфайзер Инк. Кристаллические и некристаллические формы тофацитиниба и фармацевтическая композиция, содержащая тофацитиниб, и усилитель проникновения
US9474779B2 (en) 2012-01-19 2016-10-25 Agios Pharmaceuticals, Inc. Therapeutically active compositions and their methods of use
UY35006A (es) * 2012-09-06 2014-03-31 Bayer Healthcare Llc Composición farmacéutica recubierta que contiene regorafenib
BR122023021436A2 (pt) * 2014-03-14 2023-12-12 Les Laboratoires Servier Formas cristalinas e composição farmacêutica de compostos terapeuticamente ativos
KR20240010105A (ko) * 2014-03-14 2024-01-23 아지오스 파마슈티컬스 아이엔씨. 치료적으로 활성인 화합물의 약제학적 조성물
PT3362066T (pt) 2015-10-15 2021-11-16 Celgene Corp Terapia de combinação para tratar malignidades
ES2912909T3 (es) * 2016-02-26 2022-05-30 Celgene Corp Enasidenib para su uso en el tratamiento de la leucemia mieloide aguda recidivante o refractaria
WO2019104318A1 (en) 2017-11-27 2019-05-31 Teva Pharmaceuticals Usa, Inc. Solid state forms of ivosidenib

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