JP7523440B2 - アモルファス固体分散体 - Google Patents
アモルファス固体分散体 Download PDFInfo
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- JP7523440B2 JP7523440B2 JP2021533470A JP2021533470A JP7523440B2 JP 7523440 B2 JP7523440 B2 JP 7523440B2 JP 2021533470 A JP2021533470 A JP 2021533470A JP 2021533470 A JP2021533470 A JP 2021533470A JP 7523440 B2 JP7523440 B2 JP 7523440B2
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
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- Emergency Medicine (AREA)
- Inorganic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
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| US62/779,930 | 2018-12-14 | ||
| PCT/US2019/066247 WO2020123952A1 (en) | 2018-12-14 | 2019-12-13 | Amorphous solid dispersions |
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| JP2022512239A JP2022512239A (ja) | 2022-02-02 |
| JPWO2020123952A5 JPWO2020123952A5 (https=) | 2022-12-14 |
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| IL (1) | IL283927A (https=) |
| MX (1) | MX2021006886A (https=) |
| WO (1) | WO2020123952A1 (https=) |
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| CN112584837A (zh) * | 2018-08-31 | 2021-03-30 | 细胞内治疗公司 | 新方法 |
| CN115671057A (zh) | 2022-10-19 | 2023-02-03 | 四川迈可隆生物科技有限公司 | 一种卢美哌隆药物组合物、长效微球缓释制剂及其制备方法 |
| CN118566395B (zh) * | 2024-08-02 | 2024-10-25 | 则正(济南)生物科技有限公司 | 测定甲苯磺酸卢美哌隆口崩片中杂质含量的方法、应用和系统 |
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| WO2018071233A1 (en) | 2016-10-12 | 2018-04-19 | Intra-Cellular Therapies, Inc. | Amorphous solid dispersions |
| WO2018189646A1 (en) | 2017-04-10 | 2018-10-18 | Dr. Reddy's Laboratories Limited | AMORPHOUS FORM AND SOLID DISPERSIONS OF LUMATEPERONE p-TOSYLATE |
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| US11655251B2 (en) * | 2017-11-27 | 2023-05-23 | Egis Gyogyszergyar Zrt. | Method for the production of lumateperone and its salts |
| CN112584837A (zh) * | 2018-08-31 | 2021-03-30 | 细胞内治疗公司 | 新方法 |
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- 2021-06-13 IL IL283927A patent/IL283927A/en unknown
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2018071233A1 (en) | 2016-10-12 | 2018-04-19 | Intra-Cellular Therapies, Inc. | Amorphous solid dispersions |
| WO2018189646A1 (en) | 2017-04-10 | 2018-10-18 | Dr. Reddy's Laboratories Limited | AMORPHOUS FORM AND SOLID DISPERSIONS OF LUMATEPERONE p-TOSYLATE |
Also Published As
| Publication number | Publication date |
|---|---|
| EP3893878A1 (en) | 2021-10-20 |
| IL283927A (en) | 2021-07-29 |
| JP2022512239A (ja) | 2022-02-02 |
| AU2019398451B2 (en) | 2024-12-05 |
| MX2021006886A (es) | 2021-09-14 |
| CA3123085A1 (en) | 2020-06-18 |
| EP3893878A4 (en) | 2022-08-17 |
| KR20210103501A (ko) | 2021-08-23 |
| WO2020123952A1 (en) | 2020-06-18 |
| AU2019398451A1 (en) | 2021-07-15 |
| CN113473988A (zh) | 2021-10-01 |
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