JP2022501350A5 - - Google Patents

Info

Publication number
JP2022501350A5
JP2022501350A5 JP2021515104A JP2021515104A JP2022501350A5 JP 2022501350 A5 JP2022501350 A5 JP 2022501350A5 JP 2021515104 A JP2021515104 A JP 2021515104A JP 2021515104 A JP2021515104 A JP 2021515104A JP 2022501350 A5 JP2022501350 A5 JP 2022501350A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
isomer
acceptable salt
compound according
optionally substituted
Prior art date
Application number
JP2021515104A
Other languages
English (en)
Japanese (ja)
Other versions
JP7498702B2 (ja
JP2022501350A (ja
JPWO2020057604A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2019/106687 external-priority patent/WO2020057604A1/zh
Publication of JP2022501350A publication Critical patent/JP2022501350A/ja
Publication of JP2022501350A5 publication Critical patent/JP2022501350A5/ja
Publication of JPWO2020057604A5 publication Critical patent/JPWO2020057604A5/ja
Application granted granted Critical
Publication of JP7498702B2 publication Critical patent/JP7498702B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021515104A 2018-09-19 2019-09-19 Tlr8アゴニスト Active JP7498702B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201811094969.4 2018-09-19
CN201811094969 2018-09-19
PCT/CN2019/106687 WO2020057604A1 (zh) 2018-09-19 2019-09-19 Tlr8激动剂

Publications (4)

Publication Number Publication Date
JP2022501350A JP2022501350A (ja) 2022-01-06
JP2022501350A5 true JP2022501350A5 (https=) 2022-09-21
JPWO2020057604A5 JPWO2020057604A5 (https=) 2022-09-21
JP7498702B2 JP7498702B2 (ja) 2024-06-12

Family

ID=69888288

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021515104A Active JP7498702B2 (ja) 2018-09-19 2019-09-19 Tlr8アゴニスト

Country Status (11)

Country Link
US (1) US12054482B2 (https=)
EP (1) EP3854794B1 (https=)
JP (1) JP7498702B2 (https=)
KR (1) KR102856089B1 (https=)
CN (2) CN112805283B (https=)
AU (1) AU2019344868B2 (https=)
CA (1) CA3112953A1 (https=)
ES (1) ES2999323T3 (https=)
PH (1) PH12021550601A1 (https=)
SG (1) SG11202102641RA (https=)
WO (1) WO2020057604A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG11202102641RA (en) 2018-09-19 2021-04-29 Chia Tai Tianqing Pharmaceutical Group Co Ltd Tlr8 agonist
EP4122931B1 (en) * 2020-03-18 2025-07-02 Chia Tai Tianqing Pharmaceutical Group Co., Ltd. Crystalline form of tlr8 agonist
CN116472047B (zh) * 2021-11-05 2025-06-17 中国医药研究开发中心有限公司 芳胺类衍生物及其制备方法和医药用途

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0503506D0 (en) 2005-02-21 2005-03-30 4 Aza Bioscience Nv Substituted pyrido(2,3-d) pyrimidine derivatives and pharmaceutical compositions useful as medicines for the treatment of autoimmune disorders
PT2268618E (pt) 2008-03-03 2015-10-12 Novartis Ag Compostos e composições moduladores da actividade tlr
SG194852A1 (en) 2011-05-18 2013-12-30 Janssen R & D Ireland Quinazoline derivatives for the treatment of viral infections and further diseases
WO2013022766A1 (en) 2011-08-05 2013-02-14 Flynn Gary A Preparation and methods of use for ortho-aryl 5- membered heteroaryl-carboxamide containing multi-targeted kinase inhibitors
EP2925729B1 (en) 2012-11-16 2017-10-18 Janssen Sciences Ireland UC Heterocyclic substituted 2-amino-quinazoline derivatives for the treatment of viral infections
WO2016141092A1 (en) 2015-03-04 2016-09-09 Gilead Sciences, Inc. Toll-like receptor modulating 4,6-diamino-pyrido[3,2-d]pyrimidine compounds
EP3507288B1 (en) 2016-09-02 2020-08-26 Gilead Sciences, Inc. 4,6-diamino-pyrido[3,2-d]pyrimidine derivaties as toll like receptor modulators
CN109923106B (zh) 2016-09-02 2022-09-13 吉利德科学公司 toll样受体调节剂化合物
SG11202102641RA (en) 2018-09-19 2021-04-29 Chia Tai Tianqing Pharmaceutical Group Co Ltd Tlr8 agonist

Similar Documents

Publication Publication Date Title
JP2012092103A5 (https=)
JP2022501350A5 (https=)
JP2021513534A5 (https=)
CN113365998A (zh) 用于parp抑制剂的吲哚并七元酰肟类似物
JP2018533593A5 (https=)
CN113784970A (zh) Erk抑制剂及其应用
JP2016513130A5 (https=)
JP2020507589A5 (https=)
JP2019527234A5 (https=)
JP2019524883A5 (https=)
CN114072396A (zh) 作为dna-pk抑制剂的喹啉和噌啉衍生物
JP2019510082A5 (https=)
JP2019527233A5 (https=)
JP2013545785A5 (https=)
JP2014500861A5 (https=)
JP2005523922A5 (https=)
JP2014511892A5 (https=)
JP2012506389A5 (https=)
JP2015511958A5 (https=)
JP2013032389A5 (https=)
JP2016510323A5 (https=)
JP2017523169A5 (https=)
JP2015517555A5 (https=)
JP2009527462A5 (https=)
RU2016151420A (ru) Новое терапевтическое применение производных бензилиденгуанидина для лечения протеинопатий