JP2020516671A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2020516671A5 JP2020516671A5 JP2019556238A JP2019556238A JP2020516671A5 JP 2020516671 A5 JP2020516671 A5 JP 2020516671A5 JP 2019556238 A JP2019556238 A JP 2019556238A JP 2019556238 A JP2019556238 A JP 2019556238A JP 2020516671 A5 JP2020516671 A5 JP 2020516671A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- compound
- acid
- triazole
- sulfanyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2022164773A JP2022191395A (ja) | 2017-04-14 | 2022-10-13 | 選択的hdac6阻害剤 |
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT102017000041723A IT201700041723A1 (it) | 2017-04-14 | 2017-04-14 | Nuovi inibitori selettivi di HDAC6 |
IT102017000041723 | 2017-04-14 | ||
PCT/EP2018/059468 WO2018189340A1 (en) | 2017-04-14 | 2018-04-12 | Selective hdac6 inhibitors |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2022164773A Division JP2022191395A (ja) | 2017-04-14 | 2022-10-13 | 選択的hdac6阻害剤 |
Publications (3)
Publication Number | Publication Date |
---|---|
JP2020516671A JP2020516671A (ja) | 2020-06-11 |
JP2020516671A5 true JP2020516671A5 (US07981874-20110719-C00313.png) | 2020-12-17 |
JP7241025B2 JP7241025B2 (ja) | 2023-03-16 |
Family
ID=59700099
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2019556238A Active JP7241025B2 (ja) | 2017-04-14 | 2018-04-12 | 選択的hdac6阻害剤 |
JP2022164773A Withdrawn JP2022191395A (ja) | 2017-04-14 | 2022-10-13 | 選択的hdac6阻害剤 |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2022164773A Withdrawn JP2022191395A (ja) | 2017-04-14 | 2022-10-13 | 選択的hdac6阻害剤 |
Country Status (30)
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US10357493B2 (en) | 2017-03-10 | 2019-07-23 | Selenity Therapeutics (Bermuda), Ltd. | Metalloenzyme inhibitor compounds |
CN109942564A (zh) * | 2019-04-16 | 2019-06-28 | 四川大学华西医院 | 一种组蛋白去乙酰化酶抑制剂及其制备方法和用途 |
US20220251043A1 (en) * | 2019-07-23 | 2022-08-11 | Taipei Medical University | Histone deacetylase 6 inhibitors and method for treating neuropathic pain |
CA3189738A1 (en) * | 2020-08-07 | 2022-02-10 | Italfarmaco S.P.A. | Novel oxadiazole-based selective hdac6 inhibitors |
CN112250638B (zh) * | 2020-11-13 | 2022-05-03 | 郑州大学 | 一种1,3-二芳基-1,2,4-三氮唑类化合物及其制备方法和应用 |
IT202100009926A1 (it) | 2021-04-20 | 2022-10-20 | Italfarmaco Spa | Una combinazione comprendente un inibitore di hdac6 specifico e almeno un inibitore del checkpoint ctla4 |
TW202340480A (zh) | 2021-11-23 | 2023-10-16 | 義大利商義大利藥品股份有限公司 | 檢測rna生物標記之方法 |
WO2023219456A1 (ko) * | 2022-05-12 | 2023-11-16 | 숙명여자대학교 산학협력단 | 퀴놀린 계열 히스톤디아세틸화 효소 저해활성물질, 이의 제조방법 및 이를 유효성분으로 포함하는 약학적 조성물 |
KR20240043709A (ko) * | 2022-09-27 | 2024-04-03 | 사회복지법인 삼성생명공익재단 | 히스톤 탈아세틸화효소 억제제를 포함하는 암 치료용 조성물, 및 암 면역치료용 항암 보조제 |
CN115611823A (zh) * | 2022-10-27 | 2023-01-17 | 新天地医药技术研究院(郑州)有限公司 | 一种1,2,4-三氮唑-苯基异羟肟酸类化合物、制备方法和应用 |
CN115737549A (zh) * | 2022-11-24 | 2023-03-07 | 北京鑫开元医药科技有限公司 | 一种具有hdac抑制活性的注射液及其制备方法和用途 |
WO2024148259A1 (en) * | 2023-01-06 | 2024-07-11 | Sparrow Pharmaceuticals, Inc. | Methods and compositions for treating hsd-1-mediated disorders |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1470121B1 (en) | 2002-01-23 | 2012-07-11 | Bayer HealthCare LLC | Pyrimidine derivatives as rho-kinase inhibitors |
EP1765814A1 (en) | 2004-07-02 | 2007-03-28 | Novo Nordisk A/S | Condensed thiophene derivatives and their use as cyclic glp-1 agonists |
GB0607899D0 (en) | 2006-04-03 | 2006-05-31 | Glaxo Group Ltd | Process for preparing heterocyclic derivatives |
EP2170882A1 (en) | 2007-06-26 | 2010-04-07 | Gilead Colorado, Inc. | Imidazopyridinyl thiazolyl histone deacetylase inhibitors |
EP2445340B1 (en) | 2009-06-22 | 2016-05-18 | Millennium Pharmaceuticals, Inc. | Substituted hydroxamic acids and uses thereof |
CN102548975A (zh) * | 2009-07-07 | 2012-07-04 | 安瑟生物科技私人有限公司 | 组蛋白去乙酰化酶抑制剂 |
JP5518397B2 (ja) | 2009-08-12 | 2014-06-11 | 富士フイルム株式会社 | 水性インク組成物、複合粒子の製造方法、インクセット、及び、画像形成方法 |
WO2011106650A2 (en) | 2010-02-27 | 2011-09-01 | University Of Pittsburgh - Of The Commonwealth System Of Higher Education | Novel p53-mdm2/p53-mdm4 antagonists to treat proliferative disease |
KR20130115300A (ko) * | 2010-11-16 | 2013-10-21 | 에이스틸론 파마수티컬스 인코포레이티드 | 단백질 탈아세틸화 효소 억제제로서 피리미딘 하이드록시 아미드 화합물 및 그의 사용방법 |
USRE47009E1 (en) * | 2011-02-01 | 2018-08-28 | The Children's Hospital Of Philadelphia | HDAC inhibitors and therapeutic methods using the same |
EP2487159A1 (en) | 2011-02-11 | 2012-08-15 | MSD Oss B.V. | RorgammaT inhibitors |
US20150197497A1 (en) * | 2011-06-24 | 2015-07-16 | Dana-Farber Cancer Institute, Inc. | Selective inhibitors of histone deacetylase isoform 6 and methods thereof |
WO2015087151A1 (en) | 2013-12-12 | 2015-06-18 | Chong Kun Dang Pharmaceutical Corp. | Novel azaindole derivatives as selective histone deacetylase (hdac) inhibitors and pharmaceutical compositions comprising the same |
KR101685639B1 (ko) | 2014-01-03 | 2016-12-12 | 주식회사 종근당 | 신규한 인돌 유도체 화합물 및 이를 포함하는 약제학적 조성물 |
BR112016026518A2 (pt) * | 2014-05-14 | 2017-08-15 | Univ Colorado Regents | Ácidos hidroxâmicos heterocíclicos como inibidores da proteína desacetilase e inibidores duais de proteína desacetilase-proteína cinase e métodos de uso dos mesmos |
CN106794175B (zh) * | 2014-06-12 | 2020-06-09 | 西达-赛奈医疗中心 | 用于治疗癌症的组合物 |
-
2017
- 2017-04-14 IT IT102017000041723A patent/IT201700041723A1/it unknown
-
2018
- 2018-04-09 TW TW107112124A patent/TWI813564B/zh active
- 2018-04-12 BR BR112019021078-4A patent/BR112019021078A2/pt active Search and Examination
- 2018-04-12 PL PL18716299.5T patent/PL3562810T3/pl unknown
- 2018-04-12 FI FIEP18716299.5T patent/FI3562810T3/fi active
- 2018-04-12 ES ES18716299T patent/ES2951476T3/es active Active
- 2018-04-12 LT LTEPPCT/EP2018/059468T patent/LT3562810T/lt unknown
- 2018-04-12 NZ NZ756603A patent/NZ756603A/en unknown
- 2018-04-12 AU AU2018252172A patent/AU2018252172B9/en active Active
- 2018-04-12 EP EP18716299.5A patent/EP3562810B1/en active Active
- 2018-04-12 RS RS20230576A patent/RS64376B1/sr unknown
- 2018-04-12 CA CA3056381A patent/CA3056381A1/en active Pending
- 2018-04-12 RU RU2019132212A patent/RU2764718C2/ru active
- 2018-04-12 JP JP2019556238A patent/JP7241025B2/ja active Active
- 2018-04-12 DK DK18716299.5T patent/DK3562810T3/da active
- 2018-04-12 KR KR1020197033482A patent/KR102525375B1/ko active IP Right Grant
- 2018-04-12 US US16/491,827 patent/US11351178B2/en active Active
- 2018-04-12 HR HRP20230789TT patent/HRP20230789T8/hr unknown
- 2018-04-12 PT PT187162995T patent/PT3562810T/pt unknown
- 2018-04-12 WO PCT/EP2018/059468 patent/WO2018189340A1/en active Search and Examination
- 2018-04-12 HU HUE18716299A patent/HUE063079T2/hu unknown
- 2018-04-12 CN CN201880024895.9A patent/CN110546140B/zh active Active
- 2018-04-12 MX MX2019011876A patent/MX2019011876A/es unknown
- 2018-04-12 PE PE2019001995A patent/PE20200446A1/es unknown
- 2018-04-12 SI SI201830949T patent/SI3562810T1/sl unknown
- 2018-04-13 AR ARP180100940A patent/AR111466A1/es unknown
-
2019
- 2019-08-27 IL IL268955A patent/IL268955B/en unknown
- 2019-10-08 CL CL2019002869A patent/CL2019002869A1/es unknown
- 2019-10-28 CO CONC2019/0011993A patent/CO2019011993A2/es unknown
-
2022
- 2022-10-13 JP JP2022164773A patent/JP2022191395A/ja not_active Withdrawn
-
2023
- 2023-07-26 CY CY20231100364T patent/CY1126110T1/el unknown