ITPD910163A1 - Uso di esteri della colina con polisaccaridi acidi come agenti antiulcera e gastroprotettivi - Google Patents

Uso di esteri della colina con polisaccaridi acidi come agenti antiulcera e gastroprotettivi

Info

Publication number
ITPD910163A1
ITPD910163A1 IT000163A ITPD910163A ITPD910163A1 IT PD910163 A1 ITPD910163 A1 IT PD910163A1 IT 000163 A IT000163 A IT 000163A IT PD910163 A ITPD910163 A IT PD910163A IT PD910163 A1 ITPD910163 A1 IT PD910163A1
Authority
IT
Italy
Prior art keywords
ulcer
china
esters
acid polysaccharides
gastroprotective agents
Prior art date
Application number
IT000163A
Other languages
English (en)
Inventor
Lanfranco Callegaro
Aurelio Romeo
Gino Toffano
Original Assignee
Fidia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fidia Spa filed Critical Fidia Spa
Priority to ITPD910163A priority Critical patent/IT1263755B/it
Publication of ITPD910163A0 publication Critical patent/ITPD910163A0/it
Priority to EP92919162A priority patent/EP0605478A1/en
Priority to AU25481/92A priority patent/AU2548192A/en
Priority to PCT/EP1992/002133 priority patent/WO1993005792A1/en
Priority to US07/945,495 priority patent/US5300493A/en
Publication of ITPD910163A1 publication Critical patent/ITPD910163A1/it
Application granted granted Critical
Publication of IT1263755B publication Critical patent/IT1263755B/it

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/045Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A61K31/726Glycosaminoglycans, i.e. mucopolysaccharides
    • A61K31/728Hyaluronic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A61K31/716Glucans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A61K31/716Glucans
    • A61K31/717Celluloses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A61K31/734Alginic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ITPD910163A 1991-09-16 1991-09-16 Uso di esteri della colina con polisaccaridi acidi come agenti antiulcera e gastroprotettivi IT1263755B (it)

Priority Applications (5)

Application Number Priority Date Filing Date Title
ITPD910163A IT1263755B (it) 1991-09-16 1991-09-16 Uso di esteri della colina con polisaccaridi acidi come agenti antiulcera e gastroprotettivi
EP92919162A EP0605478A1 (en) 1991-09-16 1992-09-14 New use of acidic polysaccharide esters as anti-ulcer agents
AU25481/92A AU2548192A (en) 1991-09-16 1992-09-14 New use of acidic polysaccharide esters as anti-ulcer agents
PCT/EP1992/002133 WO1993005792A1 (en) 1991-09-16 1992-09-14 New use of acidic polysaccharide esters as anti-ulcer agents
US07/945,495 US5300493A (en) 1991-09-16 1992-09-16 Ulcer treatment using choline esters of polysaccharides

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITPD910163A IT1263755B (it) 1991-09-16 1991-09-16 Uso di esteri della colina con polisaccaridi acidi come agenti antiulcera e gastroprotettivi

Publications (3)

Publication Number Publication Date
ITPD910163A0 ITPD910163A0 (it) 1991-09-16
ITPD910163A1 true ITPD910163A1 (it) 1993-03-16
IT1263755B IT1263755B (it) 1996-08-29

Family

ID=11389683

Family Applications (1)

Application Number Title Priority Date Filing Date
ITPD910163A IT1263755B (it) 1991-09-16 1991-09-16 Uso di esteri della colina con polisaccaridi acidi come agenti antiulcera e gastroprotettivi

Country Status (5)

Country Link
US (1) US5300493A (it)
EP (1) EP0605478A1 (it)
AU (1) AU2548192A (it)
IT (1) IT1263755B (it)
WO (1) WO1993005792A1 (it)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR950701312A (ko) * 1992-05-12 1995-03-23 이베 사치아키 신규 4급 암모늄염 및 약제로서 그의 사용
US5952314A (en) 1994-04-01 1999-09-14 Demichele; Stephen Joseph Nutritional product for a person having ulcerative colitis
US5780451A (en) * 1994-04-01 1998-07-14 Abbott Laboratories Nutritional product for a person having ulcerative colitis
ITPD980168A1 (it) * 1998-07-06 2000-01-06 Fidia Advanced Biopolymers Srl Composizioni biocompatibili e biodegradabili comprendenti acido ialuronico e suoi derivati per il trattamento delle ulcere dell'appara
WO2000005269A1 (en) * 1998-07-21 2000-02-03 Alpenstock Holdings Limited Polymer complexes of glucuronoglucanes
GB0012094D0 (en) * 2000-05-19 2000-07-12 Reckitt & Colmann Prod Ltd Pharmaceutical compositions
DE10033197C1 (de) * 2000-07-07 2002-01-10 Fraunhofer Ges Forschung Verfahren zur Herstellung von hochsubstituierter Carboxymethylstärke
EP4311552A1 (en) * 2022-07-28 2024-01-31 Bioiberica, S.A.U. Gastrointestinal protectant composition

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2902479A (en) * 1957-03-01 1959-09-01 Kelco Co Carboxymethyl alginate product and methods of preparing carboxymethyl alginate
US3364111A (en) * 1964-11-20 1968-01-16 Meito Sangyo Kk Carboxymethylated dextran for peptic ulcers
US4287174A (en) * 1978-03-31 1981-09-01 The Proctor & Gamble Company Anti-ulcer composition
DE3374914D1 (en) * 1982-04-12 1988-01-28 Univ Texas Methods and compositions for treating gastro-intestinal ulcer diesease
IT1172580B (it) * 1983-01-05 1987-06-18 F I R M A Fabbrica Italiana Ri Composizione farmaceutica avente proprieta' gastro-protettive ed antiulcera, a base di carbossimetilcellulosa
DE3482812D1 (de) * 1983-10-11 1990-08-30 Fidia Spa Fraktionen von hyaluronsaeure mit pharmazeutischer aktivitaet, verfahren zu deren herstellung und sie enthaltende pharmazeutische zusammensetzungen.
US4729989A (en) * 1985-06-28 1988-03-08 Merck & Co., Inc. Enhancement of absorption of drugs from gastrointestinal tract using choline ester salts
US4851521A (en) * 1985-07-08 1989-07-25 Fidia, S.P.A. Esters of hyaluronic acid
IT1203814B (it) * 1986-06-30 1989-02-23 Fidia Farmaceutici Esteri dell'acido alginico
IT1219942B (it) * 1988-05-13 1990-05-24 Fidia Farmaceutici Esteri polisaccaridici

Also Published As

Publication number Publication date
EP0605478A1 (en) 1994-07-13
WO1993005792A1 (en) 1993-04-01
IT1263755B (it) 1996-08-29
AU2548192A (en) 1993-04-27
ITPD910163A0 (it) 1991-09-16
US5300493A (en) 1994-04-05

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Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19950925