IT1164097B - "1,4-DI HYDROPYRIDINE THEIR PREPARATION AND THEIR APPLICATION AS MEDICATIONS" - Google Patents
"1,4-DI HYDROPYRIDINE THEIR PREPARATION AND THEIR APPLICATION AS MEDICATIONS"Info
- Publication number
- IT1164097B IT1164097B IT51095/79A IT5109579A IT1164097B IT 1164097 B IT1164097 B IT 1164097B IT 51095/79 A IT51095/79 A IT 51095/79A IT 5109579 A IT5109579 A IT 5109579A IT 1164097 B IT1164097 B IT 1164097B
- Authority
- IT
- Italy
- Prior art keywords
- hydropyridine
- medications
- preparation
- application
- Prior art date
Links
- JUJWROOIHBZHMG-UHFFFAOYSA-N Pyridine Chemical compound C1=CC=NC=C1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 title 1
- 229940079593 drug Drugs 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH1283578A CH639659A5 (en) | 1978-12-18 | 1978-12-18 | NEW 1,4-DIHYDROPYRIDINE DERIVATIVES, THEIR PRODUCTION AND USE. |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IT7951095A0 IT7951095A0 (en) | 1979-12-14 |
| IT1164097B true IT1164097B (en) | 1987-04-08 |
Family
ID=4386824
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT51095/79A IT1164097B (en) | 1978-12-18 | 1979-12-14 | "1,4-DI HYDROPYRIDINE THEIR PREPARATION AND THEIR APPLICATION AS MEDICATIONS" |
Country Status (18)
| Country | Link |
|---|---|
| JP (1) | JPS5583783A (en) |
| AU (1) | AU536055B2 (en) |
| BE (1) | BE880591A (en) |
| CH (1) | CH639659A5 (en) |
| CY (1) | CY1321A (en) |
| DE (1) | DE2949491A1 (en) |
| FR (1) | FR2444681A1 (en) |
| GB (2) | GB2103203B (en) |
| HK (1) | HK16086A (en) |
| IE (1) | IE49496B1 (en) |
| IT (1) | IT1164097B (en) |
| KE (1) | KE3593A (en) |
| MY (1) | MY8500130A (en) |
| NL (2) | NL193066C (en) |
| NZ (1) | NZ192422A (en) |
| SE (1) | SE445219B (en) |
| SG (1) | SG97585G (en) |
| ZA (1) | ZA796842B (en) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3022030A1 (en) * | 1980-06-12 | 1981-12-17 | Bayer Ag, 5090 Leverkusen | 4-THIAZOLE or 4-IMIDAZOLE-SUBSTITUTED, 1,4-DIHYDROPYRIDINE, METHOD FOR THE PRODUCTION THEREOF AND THE MEDICINAL PRODUCTS CONTAINING THEM |
| CH655658B (en) * | 1980-09-18 | 1986-05-15 | ||
| EP0080220B1 (en) * | 1981-11-17 | 1986-02-19 | FISONS plc | Dihydropyridines, methods for their production and their formulation and use as pharmaceuticals |
| ZA83959B (en) * | 1982-03-10 | 1984-09-26 | Sandoz Ltd | 1,4-dihydropyridine derivatives,their preparation and pharmaceutical compositions containing them |
| US4414213A (en) * | 1982-03-22 | 1983-11-08 | Mead Johnson & Company | Dihydropyridyl cyclic imidate esters and their pharmaceutical use |
| IL68975A (en) * | 1982-06-15 | 1987-01-30 | Sandoz Ag | 4-(2,1,3-benzoxadiazol-4-yl)-1,4-dihydropyridine-3,5-dicarboxylic acid ester derivatives in optically active form,their preparation and pharmaceutical compositions containing them |
| FR2528431B1 (en) * | 1982-06-15 | 1986-01-10 | Sandoz Sa | NOVEL 1,4-DIHYDROPYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICAMENTS |
| JPS5978186A (en) * | 1982-10-27 | 1984-05-04 | Yoshitomi Pharmaceut Ind Ltd | 1,4-dihydropyridine-3,5-dicarboxylic acid ester derivative |
| US4794111A (en) * | 1984-05-23 | 1988-12-27 | Bayer Aktiengesellschaft | Dihydropyridine preparations containing β-blockers |
| HU198844B (en) * | 1984-06-14 | 1989-12-28 | Sandoz Ag | Process for producing new galenic pharmaceutical composition ensuring retarded release of active ingredient |
| US5260321A (en) * | 1984-11-12 | 1993-11-09 | Sandoz Ltd. | Use of 1,4-dihydropyridine derivatives and combinations thereof with calcitonins |
| HU197201B (en) * | 1985-10-01 | 1989-03-28 | Sandoz Ag | Process for producing oral pharmaceutical compositions of controlled solubility of the active components |
| DE3542794A1 (en) * | 1985-12-04 | 1987-06-11 | Bayer Ag | ANTI-HYPERTENSIVE COMBINATION PREPARATION |
| GB8626217D0 (en) * | 1986-11-03 | 1986-12-03 | Sandoz Ltd | Pharmaceutical compositions |
| US4816263A (en) * | 1987-10-02 | 1989-03-28 | Alza Corporation | Dosage form for treating cardiovascular diseases comprising isradipine |
| KR940003492B1 (en) * | 1988-10-27 | 1994-04-23 | 주식회사 유한양행 | 1,4-dihydropyridine derivative and preparation method thereof |
| DE4222770A1 (en) * | 1992-07-10 | 1994-01-13 | Bayer Ag | Light-activated 1- (2-nitrobenzyl) -substituted 1,4-dihydropyridines |
| EP2316468A1 (en) | 2002-02-22 | 2011-05-04 | Shire LLC | Delivery system and methods for protecting and administering dextroamphetamine |
| AU2003269482A1 (en) * | 2003-09-10 | 2005-03-29 | Shasun Chemicals And Drugs Limited | Process for the manufacture of 2,1,3-benzoxadiazole-4-carboxaldehyde |
| CN103613584B (en) * | 2013-11-27 | 2016-04-27 | 沈阳药科大学 | The method of a kind of Isrodipine synthetic product aftertreatment |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1670824C3 (en) * | 1967-03-20 | 1978-08-03 | Bayer Ag, 5090 Leverkusen | 1,4-Dihydropyridine-33-dicarboxylic acid alkyl ester |
| FR2320750A1 (en) * | 1975-08-12 | 1977-03-11 | Hexachimie | 1,4-DIHYDRO PYRIDINES AND THEIR THERAPEUTIC APPLICATION |
| DE2616991A1 (en) * | 1976-04-17 | 1977-10-27 | Bayer Ag | Thio-substd. dihydro-pyridine derivs. - coronary vasodilators and antihypertensives prepd. e.g. by reacting dicarbonyl cpds. with amines and thio-substd. ketones |
| JPS5373327A (en) * | 1976-12-13 | 1978-06-29 | Matsushita Electric Ind Co Ltd | Power source system |
| DK149855C (en) * | 1977-06-20 | 1987-04-21 | Sandoz Ag | METHOD OF ANALOGY FOR THE PREPARATION OF 1,4-DIHYDROPYRIDINE DERIVATIVES |
-
1978
- 1978-12-18 CH CH1283578A patent/CH639659A5/en not_active IP Right Cessation
-
1979
- 1979-12-08 DE DE19792949491 patent/DE2949491A1/en active Granted
- 1979-12-11 SE SE7910188A patent/SE445219B/en not_active IP Right Cessation
- 1979-12-13 BE BE1/9643A patent/BE880591A/en not_active IP Right Cessation
- 1979-12-14 GB GB08215988A patent/GB2103203B/en not_active Expired
- 1979-12-14 IT IT51095/79A patent/IT1164097B/en active Protection Beyond IP Right Term
- 1979-12-14 GB GB7943113A patent/GB2037766B/en not_active Expired
- 1979-12-14 CY CY1321A patent/CY1321A/en unknown
- 1979-12-14 NL NL7909024A patent/NL193066C/en not_active IP Right Cessation
- 1979-12-17 IE IE2445/79A patent/IE49496B1/en not_active IP Right Cessation
- 1979-12-17 JP JP16396579A patent/JPS5583783A/en active Granted
- 1979-12-17 NZ NZ192422A patent/NZ192422A/en unknown
- 1979-12-17 AU AU53896/79A patent/AU536055B2/en not_active Expired
- 1979-12-17 FR FR7930829A patent/FR2444681A1/en active Granted
- 1979-12-18 ZA ZA00796842A patent/ZA796842B/en unknown
-
1985
- 1985-12-20 SG SG975/85A patent/SG97585G/en unknown
- 1985-12-30 MY MY130/85A patent/MY8500130A/en unknown
-
1986
- 1986-01-08 KE KE3593A patent/KE3593A/en unknown
- 1986-03-06 HK HK160/86A patent/HK16086A/en not_active IP Right Cessation
-
1999
- 1999-05-11 NL NL990014C patent/NL990014I1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NL193066B (en) | 1998-05-06 |
| GB2037766B (en) | 1983-02-16 |
| GB2037766A (en) | 1980-07-16 |
| GB2103203A (en) | 1983-02-16 |
| IE49496B1 (en) | 1985-10-16 |
| DE2949491C2 (en) | 1988-10-27 |
| JPH0369910B2 (en) | 1991-11-05 |
| KE3593A (en) | 1986-02-07 |
| IT7951095A0 (en) | 1979-12-14 |
| NZ192422A (en) | 1982-09-14 |
| JPS5583783A (en) | 1980-06-24 |
| BE880591A (en) | 1980-06-13 |
| HK16086A (en) | 1986-03-14 |
| MY8500130A (en) | 1985-12-31 |
| FR2444681B1 (en) | 1982-10-29 |
| NL7909024A (en) | 1980-06-20 |
| FR2444681A1 (en) | 1980-07-18 |
| SG97585G (en) | 1986-07-18 |
| DE2949491A1 (en) | 1980-06-26 |
| AU5389679A (en) | 1980-06-26 |
| GB2103203B (en) | 1983-06-08 |
| CH639659A5 (en) | 1983-11-30 |
| CY1321A (en) | 1986-06-27 |
| SE7910188L (en) | 1980-06-19 |
| IE792445L (en) | 1980-06-18 |
| NL193066C (en) | 1998-09-08 |
| AU536055B2 (en) | 1984-04-19 |
| SE445219B (en) | 1986-06-09 |
| ZA796842B (en) | 1981-07-29 |
| NL990014I1 (en) | 1999-07-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ITCP | Complementary protection certificate |
Free format text: CCP 138 |
|
| MEDD | Supplementary protection certificate for pharmaceutical products: granted |
Free format text: CCP 138, 19920423; SANDOZ A.G. |
|
| TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19971205 |