IN2013MU00665A - - Google Patents
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- Publication number
- IN2013MU00665A IN2013MU00665A IN665MU2013A IN2013MU00665A IN 2013MU00665 A IN2013MU00665 A IN 2013MU00665A IN 665MU2013 A IN665MU2013 A IN 665MU2013A IN 2013MU00665 A IN2013MU00665 A IN 2013MU00665A
- Authority
- IN
- India
- Prior art keywords
- present
- novel compounds
- provides
- oxalate
- raloxifene
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/56—Radicals substituted by oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Abstract
The present invention provides raloxifene oxalate, including derivatives thereof. In particular, the present invention provides solvates and/or hydrates of raloxifene oxalate, and polymorphs thereof. The present invention also provides processes for preparing the novel compounds, pharmaceutical compositions including the novel compounds and medical uses of the novel compounds.
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN665MU2013 IN2013MU00665A (en) | 2013-03-05 | 2014-03-05 | |
ZA2014/01636A ZA201401636B (en) | 2013-03-05 | 2014-03-05 | Oxalic acid addition salts and/or solvates of a selective estrogen receptor modulator |
PCT/GB2014/000081 WO2014135834A1 (en) | 2013-03-05 | 2014-03-05 | Oxalic acid addition salts and/or solvates of a selective estrogen receptor modulator |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN665MU2013 IN2013MU00665A (en) | 2013-03-05 | 2014-03-05 |
Publications (1)
Publication Number | Publication Date |
---|---|
IN2013MU00665A true IN2013MU00665A (en) | 2015-07-03 |
Family
ID=50382470
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IN665MU2013 IN2013MU00665A (en) | 2013-03-05 | 2014-03-05 |
Country Status (3)
Country | Link |
---|---|
IN (1) | IN2013MU00665A (en) |
WO (1) | WO2014135834A1 (en) |
ZA (1) | ZA201401636B (en) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2988620A1 (en) | 2015-06-16 | 2016-12-22 | Jiangsu Hengrui Medicine Co., Ltd. | Piperidine derivative and preparation method and pharmaceutical use thereof |
KR20180095564A (en) | 2015-12-22 | 2018-08-27 | 지앙수 헨그루이 메디슨 컴퍼니 리미티드 | Benzopiperidine Derivatives, Processes for Their Preparation and Their Medical Uses |
CN116731064A (en) | 2020-01-10 | 2023-09-12 | 江苏恒瑞医药股份有限公司 | Tricyclic tetrahydroisoquinoline derivative, preparation method and application thereof in medicine |
WO2023280309A1 (en) | 2021-07-09 | 2023-01-12 | 江苏恒瑞医药股份有限公司 | Salt types of tricyclic tetrahydro isoquinoline derivative |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4133814A (en) | 1975-10-28 | 1979-01-09 | Eli Lilly And Company | 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents |
US4380635A (en) | 1981-04-03 | 1983-04-19 | Eli Lilly And Company | Synthesis of acylated benzothiophenes |
US4358593A (en) | 1981-04-03 | 1982-11-09 | Eli Lilly And Company | Process for preparing 3-(4-aminoethoxybenzoyl)benzo[b]thiophenes |
TW366342B (en) | 1992-07-28 | 1999-08-11 | Lilly Co Eli | The use of 2-phenyl-3-aroylbenzothiophenes in inhibiting bone loss |
US5629425A (en) * | 1994-09-19 | 1997-05-13 | Eli Lilly And Company | Haloalkyl hemisolvates of 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-piperidinoethoxy)-benzoyl]benzo[b]thiophene |
CO4410191A1 (en) | 1994-09-19 | 1997-01-09 | Lilly Co Eli | SYNTHESIS OF 3- [4- (2-AMINOETOXI) BENZOIL] -2-ARYL-6- HYDROXYBENZO [b] THIOPHENES |
WO1998048792A1 (en) | 1997-04-30 | 1998-11-05 | Eli Lilly And Company | A REGIOSELECTIVE ALKYLATION PROCESS FOR PREPARING SUBSTITUTED BENZO[b]THIOPHENES |
US7964734B2 (en) | 2002-09-30 | 2011-06-21 | A/S Gea Farmaceutisk Fabrik | Raloxifene acid addition salts and/or solvates thereof, improved method for purification of said raloxifene acid addition salts and/or solvates thereof and pharmaceutical compositions comprising these |
PL2032521T3 (en) * | 2006-06-27 | 2010-05-31 | Sandoz Ag | New method for salt preparation |
GB2456096B (en) * | 2006-10-17 | 2011-08-17 | Cipla Ltd | Crystalline form of benzothiophene compound and process for preparation thereof |
WO2011099942A1 (en) | 2010-02-09 | 2011-08-18 | Silverstone Pharma | New addition salts of raloxifene, process for the preparation thereof and use thereof in therapy |
-
2014
- 2014-03-05 IN IN665MU2013 patent/IN2013MU00665A/en unknown
- 2014-03-05 ZA ZA2014/01636A patent/ZA201401636B/en unknown
- 2014-03-05 WO PCT/GB2014/000081 patent/WO2014135834A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
WO2014135834A1 (en) | 2014-09-12 |
WO2014135834A8 (en) | 2014-11-27 |
ZA201401636B (en) | 2014-11-26 |
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