IN2011KN05169A - - Google Patents

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IN2011KN05169A
IN2011KN05169A IN5169KON2011A IN2011KN05169A IN 2011KN05169 A IN2011KN05169 A IN 2011KN05169A IN 5169KON2011 A IN5169KON2011 A IN 5169KON2011A IN 2011KN05169 A IN2011KN05169 A IN 2011KN05169A
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India
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well
human
general formula
veterinary medicine
relates
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Laurence Clary
Sandrine Chambon
Laurent Chantalat
Carine Rosignoli
Olivier Roye
Jean-Claude Pascal
Marlène Schuppli
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Galderma Res & Dev
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Publication of IN2011KN05169A publication Critical patent/IN2011KN05169A/en

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    • C07D241/04—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
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    • C07D295/15—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
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Abstract

The present invention relates to novel benzenesulfonamide compounds having a structure of general formula (I) below: as well as to the method for synthesizing same and to the use thereof in pharmaceutical compositions to be used in human or veterinary medicine, as well as to the use thereof in cosmetic compositions.
IN5169KON2011 2009-06-30 2010-06-28 IN2011KN05169A (en)

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FR0954460A FR2947268B1 (en) 2009-06-30 2009-06-30 NOVEL BENZENE-SULFONAMIDE COMPOUNDS, PROCESS FOR THE SYNTHESIS AND THEIR USE IN MEDICINE AND COSMETICS
PCT/FR2010/051331 WO2011001089A1 (en) 2009-06-30 2010-06-28 Novel benzenesulfonamide compounds, method for synthesizing same, and use thereof in medicine as well as in cosmetics

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RU (2) RU2528826C2 (en)
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FR2947268B1 (en) * 2009-06-30 2011-08-26 Galderma Res & Dev NOVEL BENZENE-SULFONAMIDE COMPOUNDS, PROCESS FOR THE SYNTHESIS AND THEIR USE IN MEDICINE AND COSMETICS
FR2950057B1 (en) * 2009-09-17 2011-08-26 Galderma Res & Dev NOVEL BENZENE CARBOXYLAMIDE COMPOUNDS, PROCESS FOR THEIR SYNTHESIS AND THEIR USE IN MEDICINE AND COSMETICS
US9586832B2 (en) * 2013-03-15 2017-03-07 Dru L. DeLaet Method for destruction of halons
US20140275108A1 (en) * 2013-03-15 2014-09-18 Galderma Research & Development Novel benzenesulfonamide compounds, method for synthesizing same, and use thereof in medicine as well as in cosmetics
CN103224476A (en) * 2013-05-25 2013-07-31 上高县瑞雅精细化工有限公司 New process for preparing 1-[2-(2-hydroxyethoxy)ethyl]piperazine through diethanolamine method
FR3030521B1 (en) * 2014-12-23 2019-07-26 Galderma Research & Development NOVEL HETEROCYCLIC COMPOUNDS AND THEIR USE IN MEDICINE AND COSMETICS
ES2695533T3 (en) 2016-02-01 2019-01-08 Galderma Res & Dev Benzenesulfonamide compounds, method for their synthesis and use in medicine and cosmetics
US12023310B2 (en) * 2022-08-30 2024-07-02 Gongwin Biopharm Co., Ltd Method for treating peripheral nerve sheath tumor

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RU2528826C2 (en) 2014-09-20
SMT201400168B (en) 2015-01-15
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US8633196B2 (en) 2014-01-21
US20120323006A1 (en) 2012-12-20
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AU2010267872B2 (en) 2013-10-10
MX2011013130A (en) 2012-02-13
JP2012531460A (en) 2012-12-10
AU2010267872A1 (en) 2012-01-19
RU2012102925A (en) 2013-08-10
SI2448920T1 (en) 2014-12-31
EP2448920B1 (en) 2014-08-13
DK2448920T3 (en) 2014-09-29
WO2011001089A1 (en) 2011-01-06
CN102471260A (en) 2012-05-23
US20160280650A1 (en) 2016-09-29
US20140107129A1 (en) 2014-04-17
FR2947268B1 (en) 2011-08-26
US20150158834A1 (en) 2015-06-11
US9365529B2 (en) 2016-06-14
AU2010267872C1 (en) 2014-04-10
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EP2448920A1 (en) 2012-05-09
US20130172363A1 (en) 2013-07-04
US8420632B2 (en) 2013-04-16
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