IL99166A - History 3-) 1,3-Benziazoxazole-3-Il-4-pyridiamine, their preparation and pharmaceutical preparations containing them - Google Patents

History 3-) 1,3-Benziazoxazole-3-Il-4-pyridiamine, their preparation and pharmaceutical preparations containing them

Info

Publication number
IL99166A
IL99166A IL9916691A IL9916691A IL99166A IL 99166 A IL99166 A IL 99166A IL 9916691 A IL9916691 A IL 9916691A IL 9916691 A IL9916691 A IL 9916691A IL 99166 A IL99166 A IL 99166A
Authority
IL
Israel
Prior art keywords
compound
hydrogen
benzisoxazol
loweralkyl
arylalkyl
Prior art date
Application number
IL9916691A
Other languages
English (en)
Hebrew (he)
Other versions
IL99166A0 (en
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of IL99166A0 publication Critical patent/IL99166A0/xx
Publication of IL99166A publication Critical patent/IL99166A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
IL9916691A 1990-08-13 1991-08-12 History 3-) 1,3-Benziazoxazole-3-Il-4-pyridiamine, their preparation and pharmaceutical preparations containing them IL99166A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/566,932 US5055476A (en) 1990-08-13 1990-08-13 3-(1,2-benzisoxazol-3-yl)-4-pyridinamines and derivatives

Publications (2)

Publication Number Publication Date
IL99166A0 IL99166A0 (en) 1992-07-15
IL99166A true IL99166A (en) 1995-12-08

Family

ID=24265033

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9916691A IL99166A (en) 1990-08-13 1991-08-12 History 3-) 1,3-Benziazoxazole-3-Il-4-pyridiamine, their preparation and pharmaceutical preparations containing them

Country Status (24)

Country Link
US (1) US5055476A (fr)
EP (1) EP0471297B1 (fr)
JP (1) JP3057829B2 (fr)
KR (1) KR100191386B1 (fr)
AT (1) ATE130004T1 (fr)
AU (1) AU633791B2 (fr)
CA (1) CA2048959C (fr)
CZ (1) CZ280568B6 (fr)
DE (1) DE69114405T2 (fr)
DK (1) DK0471297T3 (fr)
ES (1) ES2079531T3 (fr)
FI (1) FI103970B (fr)
GR (1) GR3018184T3 (fr)
HU (1) HU213201B (fr)
IE (1) IE70597B1 (fr)
IL (1) IL99166A (fr)
MX (1) MX9100639A (fr)
NO (1) NO179519C (fr)
NZ (1) NZ239326A (fr)
PT (1) PT98645B (fr)
RU (1) RU2012561C1 (fr)
TW (1) TW202446B (fr)
YU (1) YU140991A (fr)
ZA (1) ZA916342B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5308826A (en) * 1993-04-22 1994-05-03 Zeneca Limited Herbicidal 4-substituted pyridyl-3-carbinols
US5595958A (en) * 1994-05-02 1997-01-21 Zeneca Limited 3-substituted pyridine compounds and derivatives thereof
AU2313995A (en) * 1994-05-02 1995-11-29 Zeneca Limited Herbicidal hydroxybenzyl-substituted heteroaryl compounds and derivatives thereof
KR20140007954A (ko) 2011-06-10 2014-01-20 메르크 파텐트 게엠베하 Btk 억제 활성을 갖는 피리미딘 및 피리딘 화합물의 조성물 및 제조방법
RU2626650C2 (ru) * 2015-08-31 2017-07-31 Федеральное государственное бюджетное образовательное учреждение высшего образования "Пермский государственный национальный исследовательский университет" 2-Арил-2,4-дигидрокси-2,5-дигидро-3-гетерил-5-оксо-1Н-пиррол-1-ил-4-метилбелзолсульфаниламиды, обладающие анальгетической активностью
EP4429465A1 (fr) 2021-11-10 2024-09-18 Symrise AG Compositions comprenant des agents de refroidissement agonistes de trpm8

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4355037A (en) * 1981-11-12 1982-10-19 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidyl)-1,2-benzisoxales
IL66866A (en) * 1982-04-09 1987-08-31 Hoechst Roussel Pharma 1-(3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl)-4-(substituted)-piperazines and-piperidines,a process for the preparation thereof,and pharmaceutical compositions containing them
CA1335289C (fr) * 1987-10-26 1995-04-18 Fujio Antoku Derives piperidinylbenzisoxazole, leur production et leur utilisation pharmaceutique
MY107955A (en) * 1990-07-27 1996-07-15 Ici Plc Fungicides.

Also Published As

Publication number Publication date
FI913800A (fi) 1992-02-14
KR100191386B1 (ko) 1999-06-15
RU2012561C1 (ru) 1994-05-15
FI103970B1 (fi) 1999-10-29
KR920004383A (ko) 1992-03-27
HU213201B (en) 1997-03-28
ES2079531T3 (es) 1996-01-16
DE69114405D1 (de) 1995-12-14
EP0471297A1 (fr) 1992-02-19
DK0471297T3 (da) 1996-03-04
JPH05112562A (ja) 1993-05-07
JP3057829B2 (ja) 2000-07-04
CA2048959A1 (fr) 1992-02-14
GR3018184T3 (en) 1996-02-29
PT98645B (pt) 1999-01-29
IL99166A0 (en) 1992-07-15
NO179519B (no) 1996-07-15
EP0471297B1 (fr) 1995-11-08
HUT61755A (en) 1993-03-01
TW202446B (fr) 1993-03-21
YU140991A (sh) 1995-01-31
AU633791B2 (en) 1993-02-04
DE69114405T2 (de) 1996-05-02
US5055476A (en) 1991-10-08
CZ280568B6 (cs) 1996-02-14
ATE130004T1 (de) 1995-11-15
NZ239326A (en) 1994-04-27
NO913142L (no) 1992-02-14
FI103970B (fi) 1999-10-29
HU912673D0 (en) 1992-01-28
CA2048959C (fr) 2003-07-29
CS248991A3 (en) 1992-03-18
MX9100639A (es) 1992-04-01
IE70597B1 (en) 1996-12-11
FI913800A0 (fi) 1991-08-09
NO913142D0 (no) 1991-08-12
NO179519C (no) 1996-10-23
AU8176591A (en) 1992-02-20
IE912851A1 (en) 1992-02-26
ZA916342B (en) 1992-04-29
PT98645A (pt) 1992-06-30

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Legal Events

Date Code Title Description
FF Patent granted
HC Change of name of proprietor(s)
KB Patent renewed
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees